GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(55 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5985 products of "GPCR/G-Protein"
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Poloxamer 407
CAS:Poloxamer 407 is a nonionic surfactant.Purity:98%Color and Shape:White Crystalline PowderMolecular weight:12000 (Average)Zacopride hydrochloride
CAS:Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.Formula:C15H20ClN3O2·HClPurity:98.32%Color and Shape:SolidMolecular weight:346.26Ref: TM-T5336
1mg34.00€5mg71.00€10mg99.00€25mg212.00€50mg385.00€100mg618.00€200mg859.00€1mL*10mM (DMSO)79.00€Decynium 22
CAS:Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitorFormula:C23H23IN2Purity:99.92%Color and Shape:Dark Red CrystalsMolecular weight:454.35PGS-IN-1
CAS:PGS-IN-1 (KME-4) is a potent inhibitor of prostaglandin synthetase (PGS, IC50: 0.28 μM) and 5-lipoxygenase (IC50: 1.05 μM).Formula:C19H26O3Purity:99.39%Color and Shape:SolidMolecular weight:302.41Ref: TM-T10098
1mg52.00€5mg97.00€10mg170.00€25mg369.00€50mg540.00€100mg772.00€200mg1,035.00€1mL*10mM (DMSO)110.00€Maropitant
CAS:Maropitant is a selective neurokinin (NK1) receptor antagonist.Formula:C32H40N2OPurity:97.35% - 99.75%Color and Shape:SolidMolecular weight:468.67Ref: TM-T7209
5mg50.00€10mg80.00€25mg116.00€50mg212.00€100mg316.00€200mg454.00€1mL*10mM (DMSO)To inquirePF-4136309
CAS:PF-4136309 (INCB8761) is a specific, effective, and orally bioavailable CCR2 antagonist.Formula:C29H31F3N6O3Purity:98.85% - 99.47%Color and Shape:SolidMolecular weight:568.59Cutamesine dihydrochloride
CAS:Cutamesine dihydrochloride is a σ1 receptor agonist, selective over σ2, combating cardiomyocyte hypertrophy and improving stroke recovery.Formula:C23H32N2O2·2HClPurity:99.96%Color and Shape:SolidMolecular weight:441.43Ref: TM-T3597
2mg35.00€5mg52.00€10mg90.00€25mg170.00€50mg274.00€100mg424.00€200mg612.00€1mL*10mM (DMSO)58.00€Aprepitant
CAS:Aprepitant (Aprepitant`) is a Substance P/Neurokinin-1 Receptor Antagonist.Formula:C23H21F7N4O3Purity:98% - 99.68%Color and Shape:Off-White To Light Yellow Cyrstalline SolidMolecular weight:534.43Aripiprazole monohydrate
CAS:Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.Formula:C23H29Cl2N3O3Color and Shape:SolidMolecular weight:466.4Domperidone monomaleate
CAS:Domperidone monomaleate, a selective oral dopamine-2 antagonist, aids gastric motility and has antiemetic properties.Formula:C26H28ClN5O6Color and Shape:SolidMolecular weight:541.98Sarpogrelate hydrochloride
CAS:Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.
Formula:C24H32ClNO6Purity:99.73%Color and Shape:Colorless LiquidMolecular weight:465.97Ozagrel hydrochloride
CAS:Ozagrel hydrochloride (OKY-046 HCl) is a selective thromboxane A(2) synthetase inhibitor used for the improvement of postoperative cerebrovascular contractionFormula:C13H12N2O2·HClPurity:99.80%Color and Shape:White Or Off White Crystalline PowderMolecular weight:264.71Bromopride hydrochloride
CAS:Bromopride HCl: Salt of a D2 blocker used for upper GI disorders, like dyspepsia and emesis.Formula:C14H23BrClN3O2Color and Shape:SolidMolecular weight:380.71LY334370
CAS:LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nMFormula:C21H22FN3OPurity:99.32%Color and Shape:SolidMolecular weight:351.42Prasugrel Hydrochloride
CAS:Prasugrel Hydrochloride (LY 640315 Hydrochloride) is pletelet aggregation inhibitor that is used to prevent thrombosis in patients with acute coronary syndrome.
Formula:C20H20FNO3S·HClPurity:99.39% - 99.79%Color and Shape:SolidMolecular weight:409.9Chlorprothixene
CAS:Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.Formula:C18H18ClNSPurity:98.77% - 99.756%Color and Shape:Pale Yellow Crystals SolidMolecular weight:315.86Nitrobenzylthioinosine
CAS:Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.
Formula:C17H17N5O6SPurity:99.69% - 99.74%Color and Shape:Off-White SolidMolecular weight:419.41Litorin acetate(55749-97-8 Free base)
Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.Formula:C53H72N14O13SPurity:98.61%Color and Shape:SolidMolecular weight:1145.29JNJ-31020028
CAS:JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity (pIC50=8.07, human; pIC50=8.22, rat).Formula:C34H36FN5O2Purity:95.92% - 99.65%Color and Shape:SolidMolecular weight:565.68AC-55541
CAS:AC-55541 (AOB2796), a PAR2 agonist, activates PAR2 in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays.
Formula:C25H20BrN5O3Purity:98% - 99.33%Color and Shape:SolidMolecular weight:518.36
