GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,023 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5990 products of "GPCR/G-Protein"
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Tandospirone
CAS:Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.Formula:C21H29N5O2Purity:99.94%Color and Shape:SolidMolecular weight:383.49Ref: TM-TQ0315
2mg37.00€5mg54.00€1mL*10mM (DMSO)59.00€10mg87.00€25mg141.00€50mg193.00€100mg308.00€200mg441.00€Fenoprofen
CAS:Fenoprofen (LILLY-5385) is a non-steroidal anti-inflammatory compound and a modifier enhancer of the melanocortin receptor, increasing ERK1/2 activation.Formula:C15H14O3Purity:98.4%Color and Shape:SolidMolecular weight:242.27SID 7969543
CAS:SID 7969543 is a selective SF-1 inhibitor with potential anticancer activity, inhibits SF-1-triggered luciferase expression and can be used for cancer research.Formula:C24H24N2O7Purity:98.94%Color and Shape:SolidMolecular weight:452.46INCB 3284
CAS:INCB 3284, a potent human CCR2 antagonist with an IC50 of 3.7 nM, is researchable for acute liver failure and inhibits MCP-1/hCCR2 binding.Formula:C26H31F3N4O4Purity:97.81% - 99.42%Color and Shape:SolidMolecular weight:520.54ACT-462206
CAS:ACT-462206 is a Orexin 1/Orexin 2 receptor antagonist.ACT-462206 is highly potent and can be used to study sleep and anxiety.Formula:C20H24N2O4SPurity:99.45%Color and Shape:SolidMolecular weight:388.48Ref: TM-T26559
1mg42.00€1mL*10mM (DMSO)87.00€5mg88.00€10mg130.00€25mg264.00€50mg423.00€100mg670.00€500mg1,341.00€Atogepant
CAS:Atogepant (MK-8031) is an orally available, selective and potent calcitonin gene-related peptide receptor (CGRP) antagonist for the study of migraine.Formula:C29H23F6N5O3Purity:99.66%Color and Shape:SolidMolecular weight:603.52Ref: TM-T26682
1mg147.00€5mg250.00€10mg313.00€1mL*10mM (DMSO)334.00€25mg620.00€50mg1,108.00€100mg1,611.00€200mg2,178.00€Rizatriptan
CAS:Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.Formula:C15H19N5Purity:99.74%Color and Shape:SolidMolecular weight:269.35SB 243213
CAS:SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.Formula:C22H19F3N4O2Purity:98.78% - 99.86%Color and Shape:SolidMolecular weight:428.41LP-533401 hydrochloride
CAS:LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.Formula:C27H23ClF4N4O3Purity:98%Color and Shape:SolidMolecular weight:562.94Pentoxyverine
CAS:Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor.Formula:C20H31NO3Purity:97.11%Color and Shape:SolidMolecular weight:333.47A2ti-1
CAS:A2ti-1 is an annexin A2/S100A10 heterotetramer (A2t) inhibitor that inhibits Src activation and can be used to study human papillomavirus type 16 infection.Formula:C20H22N4O2SPurity:99.86%Color and Shape:SolidMolecular weight:382.48Ref: TM-T36432
1mg94.00€5mg200.00€1mL*10mM (DMSO)286.00€10mg313.00€25mg620.00€50mg982.00€100mg1,341.00€500mg2,682.00€Opipramol
CAS:Opipramol (Ensidon) is a compound with antidepressant activity, a sigma (σ) receptor agonist, and anxiolytic activity.Formula:C23H29N3OPurity:99.84% - 99.98%Color and Shape:SolidMolecular weight:363.5L-368,899 hydrochloride
CAS:L-368,899 hydrochloride is an OXTR antagonist that prevents oxytocin-induced antiabnormal pain and anti-nausea, and may be used in the study of depression.Formula:C26H43ClN4O5S2Purity:99.59%Color and Shape:SolidMolecular weight:591.23Ref: TM-T11794
2mg105.00€5mg147.00€1mL*10mM (DMSO)200.00€10mg230.00€25mg439.00€50mg685.00€100mg964.00€S-Methoprene
CAS:S-Methoprene (ZR2458), a juvenile hormone analog, acts as an insecticide influencing redox activity and male sex differentiation.
Formula:C19H34O3Purity:97.05% - 98.55%Color and Shape:SolidMolecular weight:310.47Atipamezole
CAS:Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.Formula:C14H16N2Purity:99.88%Color and Shape:Off-White To Light Yellow Crystal PowderMolecular weight:212.29(S)-Mirtazapine
CAS:(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.Formula:C17H19N3Purity:99.37%Color and Shape:SolidMolecular weight:265.35CGP 20712 A
CAS:CGP 20712 A (CGP 20712 mesylate) is a β1-adrenergic receptor antagonist with antihypertensive activity that reverses RKT-induced gastric relaxation.Formula:C24H29F3N4O8SPurity:99.37%Color and Shape:SolidMolecular weight:590.57Medetomidine
CAS:Medetomidine (MPV785 free base) is a selective α2-adrenoceptor agonist, with sedative and analgesic and vasoconstrictive hypoxic , in small animal anesthesia.Formula:C13H16N2Purity:99.88%Color and Shape:SolidMolecular weight:200.28Ref: TM-T21492
2mg38.00€5mg57.00€1mL*10mM (DMSO)62.00€10mg77.00€25mg128.00€50mg193.00€100mg290.00€200mg447.00€Rolofylline
CAS:Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.Formula:C20H28N4O2Purity:99.53%Color and Shape:SolidMolecular weight:356.465-LOX inhibitor
CAS:5-LOX inhibitor (1-(sec-Butyl)-4-(4-(4-(4-hydroxyphenyl)piperazin-1-yl)phenyl)-1H-1,2,4-triazol-5(4H)-one) is an itraconazole impurity, a LOX-5 inhibitor.Formula:C22H27N5O2Purity:98.01%Color and Shape:SolidMolecular weight:393.48
