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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5745 products of "GPCR/G-Protein"

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  • Aripiprazole Lauroxil
    Targetmol
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    Aripiprazole Lauroxil

    CAS:
    <p>Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.</p>
    Formula:C36H51Cl2N3O4
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:660.71

    Ref: TM-T14319

  • Asenapine Maleate
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    Asenapine Maleate

    CAS:
    Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken sublingually.
    Formula:C21H20ClNO5
    Purity:99.28%
    Color and Shape:Solid
    Molecular weight:401.84

    Ref: TM-T1951

  • PF-4348235 2HCl
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    PF-4348235 2HCl

    <p>PF-4348235 2HCl is an adrenergic agonist and muscarinic receptor antagonist, and is a bronchodilator.</p>
    Formula:C36H51Cl3N4O7S
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:790.24

    Ref: TM-T72226L1

  • Midodrine hydrochloride
    Targetmol
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    Midodrine hydrochloride

    CAS:
    <p>Midodrine, metabolized to desglymidodrine, activates alpha-1 receptors, raising blood pressure without CNS effects. It's a prodrug in hydrochloride form.</p>
    Formula:C12H19ClN2O4
    Purity:99.79% - >99.99%
    Color and Shape:Crystalline Solid
    Molecular weight:290.74

    Ref: TM-T1577

  • Isoxsuprine hydrochloride
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    Isoxsuprine hydrochloride

    CAS:
    Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.
    Formula:C18H24ClNO3
    Purity:99.38%
    Color and Shape:Crystals From Water Solid
    Molecular weight:337.84

    Ref: TM-T0324

  • Dapoxetine hydrochloride
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    Dapoxetine hydrochloride

    CAS:
    Dapoxetine hydrochloride (LY-210448 hydrochloride) is a selectivity short-acting serotonin reuptake inhibitor, used for the therapy of premature ejaculation.
    Formula:C21H23NO·HCl
    Purity:99.70% - 99.91%
    Color and Shape:White To Off-White Crystalline Solid
    Molecular weight:341.87

    Ref: TM-T6461

  • Ebalzotan
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    Ebalzotan

    CAS:
    <p>NAE-086 is a high-affinity and selective 5-HT(1A) receptor ligand with a K(i) value of 4.5 nM in membranes from rat hippocampus.</p>
    Formula:C19H30N2O2
    Purity:98.09% - 99.41%
    Color and Shape:Solid
    Molecular weight:318.45

    Ref: TM-T68059

  • Orforglipron
    Targetmol
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    Orforglipron

    CAS:
    Orforglipron (LY3502970; GLP-1 receptor agonist 1) is an orally available glucagon-like peptide (GLP-1) receptor agonist for the study of obesity and type 1
    Formula:C48H48F2N10O5
    Purity:99.47% - 99.8%
    Color and Shape:Solid
    Molecular weight:882.96

    Ref: TM-T11408

  • Labetalol hydrochloride
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    Labetalol hydrochloride

    CAS:
    <p>Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.</p>
    Formula:C19H25ClN2O3
    Purity:99.54% - 99.85%
    Color and Shape:Solid
    Molecular weight:364.87

    Ref: TM-T0348

  • ML-109
    Targetmol
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    ML-109

    CAS:
    <p>ML-109 is a potent agonist of thyroid stimulating hormone receptor (TSHR) (EC50 of 40 nM)</p>
    Formula:C31H29N3O5
    Purity:98.63%
    Color and Shape:Solid
    Molecular weight:523.58

    Ref: TM-T12073

  • Mirtazapine
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    Mirtazapine

    CAS:
    <p>Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.</p>
    Formula:C17H19N3
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:265.35

    Ref: TM-T0137

  • Chlorpheniramine maleate
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    Chlorpheniramine maleate

    CAS:
    <p>Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.</p>
    Formula:C20H23ClN2O4
    Purity:99.64% - 99.98%
    Color and Shape:Odorless White Crystalline Solid Or White Powder With A Bitter Taste
    Molecular weight:390.87

    Ref: TM-T1553

  • Efloxate
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    Efloxate

    CAS:
    <p>Efloxate (Angorlisin), a vasodilator, is utilized in the treatment of chronic coronary insufficiency.</p>
    Formula:C19H16O5
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:324.33

    Ref: TM-T0151

  • Bucumolol
    Targetmol
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    Bucumolol

    CAS:
    Bucumolol (Bucumarol) is a β-adrenergic blocking agent and a local anesthetic with antihypertensive activity and can be used to study myocardial infarction.
    Formula:C17H23NO4
    Purity:99.66%
    Color and Shape:Soild
    Molecular weight:305.37

    Ref: TM-T30606L

  • Dazmegrel HCl
    Targetmol
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    Dazmegrel HCl

    Dazmegrel HCl is a platelet thromboxane inhibitor used in the study of myocardial infarction and arrhythmias.
    Formula:C16H18ClN3O2
    Purity:98.30%
    Color and Shape:Solid
    Molecular weight:319.79

    Ref: TM-T31213L

  • AC265347
    Targetmol
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    AC265347

    CAS:
    <p>AC265347 is a potent calcium-sensitive receptor (CaSR) agonist and ago-PAM orthosteric modulator with antitumour activity for the study of neuroblastoma.</p>
    Formula:C17H17NOS
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:283.39

    Ref: TM-T29541

  • Azelastine hydrochloride
    Targetmol
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    Azelastine hydrochloride

    CAS:
    Azelastine hydrochloride (Astelin) is a phthalazinone derivative with antihistaminergic activity.
    Formula:C22H24ClN3O·HCl
    Purity:98% - >99.99%
    Color and Shape:White Crystalline Powder
    Molecular weight:418.36

    Ref: TM-T0211L

  • 2',5'-Dideoxyadenosine
    Targetmol
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    2',5'-Dideoxyadenosine

    CAS:
    2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).
    Formula:C10H13N5O2
    Purity:99.55%
    Color and Shape:White Solid
    Molecular weight:235.24

    Ref: TM-T10066

  • Mepyramine maleate
    Targetmol
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    Mepyramine maleate

    CAS:
    Mepyramine maleate is a mild hypnotic, local anesthetic, and H1 histamine antagonist for allergies and colds.
    Formula:C21H27N3O5
    Purity:99.51% - 99.7%
    Color and Shape:White Crystalline Powder
    Molecular weight:401.47

    Ref: TM-T1232

  • ML604086
    Targetmol
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    ML604086

    CAS:
    ML604086 suppresses CCL1 mediated chemotaxis and enhances intracellular Ca2 concentrations.
    Formula:C27H32N4O4S
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:508.63

    Ref: TM-T16111