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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5960 products of "GPCR/G-Protein"

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  • AnaMorelin hydrochloride

    CAS:
    AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).
    Formula:C31H43ClN6O3
    Purity:99.18% - ≥98%
    Color and Shape:Solid
    Molecular weight:583.16

    Ref: TM-T7225

    1mg
    35.00€
    2mg
    50.00€
    5mg
    73.00€
    10mg
    96.00€
    25mg
    145.00€
    50mg
    177.00€
    100mg
    235.00€
    1mL*10mM (DMSO)
    95.00€
  • PAR-2 Activating Peptide acetate


    PAR-2 Activating Peptide acetate (SLIGRL-NH2 acetate) is an agonist of Protease-Activated Receptor-2 (PAR-2).
    Formula:C31H60N10O9
    Purity:98.5% - 99.92%
    Color and Shape:Solid
    Molecular weight:716.88

    Ref: TM-TP1046L

    1mg
    81.00€
    5mg
    185.00€
    10mg
    330.00€
    25mg
    557.00€
    50mg
    792.00€
    100mg
    1,071.00€
    200mg
    1,431.00€
  • HPI 1

    CAS:
    HPI 1 suppresses Hh pathway: IC50 = 1.5 μM (Shh, SAG), 4 μM (Gli2), 6 μM (Gli1) in Shh-LIGHT2 cells.
    Formula:C27H29NO6
    Purity:97.6%
    Color and Shape:Solid
    Molecular weight:463.52

    Ref: TM-T22089

    1mg
    47.00€
    2mg
    60.00€
    5mg
    92.00€
    10mg
    135.00€
    25mg
    217.00€
    50mg
    324.00€
    100mg
    472.00€
    500mg
    1,026.00€
    1mL*10mM (DMSO)
    107.00€
  • Gadolinium chloride

    CAS:
    Gadolinium chloride is a calcium-sensing receptor (CaSR) agonist
    Formula:Cl3Gd
    Purity:98%
    Color and Shape:White Crystalline Solid
    Molecular weight:263.61

    Ref: TM-T22795

    25mg
    46.00€
    50mg
    55.00€
    100mg
    85.00€
    200mg
    119.00€
  • H2L 5765834

    CAS:
    H2L 5765834 is a lysophosphatidic acid receptors antagonist
    Formula:C21H12N2O7
    Purity:98.25% - 99.47%
    Color and Shape:Solid
    Molecular weight:404.33

    Ref: TM-T22834

    1mg
    58.00€
    5mg
    113.00€
    10mg
    177.00€
    25mg
    334.00€
    50mg
    497.00€
    100mg
    708.00€
    1mL*10mM (DMSO)
    124.00€
  • Sultopride hydrochloride

    CAS:
    Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.
    Formula:C17H27ClN2O4S
    Purity:≥95%
    Color and Shape:White Or Yellowish Powder
    Molecular weight:390.93

    Ref: TM-T7180

    1mg
    35.00€
    5mg
    70.00€
    10mg
    97.00€
    25mg
    187.00€
    50mg
    283.00€
    100mg
    424.00€
    1mL*10mM (DMSO)
    78.00€
  • Metadoxine

    CAS:
    Metadoxine (Metadoxil) is a neurotransmitter stimulant.
    Formula:C8H11NO3·C5H7NO3
    Purity:99.19%
    Color and Shape:Off-White Powder
    Molecular weight:298.29

    Ref: TM-T3269

    1g
    108.00€
    100mg
    37.00€
    200mg
    50.00€
    500mg
    81.00€
    1mL*10mM (DMSO)
    33.00€
  • Pasireotide Acetate

    CAS:
    The pKi of Pasireotide (SOM230) acetate for sst1, 2, 3, 4, and 5 were 8.2, 9.0, 9.1, less than 7.0, and 9.9, respectively.Cost-effective and quality-assured.
    Formula:C60H70N10O11
    Purity:98.64% - 99.92%
    Color and Shape:Solid
    Molecular weight:1107.26

    Ref: TM-TP2207

    1mg
    90.00€
    2mg
    138.00€
    5mg
    236.00€
    10mg
    409.00€
    25mg
    745.00€
    50mg
    1,189.00€
    100mg
    1,684.00€
    200mg
    2,268.00€
  • Almotriptan Malate

    CAS:
    Almotriptan Malate (PNU180638), a selective 5-HT1B/1D receptor agonist, is used in the therapy of Migraine attacks in adults.
    Formula:C17H25N3O2S·C4H6O5
    Purity:99.95%
    Color and Shape:Pale Yellow Solid
    Molecular weight:469.55

    Ref: TM-T2317

    25mg
    52.00€
    50mg
    90.00€
    100mg
    131.00€
    200mg
    187.00€
    1mL*10mM (DMSO)
    34.00€
  • Cetrorelix diacetate

