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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5983 products of "GPCR/G-Protein"

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  • Alverine citrate

    CAS:
    Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.
    Formula:C26H35NO7
    Purity:98.53% - 99.43%
    Color and Shape:Coa
    Molecular weight:473.57

    Ref: TM-T0428

    1g
    58.00€
    5g
    92.00€
    10g
    130.00€
    500mg
    46.00€
    1mL*10mM (DMSO)
    49.00€
  • Clozapine

    CAS:
    Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.
    Formula:C18H19ClN4
    Purity:99.91% - 99.93%
    Color and Shape:Yellow Crystals From Acetone-Petroleum Ether Solid
    Molecular weight:326.82

    Ref: TM-T0455

    1g
    425.00€
    10mg
    34.00€
    25mg
    49.00€
    50mg
    66.00€
    100mg
    90.00€
    200mg
    161.00€
    500mg
    286.00€
    1mL*10mM (DMSO)
    44.00€
  • Vilazodone

    CAS:
    Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.
    Formula:C26H27N5O2
    Purity:99.61%
    Color and Shape:Light Yellow Solid
    Molecular weight:441.52

    Ref: TM-T1279

    1mg
    56.00€
    5mg
    118.00€
    10mg
    177.00€
    25mg
    250.00€
    50mg
    296.00€
    1mL*10mM (DMSO)
    143.00€
  • AB928

    CAS:
    AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].
    Formula:C23H22N8O
    Purity:98.09% - >99.99%
    Color and Shape:Solid
    Molecular weight:426.47

    Ref: TM-T14078

    1mg
    52.00€
    5mg
    117.00€
    10mg
    187.00€
    25mg
    369.00€
    50mg
    437.00€
    100mg
    628.00€
    1mL*10mM (DMSO)
    127.00€
  • Levodropropizine

    CAS:
    Levodropropizine ((S)-(-)-Dropropizine) is a histamine receptor inhibitor. It is used as an effective and very well tolerated peripheral antitussive drug.
    Formula:C13H20N2O2
    Purity:99.87% - 99.93%
    Color and Shape:White Or Off White Crystalline Powder
    Molecular weight:236.31

    Ref: TM-T0217

    2g
    34.00€
    5g
    52.00€
    1mL*10mM (DMSO)
    33.00€
  • MK-0812 Succinate

    CAS:
    MK-0812 Succinate is an effective and selective CCR2 antagonist.
    Formula:C28H40F3N3O7
    Purity:98.62% - 99.93%
    Color and Shape:Solid
    Molecular weight:587.63

    Ref: TM-T16091

    1mg
    62.00€
    5mg
    137.00€
    10mg
    250.00€
    25mg
    505.00€
    1mL*10mM (DMSO)
    170.00€
  • Timonacic

    CAS:
    Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.
    Formula:C4H7NO2S
    Purity:99.99%
    Color and Shape:Solid
    Molecular weight:133.17

    Ref: TM-T0221

    200mg
    33.00€
    1mL*10mM (DMSO)
    54.00€
  • Sumatriptan succinate

    CAS:
    Sumatriptan succinate (GR 43175), a serotonin1 (5-HT1) receptor agonist, is used in the acute treatment of a migraine headache.
    Formula:C18H27N3O6S
    Purity:97.53% - 99.51%
    Color and Shape:White Powder
    Molecular weight:413.49

    Ref: TM-T0203

    25mg
    34.00€
    50mg
    49.00€
    100mg
    71.00€
    500mg
    160.00€
  • Astressin acetate


    Astressin acetate is an antagonist of corticotropin releasing factor (CRF) with low affinity for the CRF binding protein and high affinity for the cloned
    Formula:C163H273N49O44
    Purity:96.87%
    Color and Shape:Solid
    Molecular weight:3623.21

    Ref: TM-TP1448L

    1mg
    225.00€
    5mg
    894.00€
    10mg
    1,339.00€
    25mg
    2,413.00€
  • Cloroperone

    CAS:
    Cloroperone has anxiolytic activity and may be used in the study of neurologic disorders.
    Formula:C22H23ClFNO2
    Purity:98.40%
    Color and Shape:Soild
    Molecular weight:387.88

    Ref: TM-T84304

    1mg
    175.00€
    5mg
    434.00€
    10mg
    622.00€
    25mg
    973.00€
    50mg
    1,341.00€
    100mg
    1,773.00€
  • Imidazolidinyl urea

