
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(58 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5982 products of "GPCR/G-Protein"
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nifenalol.HCl
CAS:Nifenalol.HCl(INPEA) is a antagonist of β-adrenergic receptor.Formula:C11H17ClN2O3Purity:99.96%Color and Shape:SolidMolecular weight:260.72GW627368
CAS:GW627368 (GW 627368X)X is a novel, potent and selective antagonist of prostanoid EP4 receptor.Formula:C30H28N2O6SPurity:99.75% - 99.92%Color and Shape:SolidMolecular weight:544.62Flibanserin
CAS:Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.
Formula:C20H21F3N4OPurity:99.37% - 99.93%Color and Shape:White PowderMolecular weight:390.41-Oleoyl lysophosphatidic acid sodium
CAS:1-Oleoyl lysophosphatidic acid sodium (1-Oleoyl lysophosphatidic acid sodium salt) salt is an Endogenous agonist of LPA1 and LPA2Formula:C21H40O7P·NaPurity:98.75% - 99.24%Color and Shape:SolidMolecular weight:458.51Ref: TM-T21654
1mg40.00€2mg52.00€5mg85.00€10mg137.00€25mg283.00€50mg494.00€100mg727.00€200mg1,017.00€BAY 41-2272
CAS:BAY 41-2272 is a direct and NO-independent soluble guanylate cyclase (sGC) stimulator.Formula:C20H17FN6Purity:99.54%Color and Shape:SolidMolecular weight:360.39SB-200646
CAS:SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptorFormula:C15H14N4OPurity:99.61%Color and Shape:SolidMolecular weight:266.3Decloxizine dihydrochloride
CAS:Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.
Formula:C21H28N2O2·2ClHPurity:99.73%Color and Shape:SolidMolecular weight:413.39ML221
CAS:ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM inFormula:C17H11N3O6SPurity:97.74%Color and Shape:SolidMolecular weight:385.35Ref: TM-T4390
2mgTo inquire5mg52.00€10mg85.00€25mg144.00€50mg227.00€100mg369.00€200mgTo inquire1mL*10mM (DMSO)55.00€Piperacetazine
CAS:Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.Formula:C24H30N2O2SPurity:99.9% - 99.92%Color and Shape:SolidMolecular weight:410.57Relugolix
CAS:Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFormula:C29H27F2N7O5SPurity:98.64% - 99.97%Color and Shape:SolidMolecular weight:623.63Ref: TM-T3630
2mg39.00€5mg58.00€10mg93.00€25mg167.00€50mg250.00€100mg408.00€200mg585.00€1mL*10mM (DMSO)81.00€Obestatin (rat) acetate
Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).Formula:C114H174N34O31Purity:99.05%Color and Shape:SolidMolecular weight:2516.81Ref: TM-TP2279L
1mg77.00€2mg97.00€5mg156.00€10mg225.00€25mg375.00€50mg535.00€100mg730.00€200mg938.00€Spexin acetate(1370290-58-6 free base)
Spexin acetate: GAL2/GAL3 agonist. EC50: 45.7/112.2 nM. Inactive at GAL1. Reduces appetite, fat uptake, and food intake; lowers LH in fish; anxiolytic.Formula:C76H117N19O22SPurity:95.43%Color and Shape:SolidMolecular weight:1680.94Opiranserin hydrochloride
CAS:Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μMFormula:C21H35ClN2O5Purity:99.33%Color and Shape:SolidMolecular weight:430.97Ref: TM-T9833
1mg90.00€5mg215.00€10mg340.00€25mg618.00€50mg879.00€100mg1,224.00€500mg2,457.00€1mL*10mM (DMSO)236.00€AC-90179 HCl
CAS:AC-90179 HCl: selective 5-HT2A inverse agonist, atypical antipsychotic, reduces hallucinogen-induced vasoconstriction.Formula:C23H31ClN2O2Purity:99.71%Color and Shape:SolidMolecular weight:402.96Melanotan (MT)-II
CAS:Melanotan (MT)-II, a synthetic melanocortin receptor agonist, is a synthetic analogue of the peptide hormone α-melanocyte-stimulating hormone (α-MSH).Formula:C50H69N15O9Purity:>99.99%Color and Shape:SolidMolecular weight:1024.18FAUC-365
CAS:FAUC-365 is a D3 dopamine receptor agonist.Formula:C23H25Cl2N3OSPurity:99.62%Color and Shape:SolidMolecular weight:462.44Ref: TM-T21667
1mg52.00€5mg111.00€10mg169.00€25mg323.00€50mg512.00€100mg740.00€500mg1,539.00€1mL*10mM (DMSO)123.00€AVN-492
CAS:AVN-49 is a potent and selective 5-HT6R Antagonist (Ki: 91 pM).Formula:C17H21N5O2SPurity:99.81%Color and Shape:SolidMolecular weight:359.45Ref: TM-T5179
1mg37.00€2mg50.00€5mg77.00€10mg114.00€25mg225.00€50mg335.00€100mg484.00€1mL*10mM (DMSO)85.00€Vorapaxar sulfate
CAS:Vorapaxar sulfate (Zontivity) is a potent and orally active thrombin receptor (PAR-1) antagonist.Formula:C29H35FN2O8SPurity:99.9% - >99.99%Color and Shape:SolidMolecular weight:590.66Ref: TM-T3098
1mg38.00€2mg49.00€5mg79.00€10mg119.00€25mg210.00€50mg354.00€100mg528.00€500mg1,159.00€1mL*10mM (DMSO)99.00€Tozadenant
CAS:Tozadenant (SYN115) is an adenosine A2A receptor antagonist(Ki of 11.5 nM and 6 nM on human and rhesus,respectively)Formula:C19H26N4O4SPurity:98%Color and Shape:SolidMolecular weight:406.5Vipadenant
CAS:Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).Formula:C16H15N7OPurity:97.25% - 97.36%Color and Shape:SolidMolecular weight:321.34Ref: TM-T2373
2mg35.00€5mg51.00€10mg80.00€25mg131.00€50mg210.00€100mg313.00€200mg445.00€1mL*10mM (DMSO)215.00€