    CAS:
    Cetrorelix diacetate (NS-75A) is is a gonadotropin-releasing hormone antagonist.
    Formula:C74H100ClN17O18
    Purity:98.38%
    Color and Shape:Solid
    Molecular weight:1551.17

    Ref: TM-T5520L

    1mg
    52.00€
    5mg
    90.00€
    10mg
    150.00€
    25mg
    291.00€
    50mg
    437.00€
    100mg
    642.00€
    500mg
    1,359.00€
    1mL*10mM (DMSO)
    251.00€
  • CHEMBL241987

    CAS:
    CHEMBL241987 targets the Adenosine receptor A3 (human)
    Formula:C16H11N3O
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:261.28

    Ref: TM-T8598

    5mg
    34.00€
    10mg
    48.00€
    25mg
    80.00€
    50mg
    107.00€
    100mg
    161.00€
    200mg
    233.00€
    1mL*10mM (DMSO)
    35.00€
  • Pentagastrin

    CAS:
    Pentagastrin (ICI-50123) is a synthetic polypeptide that has effects like gastrin when given parenterally, which can cause the secretion and synthesis of
    Formula:C37H49N7O9S
    Purity:96.98% - 99.49%
    Color and Shape:Fine Colorless Needle-Shaped Crystals From 2-Ethoxyethanol + Water Solid
    Molecular weight:767.89

    Ref: TM-T4579

    5mg
    49.00€
    10mg
    69.00€
    25mg
    127.00€
    50mg
    202.00€
    100mg
    324.00€
    1mL*10mM (DMSO)
    69.00€
  • Serotonin hydrochloride

    CAS:
    Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (
    Formula:C10H13ClN2O
    Purity:98.05% - 99.93%
    Color and Shape:White To Cream Powder
    Molecular weight:212.676

    Ref: TM-T2209

    25mg
    34.00€
    50mg
    47.00€
    100mg
    54.00€
    200mg
    74.00€
    1mL*10mM (DMSO)
    49.00€
  • Chlorprothixene

    CAS:
    Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.
    Formula:C18H18ClNS
    Purity:98.77% - 99.756%
    Color and Shape:Pale Yellow Crystals Solid
    Molecular weight:315.86

    Ref: TM-T0074

    1g
    133.00€
    100mg
    34.00€
    200mg
    50.00€
    500mg
    92.00€
  • [Des-Arg9]-Bradykinin TFA

    CAS:
    [Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.
    Formula:C46H62F3N11O12
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:1018.05

    Ref: TM-T8809

    2mg
    34.00€
    5mg
    37.00€
    10mg
    50.00€
    25mg
    94.00€
    50mg
    126.00€
    100mg
    182.00€
    200mg
    264.00€
  • Cinanserin

    CAS:
    Cinanserin is a serotonin 5-HT2 antagonist.
    Formula:C20H24N2OS
    Color and Shape:Solid
    Molecular weight:340.48

    Ref: TM-T71350

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Liraglutide

    CAS:
    Liraglutide (Liraglutida) is a synthetic analog of GLP-1, an agonist of the GLP-1 receptor. Liraglutide is an antidiabetic agent. Cost effective and quality assured.
    Formula:C172H265N43O51
    Purity:97.65% - 99.04%
    Color and Shape:Solid
    Molecular weight:3751.25

    Ref: TM-T6876

    1mg
    111.00€
    2mg
    197.00€
    5mg
    447.00€
    10mg
    527.00€
    25mg
    843.00€
    50mg
    1,144.00€
    100mg
    1,521.00€
    200mg
    2,052.00€
  • GRK5-IN-2

    CAS:
    GRK5-IN-2, a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor.
    Formula:C20H20N4O4
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:380.4

    Ref: TM-T9609

    2mg
    34.00€
    5mg
    52.00€
    10mg
    75.00€
    25mg
    138.00€
    50mg
    215.00€
    100mg
    318.00€
    200mg
    444.00€
    1mL*10mM (DMSO)
    52.00€
  • ML-18

    CAS:
    ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of 4.8 μM.
    Formula:C32H35N5O5
    Purity:98.62% - >99.99%
    Color and Shape:Solid
    Molecular weight:569.65

    Ref: TM-T4540

    1mg
    34.00€
    5mg
    60.00€
    10mg
    96.00€
    25mg
    170.00€
    50mg
    264.00€
    100mg
    425.00€
    200mg
    587.00€
    1mL*10mM (DMSO)
    75.00€
  • Alizapride hydrochloride

    CAS:
    Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.
    Formula:C16H21N5O2·HCl
    Purity:99.35% - 99.48%
    Color and Shape:Coa
    Molecular weight:351.83

    Ref: TM-T2574

    25mg
    34.00€
    50mg
    46.00€
    100mg
    66.00€
    500mg
    144.00€
    1mL*10mM (DMSO)
    44.00€