
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(942 products)
- Adenosine Receptor(242 products)
- Adrenergic Receptor(2,949 products)
- Bombesin Receptor(30 products)
- Bradykinin Receptor(59 products)
- CXCR(149 products)
- CaSR(32 products)
- Cannabinoid Receptor(195 products)
- Dopamine Receptor(410 products)
- Endothelin Receptor(75 products)
- GNRH Receptor(73 products)
- GPCR19(31 products)
- GRK(32 products)
- GTPase(21 products)
- Glucagon Receptor(166 products)
- Hedgehog/Smoothened(45 products)
- Histamine Receptor(359 products)
- LPA Receptor(21 products)
- Melatonin Receptor(24 products)
- OX Receptor(40 products)
- Opioid Receptor(298 products)
- PAFR(11 products)
- PKA(49 products)
- S1P Receptor(17 products)
- SGLT(30 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5378 products of "GPCR/G-Protein"
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Picotamide
CAS:<p>Picotamide has anticoagulant and fibrinolytic properties.</p>Formula:C21H20N4O3Purity:98.90%Color and Shape:SolidMolecular weight:376.41Bevantolol
CAS:<p>Bevantolol, a selective β-1 adrenoceptor antagonist, is utilized for the investigation of angina pectoris and hypertension [1].</p>Formula:C20H27NO4Color and Shape:SolidMolecular weight:345.43Lodoxamide
CAS:<p>Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.</p>Formula:C11H6ClN3O6Purity:99.13% - 99.81%Color and Shape:SolidMolecular weight:311.63NPS ALX Compound 4a
CAS:NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)Formula:C25H25N3O2SPurity:98%Color and Shape:SolidMolecular weight:431.55Carbazochrome
CAS:<p>Carbazochrome (Adchnon) is an antihemorrhagic that promotes platelet aggregation to stop bleeding, possibly for surgeries and hemorrhoids treatment.</p>Formula:C10H12N4O3Purity:98.36%Color and Shape:Nacarat Crystalline PowderMolecular weight:236.23Quipazine maleate
CAS:<p>Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.</p>Formula:C17H19N3O4Color and Shape:SolidMolecular weight:329.36Volinanserin
CAS:Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.Formula:C22H28FNO3Purity:98.94% - 99.95%Color and Shape:SolidMolecular weight:373.46Enprofylline
CAS:<p>Enprofylline (Enprofilina), a bronchodilator, acts primarily as a competitive nonselective phosphodiesterase inhibitor.</p>Formula:C8H10N4O2Purity:98.37%Color and Shape:SolidMolecular weight:194.19Rimcazole dihydrochloride
CAS:<p>Rimcazole dihydrochloride: a σ receptor antagonist, hydrochloride salt, blocks dopamine uptake.</p>Formula:C21H28ClN3Purity:99.63%Color and Shape:SolidMolecular weight:357.92Tavapadon
CAS:<p>Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.</p>Formula:C19H16F3N3O3Purity:99.33% - 99.8%Color and Shape:SolidMolecular weight:391.34Piboserod hydrochloride
CAS:<p>Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.</p>Formula:C22H32ClN3O2Color and Shape:SolidMolecular weight:405.96YIL781 hydrochloride
CAS:<p>YIL781 is a ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM) with no significant affinity for the motilin receptor (Ki = 6 μM).</p>Formula:C24H29ClFN3O2Color and Shape:SolidMolecular weight:445.96Cyclopiazonic acid
CAS:<p>Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.</p>Formula:C20H20N2O3Purity:99.27% - 99.80%Color and Shape:SolidMolecular weight:336.38ML-193
CAS:ML-193: GPR55 antagonist, IC50 221nM, 27x selective over GPR35/CB1/CB2, may aid Parkinson's symptoms.Formula:C28H25N5O4SPurity:97.74%Color and Shape:SolidMolecular weight:527.59Fertirelin
CAS:<p>Fertirelin, or fertirelin acetate, sold under the brand name Ovalyse, is a gonadotropin-releasing hormone agonist (GnRH agonist).</p>Formula:C55H76N16O12Purity:>99.99%Color and Shape:SolidMolecular weight:1153.29Bretylium tosylate
CAS:<p>Bretylium tosylate is an inhibitor of the presynaptic release of vasoconstrictor neurotransmitters, a available antiarrhythmic drug for ventricular arrhythmias.</p>Formula:C18H24BrNO3SPurity:>99.99%Color and Shape:SolidMolecular weight:414.36MK 571
CAS:<p>MK 571 (L660711) is an orally active antagonist of CysLT1 receptor.</p>Formula:C26H27ClN2O3S2Purity:98.69% - 99.65%Color and Shape:SolidMolecular weight:515.09Trimethobenzamide hydrochloride
CAS:<p>Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.</p>Formula:C21H29ClN2O5Purity:99.52%Color and Shape:SolidMolecular weight:424.92CRF (6-33) acetate(120066-38-8 free base)
<p>CRFBP inhibitor peptide; reduces weight gain, boosts activity in obese rats.</p>Formula:C143H235N41O45SPurity:97.12%Color and Shape:SolidMolecular weight:3280.76Benzotript
CAS:<p>Benzotript is an gastrin-receptor antagonist, with anti-gastrinic.</p>Formula:C18H15ClN2O3Purity:97.82%Color and Shape:SolidMolecular weight:342.776
