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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5378 products of "GPCR/G-Protein"

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  • (R)-Elagolix
    Targetmol
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    (R)-Elagolix

    CAS:
    <p>(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.</p>
    Formula:C32H30F5N3O5
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:631.59

    Ref: TM-T11174

  • Noradrenaline bitartrate
    Targetmol
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    Noradrenaline bitartrate

    CAS:
    <p>Norepinephrine bitartrate acts directly on the α- and β-adrenergic receptors.</p>
    Formula:C12H19NO10
    Purity:99.53% - >99.99%
    Color and Shape:Solid
    Molecular weight:337.28

    Ref: TM-T0871

  • Phenothiazine
    Targetmol
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    Phenothiazine

    CAS:
    <p>Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.</p>
    Formula:C12H9NS
    Purity:99.95%
    Color and Shape:Yellow Solid Pellets
    Molecular weight:199.27

    Ref: TM-T0776

  • Venlafaxine hydrochloride
    Targetmol
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    Venlafaxine hydrochloride

    CAS:
    <p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>
    Formula:C17H28ClNO2
    Purity:97.32% - 99.86%
    Color and Shape:White Crystalline Powder
    Molecular weight:313.86

    Ref: TM-T0472

  • Urocortin (rat) acetate
    Targetmol
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    Urocortin (rat) acetate

    Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.
    Purity:97.76%
    Color and Shape:Soild

    Ref: TM-TP1020L

  • 2-Bromo-6-methoxynaphthalene
    Targetmol
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    2-Bromo-6-methoxynaphthalene

    CAS:
    <p>2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.</p>
    Formula:C11H9BrO
    Purity:98.51%
    Color and Shape:White To Off-White Powder
    Molecular weight:237.09

    Ref: TM-T0663

  • Ondansetron hydrochloride dihydrate
    Targetmol
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    Ondansetron hydrochloride dihydrate

    CAS:
    <p>Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.</p>
    Formula:C18H19N3O·HCl·2H2O
    Purity:99.92%
    Color and Shape:White Crystal Powder
    Molecular weight:365.86

    Ref: TM-T1478

  • CYM 50769
    Targetmol
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    CYM 50769

    CAS:
    <p>CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).</p>
    Formula:C24H17ClN2O3
    Purity:98% - 99.08%
    Color and Shape:Solid
    Molecular weight:416.86

    Ref: TM-T22702

  • Talastine
    Targetmol
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    Talastine

    CAS:
    <p>Talastine is an antihistamine compound that can induce an allergic rash.</p>
    Formula:C19H21N3O
    Purity:98.50% - 99.44%
    Color and Shape:Solid
    Molecular weight:307.39

    Ref: TM-T68150

  • hGPR91 antagonist 1
    Targetmol
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    hGPR91 antagonist 1

    CAS:
    <p>hGPR91 antagonist 1 is a potent and selective hGPR91 antagonist (IC50: 7 μM).</p>
    Formula:C31H23F4N3O
    Purity:98.89%
    Color and Shape:Solid
    Molecular weight:529.53

    Ref: TM-T11560

  • Roxatidine Acetate hydrochloride
    Targetmol
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    Roxatidine Acetate hydrochloride

    CAS:
    <p>Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.</p>
    Formula:C19H29ClN2O4
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:384.9

    Ref: TM-T0157

  • (3aR,9aR)-Fluparoxan
    Targetmol
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    (3aR,9aR)-Fluparoxan

    CAS:
    <p>(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Formula:C10H10FNO2
    Purity:97.82%
    Color and Shape:Soild
    Molecular weight:195.19

    Ref: TM-T77566

  • Lafutidine
    Targetmol
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    Lafutidine

    CAS:
    <p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>
    Formula:C22H29N3O4S
    Purity:98.55%
    Color and Shape:Yellowish White Crystalline Powder
    Molecular weight:431.55

    Ref: TM-T0081

  • AH 6809
    Targetmol
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    AH 6809

    CAS:
    <p>AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).</p>
    Formula:C17H14O5
    Purity:97.59%
    Color and Shape:Solid
    Molecular weight:298.29

    Ref: TM-T14148

  • Fluparoxan hydrochloride
    Targetmol
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    Fluparoxan hydrochloride

    CAS:
    <p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Formula:C10H11ClFNO2
    Purity:99.98%
    Color and Shape:Soild
    Molecular weight:231.65

    Ref: TM-T77565

  • Levosulpiride
    Targetmol
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    Levosulpiride

    CAS:
    <p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>
    Formula:C15H23N3O4S
    Purity:98.20% - 99.88%
    Color and Shape:White Crystalline Powder
    Molecular weight:341.43

    Ref: TM-T1211

  • Moxisylyte hydrochloride
    Targetmol
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    Moxisylyte hydrochloride

    CAS:
    Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
    Formula:C16H26ClNO3
    Purity:99.94% - ≥95%
    Color and Shape:Solid
    Molecular weight:315.84

    Ref: TM-T0394

  • Rimonabant
    Targetmol
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    Rimonabant

    CAS:
    <p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>
    Formula:C22H21Cl3N4O
    Purity:98% - 99.91%
    Color and Shape:White Or Almost White Crystalline Powder
    Molecular weight:463.79

    Ref: TM-T1519L

  • Aripiprazole
    Targetmol
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    Aripiprazole

    CAS:
    Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.
    Formula:C23H27Cl2N3O2
    Purity:99.43% - 99.62%
    Color and Shape:Colourless Flake Crystalline Solid
    Molecular weight:448.39

    Ref: TM-T1566

  • Quetiapine
    Targetmol
    + Info

    Quetiapine

    CAS:
    <p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>
    Formula:C21H25N3O2S
    Purity:99.14% - 99.63%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:383.51

    Ref: TM-T0162