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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5959 products of "GPCR/G-Protein"

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  • Plecanatide

    CAS:
    Plecanatide acetate is an analogue of Uroguanylin. It is an orally active guanylate cyclase-C (GC-C) receptor agonist.
    Formula:C65H104N18O26S4
    Purity:97.51%
    Color and Shape:Solid
    Molecular weight:1681.89

    Ref: TM-T9080

    1mg
    79.00€
    5mg
    180.00€
    10mg
    298.00€
    25mg
    590.00€
    50mg
    835.00€
    100mg
    1,121.00€
  • Etrasimod

    CAS:
    Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: 1.88 nM in CHO cells).
    Formula:C26H26F3NO3
    Purity:98.52% - 99.73%
    Color and Shape:Solid
    Molecular weight:457.48

    Ref: TM-TQ0227

    1mg
    50.00€
    5mg
    105.00€
    10mg
    170.00€
    25mg
    230.00€
    50mg
    289.00€
    100mg
    401.00€
    1mL*10mM (DMSO)
    107.00€
  • Vanoxerine dihydrochloride

    CAS:
    Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)
    Formula:C28H34Cl2F2N2O
    Purity:98.16% - 98.35%
    Color and Shape:White Solid
    Molecular weight:523.49

    Ref: TM-T7153

    10mg
    49.00€
    25mg
    81.00€
    50mg
    114.00€
    100mg
    167.00€
    1mL*10mM (DMSO)
    34.00€
  • CCG215022

    CAS:
    CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.
    Formula:C26H22FN7O3
    Purity:97.63% - 99.69%
    Color and Shape:Solid
    Molecular weight:499.5

    Ref: TM-T3498

    1mg
    56.00€
    5mg
    114.00€
    10mg
    178.00€
    25mg
    394.00€
    50mg
    655.00€
    100mg
    1,035.00€
    1mL*10mM (DMSO)
    127.00€
  • Clemizole hydrochloride

    CAS:
    Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.
    Formula:C19H21Cl2N3
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:362.3

    Ref: TM-T1822L

    5mg
    34.00€
    10mg
    50.00€
    25mg
    92.00€
    50mg
    147.00€
    100mg
    222.00€
    1mL*10mM (DMSO)
    39.00€
  • Hemopressin (rat) acetate(568588-77-2 free base)


    Hemopressin is a nonapeptide, CB2 agonist, derived from rat hemoglobin, with antinociceptive properties.
    Formula:C5H81N13O14
    Purity:99.37%
    Color and Shape:Solid
    Molecular weight:1148.31

    Ref: TM-TP1901L1

    1mg
    161.00€
    5mg
    350.00€
    10mg
    477.00€
    25mg
    705.00€
    50mg
    945.00€
    100mg
    1,279.00€
    200mg
    1,720.00€
  • LY 78335

    CAS:
    LY 78335 (1-(2,3-Dichlorophenyl)ethanamine hydrochloride) is a phenylethanolamine-N-methyltransferase (PNMT) inhibitor.
    Formula:C8H10Cl3N
    Purity:99.30% - 99.81%
    Color and Shape:Solid
    Molecular weight:226.53

    Ref: TM-T22956

    2mg
    33.00€
    5mg
    50.00€
    10mg
    80.00€
    25mg
    161.00€
    50mg
    245.00€
    100mg
    354.00€
    200mg
    515.00€
  • Norepinephrine bitartrate salt

    CAS:
    Norepinephrine bitartrate salt is an adrenergic neurotransmitter.
    Formula:C12H17NO9
    Purity:97.32% - 99.97%
    Color and Shape:Solid
    Molecular weight:319.27

    Ref: TM-T21066

    10mg
    48.00€
    25mg
    74.00€
    50mg
    97.00€
    100mg
    153.00€
    500mg
    368.00€
    1mL*10mM (DMSO)
    35.00€
  • BMS-813160

    CAS:
    BMS-813160 is the first dual CCR2/CCR5 antagonist to enter Clinical development for cardiovascular.
    Formula:C25H40N8O2
    Purity:99.66% - 99.79%
    Color and Shape:Solid
    Molecular weight:484.64

    Ref: TM-T4584

    1mg
    63.00€
    5mg
    137.00€
    10mg
    187.00€
    25mg
    341.00€
    50mg
    567.00€
    100mg
    810.00€
    500mg
    1,644.00€
    1mL*10mM (DMSO)
    145.00€
  • 4i

    CAS:
    4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.
    Formula:C16H12ClN3O
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:297.74

