GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(55 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5985 products of "GPCR/G-Protein"
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Fenoprofen Calcium
CAS:Fenoprofen Calcium is a nonsteroidal, anti-inflammatory antiarthritic agent.Formula:C30H26CaO6Purity:99.24% - 99.66%Color and Shape:SolidMolecular weight:522.6cicloprofen
CAS:cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.Formula:C16H14O2Purity:98.15%Color and Shape:SolidMolecular weight:238.2812Ref: TM-T8586
1mg62.00€5mg123.00€10mg180.00€25mg298.00€50mg419.00€100mg567.00€200mg752.00€1mL*10mM (DMSO)111.00€Melperone
CAS:Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.Formula:C16H22FNOPurity:98.84%Color and Shape:SolidMolecular weight:263.35Metiamide
CAS:Metiamide (SK&F 92058) is a histamine H2-receptor antagonist .Formula:C9H16N4S2Purity:97.41%Color and Shape:SolidMolecular weight:244.38Atrasentan
CAS:Atrasentan (ABT-627) is an endothelin receptor antagonist that can inhibit the activity of ETA.Cost-effective and quality-assured.Formula:C29H38N2O6Purity:97.65% - 99.08%Color and Shape:SolidMolecular weight:510.62Ref: TM-TQ0259
1mg46.00€5mg90.00€10mg130.00€25mg250.00€50mg356.00€100mg580.00€200mg798.00€1mL*10mM (DMSO)109.00€GSK163090
CAS:GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).Formula:C25H29N5OPurity:99.2%Color and Shape:SolidMolecular weight:415.53Ref: TM-TQ0311
1mg34.00€2mg49.00€5mg75.00€10mg118.00€25mgTo inquire50mgTo inquire1mL*10mM (DMSO)82.00€[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
Broad-spectrum neuropeptide inverse agonist/antagonist; potent at ghrelin receptor (EC50 = 5.2 nM); inhibits cancer growth, induces apoptosis.Formula:C81H113N19O14Purity:97.68%Color and Shape:SolidMolecular weight:1576.91DOPEXAMINE
CAS:Dopexamine is a dopaminergic agonistFormula:C22H32N2O2Purity:99.42%Color and Shape:SolidMolecular weight:356.5Ref: TM-T8653
1mg131.00€2mg188.00€5mg284.00€10mg430.00€25mg710.00€50mg998.00€100mg1,349.00€1mL*10mM (DMSO)306.00€RS-127445 hydrochloride
CAS:RS-127445 hydrochloride (MT 500) is a selective, high affinity, orally bioavailable 5-HT2B receptor antagonist(pKi : 9.5).Formula:C17H17ClFN3Purity:99.48%Color and Shape:SolidMolecular weight:317.79PRX-08066
CAS:PRX-08066 is a selective 5-hydroxytryptamine receptor 2B (5-HT2BR, IC50= 3.4 nM) antagonist that induces selective vasodilation of pulmonary arteries.Formula:C19H17ClFN5SPurity:97.79% - 98.07%Color and Shape:SolidMolecular weight:401.89Ref: TM-T16669
1mg60.00€5mg119.00€10mg170.00€25mg350.00€50mg522.00€100mg748.00€200mg1,026.00€1mL*10mM (DMSO)111.00€Zacopride hydrochloride
CAS:Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.Formula:C15H20ClN3O2·HClPurity:98.32%Color and Shape:SolidMolecular weight:346.26Ref: TM-T5336
1mg34.00€5mg71.00€10mg99.00€25mg212.00€50mg385.00€100mg618.00€200mg859.00€1mL*10mM (DMSO)79.00€BD 1008 Free Base
CAS:BD 1008 Free Base: Sigma-1 receptor antagonist, Kᵢ = 2 ± 1 nM, 4x more selective for sigma-1 than sigma-2.Formula:C15H22Cl2N2Color and Shape:SolidMolecular weight:301.25Sonepiprazole hydrochloride
CAS:Sonepiprazole HCl is a a selective dopamine D4 antagonist.Formula:C21H28ClN3O3SColor and Shape:SolidMolecular weight:437.98Bupranolol HCl
CAS:Bupranolol: non-selective beta blocker, no ISA, strong membrane stabilizer, fast gut absorption, high first-pass metabolism, 2-4hr half-life.Formula:C14H23Cl2NO2Color and Shape:SolidMolecular weight:308.243Carmoxirole (free base)
CAS:Carmoxirole: a dopamine D2 agonist, reduces pre-load/afterload, aids heart failure, lowers blood pressure by inhibiting noradrenaline release.Formula:C24H26N2O2Color and Shape:SolidMolecular weight:374.48Milveterol
CAS:Milveterol is a long-acting β(2)-adrenoceptor agonist.Formula:C25H29N3O4Color and Shape:SolidMolecular weight:435.52Vicriviroc
CAS:Vicriviroc, also known as MK4176 is a CCR5 antagonist.Formula:C28H38F3N5O2Color and Shape:SolidMolecular weight:533.63Batefenterol Succinate
CAS:Batefenterol Succinate is a first-in-class inhaled bifunctional bronchodilator possessing muscarinic receptor antagonist and β2-adrenoceptor agonist properties.Formula:C44H48ClN5O11Color and Shape:SolidMolecular weight:858.34Atipamezole hydrochloride
CAS:Atipamezole is a synthetic α2 adrenergic receptor antagonist.Formula:C14H16N2·HClPurity:99.74%Color and Shape:SolidMolecular weight:248.75Ref: TM-T6765
5mg51.00€10mg74.00€25mg133.00€50mg230.00€100mg343.00€200mg535.00€500mg843.00€1mL*10mM (DMSO)57.00€PF-06882961 Tris
CAS:PF-06882961 Tris (UNII-2HJV78O0SS) is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.Formula:C35H41FN6O7Purity:98.74% - 99.79%Color and Shape:SolidMolecular weight:676.7
![[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1931L1.webp&w=3840&q=75)
