GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(53 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5980 products of "GPCR/G-Protein"
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Desvenlafaxine
CAS:Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.Formula:C16H25NO2Purity:99.46% - 99.81%Color and Shape:White Crystalline PowderMolecular weight:263.38Aniracetam
CAS:Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.Formula:C12H13NO3Purity:99.88% - 99.89%Color and Shape:White Crystalline Or Crystalline PowdeMolecular weight:219.24Terbutaline Sulfate
CAS:Terbutaline Sulfate (Terbutaline hemisulfate) is a selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic.Formula:C12H19NO3H2SO4Purity:99.47% - 99.94%Color and Shape:Crystalline PowderMolecular weight:274.32Doxepin hydrochloride
CAS:Doxepin hydrochloride, a dibenzoxepin tricyclic, blocks monoamine reuptake and has anticholinergic and antihistaminic effects. Mechanism partly unknown.Formula:C19H22ClNOPurity:99.65% - 99.91%Color and Shape:White To Off-White PowderMolecular weight:315.84Sulpiride
CAS:Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.Formula:C15H23N3O4SPurity:99.94%Color and Shape:White Crystalline PowderMolecular weight:341.43Sumatriptan succinate
CAS:Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment of a migraine headache.Formula:C18H27N3O6SPurity:97.53% - 99.51%Color and Shape:White PowderMolecular weight:413.49Amitriptyline hydrochloride
CAS:Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptiveFormula:C20H24ClNPurity:97% - 99.94%Color and Shape:Crystals White To Off-White PowderMolecular weight:313.86Aripiprazole Lauroxil
CAS:Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.Formula:C36H51Cl2N3O4Purity:99.64%Color and Shape:SolidMolecular weight:660.71Ref: TM-T14319
10mg48.00€25mg72.00€50mg96.00€100mg130.00€200mg188.00€500mg318.00€1mL*10mM (DMSO)49.00€Delequamine
CAS:Delequamine (RS 15385-197) is a TNIK inhibitor (IC50: 8 nM).TINK-IN-1 inhibits colorectal cancer cell viability and can be used to study mental retardation.Formula:C18H26N2O3SPurity:99.39%Color and Shape:SolidMolecular weight:350.48Lesopitron HCl
CAS:<p>Lesopitron HCl is a 5-HT1A receptor agonist with anxiolytic effects that reverses dark avoidance behavior associated with cocaine withdrawal in mice.</p>Formula:C15H22Cl2N6Purity:97.05% - 99.89%Color and Shape:SoildMolecular weight:357.28Tirzepatide monosodium salt
Tirzepatide sodium salt (LY3298176 sodium salt) is a GIP and GLP-1 receptor agonist with neuroprotective activity and can be used to treat obesity.Formula:C225H347N48O68NaPurity:99.69%Color and Shape:SoildMolecular weight:4835.51Lintopride HCl
CAS:Lintopride HCl is a 5HT-4 antagonist.Formula:C14H20Cl2N4O2Purity:98.42% - 98.81%Color and Shape:SoildMolecular weight:347.24AVN 322 free base
CAS:AVN 322 free base is an orally available, selective and potent 5-HT6R antagonist for the study of neuropathic system disorders such as Alzheimer's disease (AD) and schizophrenia.Formula:C17H19N5O2SPurity:99.24%Color and Shape:SolidMolecular weight:357.43Risperidone
CAS:Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.Formula:C23H27FN4O2Purity:99.73%Color and Shape:Crystalline SolidMolecular weight:410.48Ref: TM-T0351
10mg50.00€25mg59.00€50mg93.00€100mg128.00€200mg202.00€500mg340.00€1mL*10mM (DMSO)To inquireAzelastine hydrochloride
CAS:Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.Formula:C22H24ClN3O·HClPurity:98% - >99.99%Color and Shape:White Crystalline PowderMolecular weight:418.36Dexchlorpheniramine Maleate
CAS:Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.Formula:C20H23ClN2O4Purity:99.58%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:390.86L-741626
CAS:L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3Formula:C20H21ClN2OPurity:98.57%Color and Shape:SolidMolecular weight:340.85Iloperidone
CAS:Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.Formula:C24H27FN2O4Purity:99.42%Color and Shape:SolidMolecular weight:426.48Latozinemab
Latozinemab (AL001) is a humanized monoclonal antibody targeting Sortilin to study dementia and Alzheimer's.Purity:> 95%Color and Shape:LiquidMolecular weight:146.28 kDaBIBO3304 TFA
CAS:BIBO3304 TFA: Oral, selective NPY Y1 receptor blocker; IC50: 0.38 nM (human), 0.72 nM (rat).Formula:C31H36F3N7O5Purity:99.5%Color and Shape:SolidMolecular weight:643.66Ref: TM-T10539
1mg66.00€5mg144.00€10mg255.00€25mg580.00€50mg798.00€100mg1,074.00€1mL*10mM (DMSO)197.00€
