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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5838 products of "GPCR/G-Protein"

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  • PNU-282987
    Targetmol
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    PNU-282987

    CAS:
    PNU-282987 is a selective α7 nicotinic acetylcholine receptor(α7 nAChR) agonist with Ki of 26 nM; no affinity for α1β1γδ and α3β4 nAChRs (IC50 ≥ 60 μM).
    Formula:C14H18Cl2N2O
    Purity:99% - >99.99%
    Color and Shape:Solid
    Molecular weight:301.21

    Ref: TM-T2422

  • Liraglutide
    Targetmol
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    Liraglutide

    CAS:
    <p>Liraglutide (Liraglutida) is a synthetic analog of GLP-1, an agonist of the GLP-1 receptor. Liraglutide is an antidiabetic agent. Cost effective and quality assured.</p>
    Formula:C172H265N43O51
    Purity:97.65% - 99.04%
    Color and Shape:Solid
    Molecular weight:3751.25

    Ref: TM-T6876

  • AZD1283
    Targetmol
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    AZD1283

    CAS:
    AZD1283 is an effective P2Y12 receptor antagonist (EC50: 3.0 ug/kg/min, binding IC50: 11 nM).
    Formula:C23H26N4O5S
    Purity:98.37% - 99.63%
    Color and Shape:Solid
    Molecular weight:470.54

    Ref: TM-T3536

  • Nonapeptide-1 acetate salt (158563-45-2 free base)
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    Nonapeptide-1 acetate salt (158563-45-2 free base)

    <p>Nonapeptide-1 acetate salt (158563-45-2 free base) (Melanostatine-5 acetate salt) , a peptide hormone, is a potent α-Melanocyte-stimulating hormone (α-MSH)</p>
    Formula:C63H91N15O11S
    Purity:98.26%
    Color and Shape:Solid
    Molecular weight:1266.58

    Ref: TM-TP1101

  • [Des-Arg9]-Bradykinin TFA
    Targetmol
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    [Des-Arg9]-Bradykinin TFA

    CAS:
    [Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.
    Formula:C46H62F3N11O12
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1018.05

    Ref: TM-T8809

  • Vortioxetine
    Targetmol
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    Vortioxetine

    CAS:
    Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.
    Formula:C18H22N2S
    Purity:99.34% - 99.34%
    Color and Shape:Solid
    Molecular weight:298.45

    Ref: TM-T2395

  • Ocaperidone
    Targetmol
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    Ocaperidone

    CAS:
    Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.
    Formula:C24H25FN4O2
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:420.48

    Ref: TM-T3497

  • Mini Gastrin I, human acetate
    Targetmol
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    Mini Gastrin I, human acetate

    Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino acids 5-17 of the parent peptide.
    Formula:C76H103N15O28S
    Purity:99.35% - 99.82%
    Color and Shape:Solid
    Molecular weight:1706.78

    Ref: TM-TP1821L

  • Talnetant hydrochloride
    Targetmol
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    Talnetant hydrochloride

    CAS:
    Talnetant (SB 223412) hydrochloride, an NK3 antagonist, selectively binds hNK-3 at 1.4 nM, much less to hNK-2, none to hNK-1 at 100 μM.
    Formula:C25H23ClN2O2
    Color and Shape:Solid
    Molecular weight:418.92

    Ref: TM-T62199

  • Dioxopromethazine
    Targetmol
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    Dioxopromethazine

    CAS:
    Dioxopromethazine (Dioxoprothazine) is a drug for the treatment of a cough and expectoration. It also can be used in local anesthesia.
    Formula:C17H20N2O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:316.42

    Ref: TM-T3609

  • PD 117519
    Targetmol
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    PD 117519

    CAS:
    PD 117519 (CI947) is an agonist of adenosine receptor
    Formula:C19H21N5O4
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:383.4

    Ref: TM-T7509

  • Decynium 22
    Targetmol
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    Decynium 22

    CAS:
    Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitor
    Formula:C23H23IN2
    Purity:99.92%
    Color and Shape:Dark Red Crystals
    Molecular weight:454.35

    Ref: TM-T22714

  • Cimetidine hydrochloride
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    Cimetidine hydrochloride

    CAS:
    Cimetidine (SKF-92334) is an oral H2 blocker with Ki 0.6 μM, anti-cancer and anti-inflammatory properties, used for ulcer research.
    Formula:C10H17ClN6S
    Color and Shape:Solid
    Molecular weight:288.8

    Ref: TM-T60584

  • SSR240612
    Targetmol
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    SSR240612

    CAS:
    SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,
    Formula:C42H53ClN4O7S
    Purity:98.59% - 99.16%
    Color and Shape:Solid
    Molecular weight:793.41

    Ref: TM-T5048

  • Montelukast dicyclohexylamine
    Targetmol
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    Montelukast dicyclohexylamine

    CAS:
    Montelukast (MK0476), a selective CysLT1 antagonist, treats asthma, liver injury, and is researched for COVID-19.
    Formula:C47H59ClN2O3S
    Color and Shape:Solid
    Molecular weight:767.5

    Ref: TM-T72145

  • GSK189254A
    Targetmol
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    GSK189254A

    CAS:
    <p>GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).</p>
    Formula:C21H25N3O2
    Purity:98.71% - 99.858%
    Color and Shape:Solid
    Molecular weight:351.44

    Ref: TM-TQ0066

  • [Sar9,Met(O2)11]-Substance P
    Targetmol
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    [Sar9,Met(O2)11]-Substance P

    CAS:
    [Sar9,Met(O2)11]-Substance P (NA) is an agonist of NK1 receptor.
    Formula:C64H100N18O15S
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1393.66

    Ref: TM-T7828

  • Takeda103A
    Targetmol
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    Takeda103A

    CAS:
    <p>Takeda103A (CMPD103A) is the GRK2-dependent bovine tubulin oxidation effective inhibitor.</p>
    Formula:C24H23F2N7O
    Purity:97.17%
    Color and Shape:Solid
    Molecular weight:463.48

    Ref: TM-T24850

  • Ozagrel hydrochloride
    Targetmol
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    Ozagrel hydrochloride

    CAS:
    <p>Ozagrel hydrochloride (OKY-046 HCl) is a selective thromboxane A(2) synthetase inhibitor used for the improvement of postoperative cerebrovascular contraction</p>
    Formula:C13H12N2O2·HCl
    Purity:99.80%
    Color and Shape:White Or Off White Crystalline Powder
    Molecular weight:264.71

    Ref: TM-T6625

  • 2-Methoxyidazoxan monohydrochloride
    Targetmol
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    2-Methoxyidazoxan monohydrochloride

    CAS:
    L-Albizziin (2-Methoxyidazoxan monohydrochloride) is a highly potent selective antagonist of the alpha 2r adrenergic receptor.
    Formula:C12H14N2O3·HCl
    Purity:98.99%
    Color and Shape:Solid
    Molecular weight:270.72

    Ref: TM-T23283