GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(444 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(55 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5984 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
SB 242084
CAS:SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.Formula:C21H19ClN4O2Purity:99.75% - ≥98%Color and Shape:SolidMolecular weight:394.85NPY 5RA972
CAS:NPY 5RA972 is a neuropeptide Y Y5 receptor antagonistFormula:C21H25N3O2Purity:99.02% - 99.56%Color and Shape:SolidMolecular weight:351.44Orexin 2 Receptor Agonist
CAS:Orexin 2 Receptor Agonist (OX2R) is an effective (EC50: 23 nM) and OX2R-selective (OX1R/OX2R EC50 ratio: 70) agonist.Formula:C32H34N4O5SPurity:98.26% - 99.43%Color and Shape:SolidMolecular weight:586.7Ref: TM-T3177
2mg39.00€5mg60.00€10mg75.00€25mg130.00€50mg220.00€100mg323.00€200mg447.00€1mL*10mM (DMSO)77.00€Sotagliflozin
CAS:Sotagliflozin (LP-802034) is an orally bioavailable inhibitor of the sodium-glucose co-transporter subtype 1 (SGLT1) and 2 (SGLT2), with potentialFormula:C21H25ClO5SPurity:99% - 99.86%Color and Shape:SolidMolecular weight:424.94Ref: TM-T3547
1mg46.00€2mg57.00€5mg87.00€10mg131.00€25mg248.00€50mg378.00€100mg560.00€500mg1,198.00€1mL*10mM (DMSO)88.00€CS 2100
CAS:<p>CS 2100 (1-[[4-Ethyl-5-[5-(4-phenoxyphenyl)-1,2,4-oxadiazol-3-yl]-2-thienyl]methyl]-3-azetidinecarboxylic acid) is an S1P1 agonist.</p>Formula:C25H23N3O4SPurity:99.19%Color and Shape:SolidMolecular weight:461.53Bevantolol hydrochloride
CAS:Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.Formula:C20H28ClNO4Purity:99.49%Color and Shape:SolidMolecular weight:381.9Diphenhydramine
CAS:Diphenhydramine (Syntedril): first-gen antihistamine for allergies, antiemetic, antitussive, anticholinergic, sedative, treats drug-induced parkinsonism.Formula:C17H21NOPurity:98.07%Color and Shape:SolidMolecular weight:255.35Pimozide
CAS:Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.Formula:C28H29F2N3OPurity:99.63% - >99.99%Color and Shape:SolidMolecular weight:461.55Ivabradine hydrochloride
CAS:Ivabradine HCl (S 16257-2) is an If inhibitor (IC50: 2.9 μM) and SA node HCN channel blocker that slows heart rate.Formula:C27H37ClN2O5Purity:99% - 99.73%Color and Shape:SolidMolecular weight:505.05Perospirone
CAS:Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Formula:C23H30N4O2SPurity:99.23%Color and Shape:White PowderMolecular weight:426.57DAPTA
CAS:DAPTA (Adaptavir) is an inhibitor of CCR5, shows potent anti-HIV activities.Formula:C35H56N10O15Purity:>99.99%Color and Shape:SolidMolecular weight:856.88PAR-2 Activating Peptide acetate
PAR-2 Activating Peptide acetate (SLIGRL-NH2 acetate) is an agonist of Protease-Activated Receptor-2 (PAR-2).Formula:C31H60N10O9Purity:98.5% - 99.92%Color and Shape:SolidMolecular weight:716.88Ebastine
CAS:Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine.Formula:C32H39NO2Purity:99.65% - 99.99%Color and Shape:White To Off-White PowderMolecular weight:469.66BMY-25368
CAS:BMY-25368 is a long-acting antagonist of the H2-receptor.Formula:C19H25N3O3Color and Shape:SolidMolecular weight:343.42Haloperidol hydrochloride
CAS:Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist which is a potent antipsychotic agent.Formula:C21H24Cl2FNO2Color and Shape:SolidMolecular weight:412.33Dolasetron Mesylate hydrate
CAS:Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.Formula:C20H26N2O7SPurity:99.86% - 99.99%Color and Shape:SolidMolecular weight:438.49MK-3697
CAS:<p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>Formula:C23H21N5O3SPurity:97.69% - 98.15%Color and Shape:SolidMolecular weight:447.51[Des-Arg9]-Bradykinin TFA
CAS:[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.Formula:C46H62F3N11O12Purity:>99.99%Color and Shape:SolidMolecular weight:1018.05JNJ-5207852 dihydrochloride
CAS:JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptorFormula:C20H34Cl2N2OPurity:99.51%Color and Shape:SolidMolecular weight:389.4CGP71683 hydrochloride
CAS:CGP71683 hydrochloride: NPY5 receptor antagonist, Ki=1.3 nM; inactive at Y1 (Ki >4000 nM) and Y2 (Ki=200 nM).Formula:C26H30ClN5O2SPurity:99.92%Color and Shape:SolidMolecular weight:512.07
![[Des-Arg9]-Bradykinin TFA](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT8809.webp&w=3840&q=75)
