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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5982 products of "GPCR/G-Protein"

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  • nifenalol.HCl

    CAS:
    Nifenalol.HCl(INPEA) is a antagonist of β-adrenergic receptor.
    Formula:C11H17ClN2O3
    Purity:99.96%
    Color and Shape:Solid
    Molecular weight:260.72

    Ref: TM-T8663

    25mg
    42.00€
    50mg
    63.00€
    1mL*10mM (DMSO)
    33.00€
  • GW627368

    CAS:
    GW627368 (GW 627368X)X is a novel, potent and selective antagonist of prostanoid EP4 receptor.
    Formula:C30H28N2O6S
    Purity:99.75% - 99.92%
    Color and Shape:Solid
    Molecular weight:544.62

    Ref: TM-T1978

    2mg
    34.00€
    5mg
    50.00€
    10mg
    82.00€
    25mg
    124.00€
    50mg
    203.00€
    100mg
    358.00€
    1mL*10mM (DMSO)
    60.00€
  • Flibanserin

    CAS:

    Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.

    Formula:C20H21F3N4O
    Purity:99.37% - 99.93%
    Color and Shape:White Powder
    Molecular weight:390.4

    Ref: TM-T4297

    5mg
    40.00€
    10mg
    65.00€
    25mg
    107.00€
    50mg
    187.00€
    100mg
    243.00€
    200mg
    359.00€
  • 1-Oleoyl lysophosphatidic acid sodium

    CAS:
    1-Oleoyl lysophosphatidic acid sodium (1-Oleoyl lysophosphatidic acid sodium salt) salt is an Endogenous agonist of LPA1 and LPA2
    Formula:C21H40O7P·Na
    Purity:98.75% - 99.24%
    Color and Shape:Solid
    Molecular weight:458.51

    Ref: TM-T21654

    1mg
    40.00€
    2mg
    52.00€
    5mg
    85.00€
    10mg
    137.00€
    25mg
    283.00€
    50mg
    494.00€
    100mg
    727.00€
    200mg
    1,017.00€
  • BAY 41-2272

    CAS:
    BAY 41-2272 is a direct and NO-independent soluble guanylate cyclase (sGC) stimulator.
    Formula:C20H17FN6
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:360.39

    Ref: TM-T6775

    2mg
    34.00€
    5mg
    50.00€
    10mg
    82.00€
    25mg
    160.00€
    50mg
    246.00€
    100mg
    355.00€
    1mL*10mM (DMSO)
    50.00€
  • SB-200646

    CAS:
    SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptor
    Formula:C15H14N4O
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:266.3

    Ref: TM-T8357

    1mg
    62.00€
    5mg
    122.00€
    10mg
    177.00€
    25mg
    299.00€
    50mg
    430.00€
    100mg
    587.00€
    1mL*10mM (DMSO)
    128.00€
  • Decloxizine dihydrochloride

    CAS:

    Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.

    Formula:C21H28N2O2·2ClH
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:413.39

    Ref: TM-T5495

    25mg
    50.00€
    50mg
    74.00€
    100mg
    97.00€
    200mg
    160.00€
  • ML221

    CAS:
    ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in
    Formula:C17H11N3O6S
    Purity:97.74%
    Color and Shape:Solid
    Molecular weight:385.35

    Ref: TM-T4390

    2mg
    To inquire
    5mg
    52.00€
    10mg
    85.00€
    25mg
    144.00€
    50mg
    227.00€
    100mg
    369.00€
    200mg
    To inquire
    1mL*10mM (DMSO)
    55.00€
  • Piperacetazine

    CAS:
    Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.
    Formula:C24H30N2O2S
    Purity:99.9% - 99.92%
    Color and Shape:Solid
    Molecular weight:410.57

    Ref: TM-T3085

    2mg
    42.00€
    5mg
    62.00€
    10mg
    86.00€
    25mg
    130.00€
    50mg
    187.00€
    100mg
    283.00€
    1mL*10mM (DMSO)
    67.00€
  • Relugolix

    CAS:
    Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, with
    Formula:C29H27F2N7O5S
    Purity:98.64% - 99.97%
    Color and Shape:Solid
    Molecular weight:623.63

    Ref: TM-T3630

    2mg
    39.00€
    5mg
    58.00€
    10mg
    93.00€
    25mg
    167.00€
    50mg
    250.00€
    100mg
    408.00€
    200mg
    585.00€
    1mL*10mM (DMSO)
    81.00€
  • Obestatin (rat) acetate


    Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).
    Formula:C114H174N34O31
    Purity:99.05%
    Color and Shape:Solid
    Molecular weight:2516.81

    Ref: TM-TP2279L

    1mg
    77.00€
    2mg
    97.00€
    5mg
    156.00€
    10mg
    225.00€
    25mg
    375.00€
    50mg
    535.00€
    100mg
    730.00€
    200mg
    938.00€
  • Spexin acetate(1370290-58-6 free base)


    Spexin acetate: GAL2/GAL3 agonist. EC50: 45.7/112.2 nM. Inactive at GAL1. Reduces appetite, fat uptake, and food intake; lowers LH in fish; anxiolytic.
    Formula:C76H117N19O22S
    Purity:95.43%
    Color and Shape:Solid
    Molecular weight:1680.94

    Ref: TM-TP1930L1

    1mg
    114.00€
    5mg
    255.00€
    10mg
    375.00€
    25mg
    562.00€
    50mg
    787.00€
    100mg
    1,074.00€
    200mg
    1,444.00€
  • Opiranserin hydrochloride

    CAS:
    Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM
    Formula:C21H35ClN2O5
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:430.97

    Ref: TM-T9833

    1mg
    90.00€
    5mg
    215.00€
    10mg
    340.00€
    25mg
    618.00€
    50mg
    879.00€
    100mg
    1,224.00€
    500mg
    2,457.00€
    1mL*10mM (DMSO)
    236.00€
  • AC-90179 HCl

    CAS:
    AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.
    Formula:C23H31ClN2O2
    Purity:99.71%
    Color and Shape:Solid
    Molecular weight:402.96

    Ref: TM-T26543

    1mg
    35.00€
    5mg
    64.00€
    10mg
    90.00€
    25mg
    134.00€
    50mg
    235.00€
    100mg
    349.00€
    1mL*10mM (DMSO)
    85.00€
  • Melanotan (MT)-II

    CAS:
    Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone α-melanocyte-stimulating hormone (α-MSH).
    Formula:C50H69N15O9
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1024.18

    Ref: TM-TP1324

    1mg
    34.00€
    2mg
    46.00€
    5mg
    66.00€
    10mg
    88.00€
    25mg
    152.00€
    50mg
    236.00€
    100mg
    385.00€
    200mg
    560.00€
  • FAUC-365

    CAS:
    FAUC-365 is a D3 dopamine receptor agonist.
    Formula:C23H25Cl2N3OS
    Purity:99.62%
    Color and Shape:Solid
    Molecular weight:462.44

    Ref: TM-T21667

    1mg
    52.00€
    5mg
    111.00€
    10mg
    169.00€
    25mg
    323.00€
    50mg
    512.00€
    100mg
    740.00€
    500mg
    1,539.00€
    1mL*10mM (DMSO)
    123.00€
  • AVN-492

    CAS:
    AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).
    Formula:C17H21N5O2S
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:359.45

    Ref: TM-T5179

    1mg
    37.00€
    2mg
    50.00€
    5mg
    77.00€
    10mg
    114.00€
    25mg
    225.00€
    50mg
    335.00€
    100mg
    484.00€
    1mL*10mM (DMSO)
    85.00€
  • Vorapaxar sulfate

    CAS:
    Vorapaxar sulfate (Zontivity) is a potent and orally active thrombin receptor (PAR-1) antagonist.
    Formula:C29H35FN2O8S
    Purity:99.9% - >99.99%
    Color and Shape:Solid
    Molecular weight:590.66

    Ref: TM-T3098

    1mg
    38.00€
    2mg
    49.00€
    5mg
    79.00€
    10mg
    119.00€
    25mg
    210.00€
    50mg
    354.00€
    100mg
    528.00€
    500mg
    1,159.00€
    1mL*10mM (DMSO)
    99.00€
  • Tozadenant

    CAS:
    Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)
    Formula:C19H26N4O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:406.5

    Ref: TM-T7320

    5mg
    44.00€
    10mg
    67.00€
    25mg
    113.00€
    50mg
    190.00€
    100mg
    274.00€
    200mg
    394.00€
    1mL*10mM (DMSO)
    48.00€
  • Vipadenant

    CAS:
    Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).
    Formula:C16H15N7O
    Purity:97.25% - 97.36%
    Color and Shape:Solid
    Molecular weight:321.34

    Ref: TM-T2373

    2mg
    35.00€
    5mg
    51.00€
    10mg
    80.00€
    25mg
    131.00€
    50mg
    210.00€
    100mg
    313.00€
    200mg
    445.00€
    1mL*10mM (DMSO)
    215.00€