GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,997 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5958 products of "GPCR/G-Protein"
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Naftopidil dihydrochloride
CAS:Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.Formula:C24H28N2O3·2HClPurity:99.76%Color and Shape:White SolidMolecular weight:465.41Idalopirdine Hydrochloride
CAS:Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.
Formula:C20H20ClF5N2OPurity:99.77%Color and Shape:SolidMolecular weight:434.83BAR501
CAS:BAR501是高效选择性的 GPBAR1激动剂(EC50:1 μM)。Formula:C26H46O3Purity:99.29% - 99.68%Color and Shape:SolidMolecular weight:406.644F 4PP oxalate
CAS:4F 4PP oxalate is a 5-HT2A antagonist.
Formula:C22H26FNO·C2H2O4Purity:97.34%Color and Shape:SolidMolecular weight:429.49BQ-788 sodium salt
CAS:BQ-788 sodium salt is a potent and selective antagonist of ETB receptor(ETB receptors with an IC50 of 1.2 nM in human Girrardi heart cells).Formula:C34H51N5NaO7Color and Shape:SolidMolecular weight:664.8Naftopidil hydrochloride
CAS:Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 nM; it also inhibits cell growth.Formula:C24H29ClN2O3Purity:99.5%Color and Shape:SolidMolecular weight:428.95Ref: TM-T9220
1mg42.00€5mg82.00€10mg111.00€25mg192.00€50mg289.00€100mg414.00€200mg580.00€1mL*10mM (DMSO)92.00€NPS2390
CAS:NPS2390 is a first generation quinoxaline derivative that acts as a noncompetitive antagonist of mGluR1 and mGluR5 (IC50 of 5.2 and 82 nM, respectively)Formula:C19H21N3OPurity:97.13%Color and Shape:SolidMolecular weight:307.39[Des-Arg9]-Bradykinin TFA
CAS:[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.Formula:C46H62F3N11O12Purity:>99.99%Color and Shape:SolidMolecular weight:1018.05Aripiprazole monohydrate
CAS:Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.Formula:C23H29Cl2N3O3Color and Shape:SolidMolecular weight:466.4Cangrelor free acid
CAS:Cangrelor, a reversible P2Y12 inhibitor for IV use, was approved in June 2015; it rapidly blocks ADP-induced platelet aggregation.Formula:C17H25Cl2F3N5O12P3S2Color and Shape:SolidMolecular weight:776.36BCTC
CAS:BCTC is a potent TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 (IC50 of 35 and 6 nM, respectively)Formula:C20H25ClN4OPurity:99.21%Color and Shape:SolidMolecular weight:372.89GSK 789472 hydrochloride
CAS:GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.Formula:C15H22ClN3OPurity:99.89%Color and Shape:SolidMolecular weight:295.81Neuropeptide EI, rat acetate
Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.Formula:C65H102N16O25Purity:95.55%Color and Shape:SolidMolecular weight:1507.6Nomifensine maleate
CAS:Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.
Formula:C20H22N2O4Purity:98.46%Color and Shape:SolidMolecular weight:354.4SB 242084 dihydrochloride
CAS:SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.Formula:C21H21Cl3N4O2Color and Shape:SolidMolecular weight:467.78Alimemazine hemitartrate
CAS:Alimemazine hemitartrate (Trimeprazine hemitartrate) is aphenothiazine derivative that is used as an antipruritic.Formula:C18H22N2SC4H6O6Purity:98.16% - 99.69%Color and Shape:SolidMolecular weight:448.53CYM-5520
CAS:CYM-5520 is a noncompetitive allosteric agonist of S1P2Formula:C21H19N3O2Purity:99.47%Color and Shape:SolidMolecular weight:345.39Ref: TM-T22703
1mg46.00€2mg60.00€5mg88.00€10mg135.00€25mg236.00€50mg354.00€100mg528.00€1mL*10mM (DMSO)98.00€Picotamide
CAS:Picotamide has anticoagulant and fibrinolytic properties.Formula:C21H20N4O3Purity:98.90%Color and Shape:SolidMolecular weight:376.41Ref: TM-T9153
1mg38.00€5mg92.00€10mg147.00€25mg241.00€50mg349.00€100mg479.00€200mg657.00€1mL*10mM (DMSO)94.00€Benorilate
CAS:Benorilate (Salipran) is the esterification product of paracetamol and acetylsalicylic acid with anti-inflammatory, analgesic and antipyretic properties.Formula:C17H15NO5Purity:98.39% - 99.85%Color and Shape:SolidMolecular weight:313.3Olcegepant
CAS:Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4Formula:C38H47Br2N9O5Purity:96.08% - 97.24%Color and Shape:SolidMolecular weight:869.65
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