
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,027 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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Isoetharine hydrochloride
CAS:Isoetharine HCl, a selective, short-acting oral β-agonist, is used as a bronchodilator for inhalation therapy.Formula:C13H22ClNO3Color and Shape:SolidMolecular weight:275.77Trimethaphan camsylate
CAS:Trimethaphan camsylate is a nicotinic antagonist that has been used as a ganglionic blocker in hypertension.Formula:C32H40N2O5S2Color and Shape:SolidMolecular weight:596.801Ro 23-3423
CAS:Ro 23-3423 is a specific inhibitor of thromboxane synthetase.Formula:C23H22N4O2Color and Shape:SolidMolecular weight:386.45Proxodolol hydrochloride
CAS:Proxodolol, a β-adrenergic receptor antagonist, is used potentially for the treatment of glaucoma, hypertension and angina.Formula:C17H26ClN3O4Color and Shape:SolidMolecular weight:371.86Opaganib HCl
CAS:ABC294640 (Opaganib) is an SK2 inhibitor with potential anti-cancer effects; it blocks S1P production to induce apoptosis.Formula:C23H26Cl2N2OColor and Shape:SolidMolecular weight:417.37Dicentrine HCl
CAS:Dicentrine HCl is the salt form of Dicentrine, an alpha 1-adrenoceptor antagonist effective against human hyperplastic prostates.Formula:C20H22ClNO4Color and Shape:SolidMolecular weight:375.85DH-97
CAS:DH-97 is a potent MT2 melatonin receptor antagonist (pKi value = 8.03).Formula:C22H26N2OColor and Shape:SolidMolecular weight:334.45Esreboxetine
CAS:Esreboxetine( PNU-165442, (S,S) -reboxetine) is a selective inhibitor of norepinephrine reuptake.Formula:C19H23NO3Color and Shape:SolidMolecular weight:313.39Bitolterol
CAS:Bitolterol is a new beta 2-adrenergic agonist and classified as a pro-drug.Formula:C28H31NO5Color and Shape:SolidMolecular weight:461.555-HT4 antagonist 1
CAS:5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).Formula:C23H36N4O5SPurity:99.75%Color and Shape:SolidMolecular weight:480.62Glucagon Receptor Antagonist I
CAS:Glucagon antagonist I blocks the GCGR (IC50=181 nM), stops glucagon-induced glycogenolysis, and lowers glucose in glucagon-treated humanized mice.Formula:C20H30N2OSColor and Shape:SolidMolecular weight:346.53Sch 44643
CAS:Sch 44643 is an antagonist of platelet activating factor with oral activity.Formula:C25H22ClN3O2Color and Shape:SolidMolecular weight:431.91Iferanserin HCl
CAS:Iferanserin HCl is a selective serotonin receptor antagonist.Formula:C23H29ClN2OColor and Shape:SolidMolecular weight:384.95GYKI-13380
CAS:GYKI-13380, also known as LS-79445, is a small molecule with potent bioactivity. Detail information has not been published yet.Formula:C16H22N2O3Color and Shape:SolidMolecular weight:290.36VER-3323
CAS:VER-3323 is a selective agonist for the 5-HT2B and 5-HT2C serotonin receptor with potent anorectic effects in animal studies.Formula:C11H15BrN2Purity:98%Color and Shape:SolidMolecular weight:255.15Reproterol hydrochloride
CAS:Reproterol hydrochloride, a β2 adrenoreceptor agonist, is used to treat asthma and chronic obstructive pulmonary disease (COPD).Formula:C18H24ClN5O5Purity:98%Color and Shape:SolidMolecular weight:425.87U 101958
CAS:U 101958 is a putative antipsychotic agent It is also a highly selective dopamine D4 receptor antagonist.Formula:C20H27N3OColor and Shape:SolidMolecular weight:325.45Fonazine hydrochloride
CAS:Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.Formula:C19H26ClN3O2S2Color and Shape:SolidMolecular weight:428.01Sch 40120
CAS:Sch 40120 is an inhibitor of 5-lipoxygenase.Formula:C18H15ClN2OPurity:98%Color and Shape:SolidMolecular weight:310.78MRS2690
CAS:MRS2690 is a potent P2Y14 receptor agonist (EC50 = 49 nM) that displays 7-fold higher potency than UDP-glucose.Formula:C15H24N2O16P2SColor and Shape:SolidMolecular weight:582.37
