GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

Show 18 more subcategories

Found 5696 products of "GPCR/G-Protein"

Purity (%)

100

products per page.

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ETHYL 2-AMINO-4-METHYL-5-PHENYLTHIOPHENE-3-CARBOXYLATE
CAS:
- 4815-38-7
ETHYL 2-AMINO-4-METHYL-5-PHENYLTHIOPHENE-3-CARBOXYLATE targets the prostaglandin E2 receptor EP2 subtype (human)
Formula:C₁₄H₁₅NO₂S
Purity:99.98%
Color and Shape:Solid
Molecular weight:261.34
Ref: TM-T8603
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Etilevodopa hydrochloride
CAS:
- 39740-30-2
Etilevodopa hydrochloride (L-DOPA ethyl ester) is a prodrug of levodopa. It also has greater gastric solubility and significant brain penetration.
Formula:C₁₁H₁₆ClNO₄
Purity:95.00%
Color and Shape:Solid
Molecular weight:261.7
Ref: TM-T24047
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4F 4PP oxalate
CAS:
- 144734-36-1
4F 4PP oxalate is a 5-HT2A antagonist.
Formula:C₂₂H₂₆FNO·C₂H₂O₄
Purity:97.34%
Color and Shape:Solid
Molecular weight:429.49
Ref: TM-T22514
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Intepirdine
CAS:
- 607742-69-8
Intepirdine (GSK-742457) is a highly selective 5-HT6 receptor antagonist, used in trials studying the treatment of Alzheimer's Disease.
Formula:C₁₉H₁₉N₃O₂S
Purity:98% - 98.63%
Color and Shape:Solid
Molecular weight:353.44
Ref: TM-T1774
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Pranlukast hemihydrate
CAS:
- 150821-03-7
Pranlukast hemihydrate (ONO-1078 hemihydrate) is an LT antagonist with anti-asthmatic activity.
Formula:C₂₇H₂₃N₅O₄₀·5H₂O
Purity:99.28%
Color and Shape:Solid
Molecular weight:490.52
Ref: TM-T63291
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Ibutamoren Mesylate
CAS:
- 159752-10-0
Ibutamoren Mesylate (MK-0677) is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.
Formula:C₂₈H₄₀N₄O₈S₂
Purity:97.98% - ≥98%
Color and Shape:Solid
Molecular weight:624.77
Ref: TM-T7112
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Clozapine N-Oxide
CAS:
- 34233-69-7
View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.
Formula:C₁₈H₁₉ClN₄O
Purity:98.65% - 99.94%
Color and Shape:Solid
Molecular weight:342.82
Ref: TM-T4494
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Cariprazine hydrochloride
CAS:
- 1083076-69-0
Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)
Formula:C₂₁H₃₃Cl₃N₄O
Purity:99.78% - >99.99%
Color and Shape:Solid
Molecular weight:463.87
Ref: TM-T8382
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2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base)
2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) is a potent and selective protease-activated receptor 2 (PAR2) agonist.
Formula:C₃₈H₆₄F₃N₁₁O₁₀
Purity:>99.99%
Color and Shape:Solid
Molecular weight:891.98
Ref: TM-TP1378
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Ajmalicine hydrochloride
CAS:
- 4373-34-6
Ajmalicine hydrochloride is a potent α1-adrenoceptor blocker, non-competitive nicotine receptor inhibitor, anti-hypertensive, and sedative. IC50: 72.3 μM.
Formula:C₂₁H₂₅ClN₂O₃
Color and Shape:Solid
Molecular weight:388.89
Ref: TM-T69254
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PAR-2-IN-1
CAS:
- 1690176-75-0
PAR-2-IN-1 (IUN76750) is a PAR- 2 signaling pathway inhibitor with anti-inflammatory and anticancer effects.
Formula:C₁₂H₁₄ClN₃O₂
Purity:99.75%
Color and Shape:Solid
Molecular weight:267.71
Ref: TM-T8917
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Triprolidine
CAS:
- 486-12-4
Triprolidine: oral H1 receptor blocker with motor/sensory spinal effects, for allergy research.
Formula:C₁₉H₂₂N₂
Color and Shape:Solid
Molecular weight:278.39
Ref: TM-T60514
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Enavogliflozin
CAS:
- 1415472-28-4
Enavogliflozin (DWP-16001) is an orally available small molecule and sodium glucose transporter 2 inhibitor.
Formula:C₂₄H₂₇ClO₆
Purity:97.37%
Color and Shape:Solid
Molecular weight:446.92
Ref: TM-T38843
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Atipamezole hydrochloride
CAS:
- 104075-48-1
Atipamezole is a synthetic α2 adrenergic receptor antagonist.
Formula:C₁₄H₁₆N₂·HCl
Purity:99.74%
Color and Shape:Solid
Molecular weight:248.75
Ref: TM-T6765
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BD1063 dhydrochloride
CAS:
- 206996-13-6
BD1063 dhydrochloride is a potent and selective sigma 1(σ1) receptor antagonist(Ki = 9 nM).
Formula:C₁₃H₂₀Cl₄N₂
Purity:99.52% - ≥95%
Color and Shape:Solid
Molecular weight:346.12
Ref: TM-T7488
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Vortioxetine
CAS:
- 508233-74-7
Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.
Formula:C₁₈H₂₂N₂S
Purity:99.34% - 99.34%
Color and Shape:Solid
Molecular weight:298.45
Ref: TM-T2395
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Alcaftadine
CAS:
- 147084-10-4
Alcaftadine (Lastacaft) is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis.
Formula:C₁₉H₂₁N₃O
Purity:98% - 98.65%
Color and Shape:Solid
Molecular weight:307.39
Ref: TM-T2533
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Dasotraline
CAS:
- 675126-05-3
Dasotraline: a triple reuptake inhibitor targeting DA, NE, and 5-HT with IC50 values of 4, 6, 11 nM. Possible new antidepressant class.
Formula:C₁₆H₁₅Cl₂N
Color and Shape:Solid
Molecular weight:292.2
Ref: TM-T60607
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Regadenoson hydrate
CAS:
- 875148-45-1
Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.
Formula:C₁₅H₂₀N₈O₆
Purity:98%
Color and Shape:Solid
Molecular weight:408.37
Ref: TM-T26054
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GR 125743
CAS:
- 148547-33-5
GR 125743 is a novel antagonist of 5-HT1B/1D receptor.
Formula:C₂₅H₂₈N₄O₂
Purity:99.76%
Color and Shape:Solid
Molecular weight:416.52
Ref: TM-T8737