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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5378 products of "GPCR/G-Protein"

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  • Picotamide

    CAS:
    <p>Picotamide has anticoagulant and fibrinolytic properties.</p>
    Formula:C21H20N4O3
    Purity:98.90%
    Color and Shape:Solid
    Molecular weight:376.41
  • Bevantolol

    CAS:
    <p>Bevantolol, a selective β-1 adrenoceptor antagonist, is utilized for the investigation of angina pectoris and hypertension [1].</p>
    Formula:C20H27NO4
    Color and Shape:Solid
    Molecular weight:345.43
  • Lodoxamide

    CAS:
    <p>Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.</p>
    Formula:C11H6ClN3O6
    Purity:99.13% - 99.81%
    Color and Shape:Solid
    Molecular weight:311.63
  • NPS ALX Compound 4a

    CAS:
    NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)
    Formula:C25H25N3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.55
  • Carbazochrome

    CAS:
    <p>Carbazochrome (Adchnon) is an antihemorrhagic that promotes platelet aggregation to stop bleeding, possibly for surgeries and hemorrhoids treatment.</p>
    Formula:C10H12N4O3
    Purity:98.36%
    Color and Shape:Nacarat Crystalline Powder
    Molecular weight:236.23
  • Quipazine maleate

    CAS:
    <p>Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.</p>
    Formula:C17H19N3O4
    Color and Shape:Solid
    Molecular weight:329.36
  • Volinanserin

    CAS:
    Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.
    Formula:C22H28FNO3
    Purity:98.94% - 99.95%
    Color and Shape:Solid
    Molecular weight:373.46
  • Enprofylline

    CAS:
    <p>Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.</p>
    Formula:C8H10N4O2
    Purity:98.37%
    Color and Shape:Solid
    Molecular weight:194.19
  • Rimcazole dihydrochloride

    CAS:
    <p>Rimcazole dihydrochloride: a σ receptor antagonist, hydrochloride salt, blocks dopamine uptake.</p>
    Formula:C21H28ClN3
    Purity:99.63%
    Color and Shape:Solid
    Molecular weight:357.92
  • Tavapadon

    CAS:
    <p>Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.</p>
    Formula:C19H16F3N3O3
    Purity:99.33% - 99.8%
    Color and Shape:Solid
    Molecular weight:391.34
  • Piboserod hydrochloride

    CAS:
    <p>Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.</p>
    Formula:C22H32ClN3O2
    Color and Shape:Solid
    Molecular weight:405.96
  • YIL781 hydrochloride

    CAS:
    <p>YIL781 is a ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM) with no significant affinity for the motilin receptor (Ki = 6 μM).</p>
    Formula:C24H29ClFN3O2
    Color and Shape:Solid
    Molecular weight:445.96
  • Cyclopiazonic acid

    CAS:
    <p>Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.</p>
    Formula:C20H20N2O3
    Purity:99.27% - 99.80%
    Color and Shape:Solid
    Molecular weight:336.38
  • ML-193

    CAS:
    ML-193: GPR55 antagonist, IC50 221nM, 27x selective over GPR35/CB1/CB2, may aid Parkinson's symptoms.
    Formula:C28H25N5O4S
    Purity:97.74%
    Color and Shape:Solid
    Molecular weight:527.59
  • Fertirelin

    CAS:
    <p>Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist (GnRH agonist).</p>
    Formula:C55H76N16O12
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1153.29
  • Bretylium tosylate

    CAS:
    <p>Bretylium tosylate is an inhibitor of the presynaptic release of vasoconstrictor neurotransmitters, a available antiarrhythmic drug for ventricular arrhythmias.</p>
    Formula:C18H24BrNO3S
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:414.36
  • MK 571

    CAS:
    <p>MK 571 (L660711) is an orally active antagonist of CysLT1 receptor.</p>
    Formula:C26H27ClN2O3S2
    Purity:98.69% - 99.65%
    Color and Shape:Solid
    Molecular weight:515.09
  • Trimethobenzamide hydrochloride

    CAS:
    <p>Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.</p>
    Formula:C21H29ClN2O5
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:424.92
  • CRF (6-33) acetate(120066-38-8 free base)


    <p>CRFBP inhibitor peptide; reduces weight gain, boosts activity in obese rats.</p>
    Formula:C143H235N41O45S
    Purity:97.12%
    Color and Shape:Solid
    Molecular weight:3280.76
  • Benzotript

    CAS:
    <p>Benzotript is an gastrin-receptor antagonist, with anti-gastrinic.</p>
    Formula:C18H15ClN2O3
    Purity:97.82%
    Color and Shape:Solid
    Molecular weight:342.776