    CAS:
    Imidazolidinyl urea (Imidurea) is an antimicrobial preservative used in cosmetics.
    Formula:C11H16N8O8
    Purity:98.6%
    Color and Shape:White Fluid Powder With Slight Characteristic Odor
    Molecular weight:388.29

    Ref: TM-T0430

    1g
    34.00€
    1mL*10mM (DMSO)
    33.00€
  • Pipamperone

    CAS:
    Pipamperone (McN-JR 3345) binds 5-HT2A closely as receptor.
    Formula:C21H30FN3O2
    Purity:99.85%
    Color and Shape:White Powder
    Molecular weight:375.48

    Ref: TM-T12480

    1mg
    58.00€
    2mg
    80.00€
    5mg
    113.00€
    10mg
    166.00€
    25mg
    268.00€
    50mg
    408.00€
    100mg
    590.00€
    1mL*10mM (DMSO)
    124.00€
  • Tolamolol

    CAS:
    Tolamolol is a selective β-adrenergic blocker that significantly reduces the degree of exercise-induced inhibition of the S-T segment and can be used in the
    Formula:C19H24N2O4
    Purity:98.59%
    Color and Shape:Solid
    Molecular weight:344.4

    Ref: TM-T68164

    1mg
    98.00€
    5mg
    180.00€
    10mg
    253.00€
    25mg
    455.00€
    50mg
    595.00€
    100mg
    883.00€
    500mg
    1,765.00€
  • Bisoprolol hemifumarate

    CAS:
    Bisoprolol, a selective beta-1 adrenergic receptor antagonist, selectively and competitively binds to and blocks beta-1 adrenergic receptors in the heart,
    Formula:C20H33NO6
    Purity:98.69% - 99.84%
    Color and Shape:White To Offf-White Powder
    Molecular weight:383.49

    Ref: TM-T0143

    50mg
    34.00€
    1mL*10mM (DMSO)
    35.00€
  • Dazmegrel HCl


    Dazmegrel HCl is a platelet thromboxane inhibitor used in the study of myocardial infarction and arrhythmias.
    Formula:C16H18ClN3O2
    Purity:98.30%
    Color and Shape:Solid
    Molecular weight:319.79

    Ref: TM-T31213L

    1mg
    109.00€
    2mg
    160.00€
    5mg
    261.00€
    10mg
    374.00€
    25mg
    583.00€
  • Olodaterol

    CAS:
    Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding and activating beta2-adrenergic receptors
    Formula:C21H26N2O5
    Purity:98.9%
    Color and Shape:Solid
    Molecular weight:386.45

    Ref: TM-T3457

    1mg
    47.00€
    5mg
    93.00€
  • Capeserod

    CAS:
    Capeserod is a potential 5-HT4 receptor (5-hydroxytryptamine receptor 4) agonist for the study of digestive disorders and neurological disorders.
    Formula:C23H25ClN4O4
    Purity:98.10% - 99.94%
    Color and Shape:Solid
    Molecular weight:456.92

    Ref: TM-T68035

    1mg
    175.00€
    5mg
    434.00€
    10mg
    622.00€
    25mg
    973.00€
    50mg
    1,341.00€
    100mg
    1,773.00€
  • Promethazine

    CAS:
    Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .
    Formula:C17H20N2S
    Purity:99.76%
    Color and Shape:Crystals
    Molecular weight:284.42

    Ref: TM-T0445

    5mg
    42.00€
    10mg
    52.00€
    25mg
    71.00€
    50mg
    102.00€
    100mg
    133.00€
    500mg
    303.00€
    1mL*10mM (DMSO)
    46.00€
  • Efloxate

    CAS:
    Efloxate (Angorlisin), a vasodilator, is utilized in the treatment of chronic coronary insufficiency.
    Formula:C19H16O5
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:324.33

    Ref: TM-T0151

    10mg
    48.00€
    25mg
    66.00€
  • Isoxsuprine hydrochloride

    CAS:
    Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
    Formula:C18H24ClNO3
    Purity:99.38%
    Color and Shape:Crystals From Water Solid
    Molecular weight:337.84

    Ref: TM-T0324

    200mg
    34.00€
    500mg
    49.00€
    1mL*10mM (DMSO)
    37.00€