    Ref: TM-T8438

    1mg
    62.00€
    5mg
    123.00€
    10mg
    180.00€
    25mg
    298.00€
    50mg
    419.00€
    100mg
    567.00€
    200mg
    752.00€
  • Mecamylamine

    CAS:
    Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.
    Formula:C11H21N
    Color and Shape:Solid
    Molecular weight:167.29

    Ref: TM-T69019

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CRF (6-33) acetate(120066-38-8 free base)


    CRFBP inhibitor peptide; reduces weight gain, boosts activity in obese rats.
    Formula:C143H235N41O45S
    Purity:97.12%
    Color and Shape:Solid
    Molecular weight:3280.76

    Ref: TM-TP2047L

    1mg
    200.00€
    5mg
    452.00€
    10mg
    627.00€
    25mg
    928.00€
    50mg
    1,251.00€
    100mg
    1,684.00€
  • Bepotastine Besilate

    CAS:
    Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).
    Formula:C21H25ClN2O3·C6H6O3S
    Purity:99.83% - 99.9%
    Color and Shape:Brown Viscous Liquid
    Molecular weight:547.06

    Ref: TM-T6405

    100mg
    44.00€
    500mg
    94.00€
    1mL*10mM (DMSO)
    33.00€
  • BAY 41-8543

    CAS:

    BAY 41-8543 is a nitric oxide (NO)-independent stimulator of soluble guanylyl cyclase (sGC).

    Formula:C21H21FN8O
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:420.44

    Ref: TM-T21712

    2mg
    38.00€
    5mg
    52.00€
    10mg
    85.00€
    25mg
    156.00€
    50mg
    240.00€
    100mg
    350.00€
  • Zacopride hydrochloride

    CAS:
    Zacopride is a highly potent 5-HT3 receptor antagonist (Kd = 0.38 nM) and 5-HT4 receptor agonist (Ki = 373 nM). It also is a selective IK1 channel agonist.
    Formula:C15H20ClN3O2·HCl
    Purity:98.32%
    Color and Shape:Solid
    Molecular weight:346.26

    Ref: TM-T5336

    1mg
    34.00€
    5mg
    71.00€
    10mg
    99.00€
    25mg
    212.00€
    50mg
    385.00€
    100mg
    618.00€
    200mg
    859.00€
    1mL*10mM (DMSO)
    79.00€
  • RO1138452

    CAS:
    RO1138452 (CAY10441) blocks prostacyclin receptor; orally active, high affinity (Ki: 1.5 nM), analgesic in rats (2-20 mg/kg).
    Formula:C19H23N3O
    Purity:97.01% - 99.34%
    Color and Shape:Solid
    Molecular weight:309.41

    Ref: TM-T4436

    1mg
    49.00€
    2mg
    65.00€
    5mg
    90.00€
    10mg
    144.00€
    25mg
    313.00€
    50mg
    537.00€
    100mg
    767.00€
    1mL*10mM (DMSO)
    90.00€
  • TNCA

    CAS:
    TNCA (Lycoperodine-1) is a high-affinity CaSR ligand (CaSRL) with co-agonist activity.
    Formula:C12H12N2O2
    Purity:97.33% - 97.73%
    Color and Shape:Solid
    Molecular weight:216.24

    Ref: TM-T7716

    10mg
    34.00€
    25mg
    54.00€
    50mg
    84.00€
    100mg
    114.00€
    500mg
    268.00€
  • Clobenpropit 2HBr

    CAS:
    Clobenpropit 2HBr is a histamine H3 receptor antagonist. It has neuroprotective effects via stimulation of GABA release in the brain.
    Formula:C14H17ClN4S
    Color and Shape:Solid
    Molecular weight:308.83

    Ref: TM-T19762

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BRL-15572 dihydrochloride

    CAS:
    BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.
    Formula:C25H27ClN2O·2HCl
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:479.87

    Ref: TM-T6423

    10mg
    46.00€
    25mg
    67.00€
    50mg
    94.00€
    100mg
    138.00€
    1mL*10mM (DMSO)
    34.00€
  • Xaliproden hydrochloride

    CAS:
    Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.
    Formula:C24H23ClF3N
    Purity:99.99%
    Color and Shape:Solid
    Molecular weight:417.89

    Ref: TM-T9272

    1mg
    38.00€
    5mg
    80.00€
    10mg
    114.00€
    25mg
    222.00€
    50mg
    356.00€
    100mg
    512.00€
    200mg
    735.00€
    1mL*10mM (DMSO)
    92.00€