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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6011 products of "GPCR/G-Protein"

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  • Isoetharine hydrochloride

    CAS:
    Isoetharine HCl, a selective, short-acting oral β-agonist, is used as a bronchodilator for inhalation therapy.
    Formula:C13H22ClNO3
    Color and Shape:Solid
    Molecular weight:275.77

    Ref: TM-T60502

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Trimethaphan camsylate

    CAS:
    Trimethaphan camsylate is a nicotinic antagonist that has been used as a ganglionic blocker in hypertension.
    Formula:C32H40N2O5S2
    Color and Shape:Solid
    Molecular weight:596.801

    Ref: TM-T68867

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Ro 23-3423

    CAS:
    Ro 23-3423 is a specific inhibitor of thromboxane synthetase.
    Formula:C23H22N4O2
    Color and Shape:Solid
    Molecular weight:386.45

    Ref: TM-T28569

    25mg
    1,369.00€
  • Proxodolol hydrochloride

    CAS:
    Proxodolol, a β-adrenergic receptor antagonist, is used potentially for the treatment of glaucoma, hypertension and angina.
    Formula:C17H26ClN3O4
    Color and Shape:Solid
    Molecular weight:371.86

    Ref: TM-T28457

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Opaganib HCl

    CAS:
    ABC294640 (Opaganib) is an SK2 inhibitor with potential anti-cancer effects; it blocks S1P production to induce apoptosis.
    Formula:C23H26Cl2N2O
    Color and Shape:Solid
    Molecular weight:417.37

    Ref: TM-T71301

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Dicentrine HCl

    CAS:
    Dicentrine HCl is the salt form of Dicentrine, an alpha 1-adrenoceptor antagonist effective against human hyperplastic prostates.
    Formula:C20H22ClNO4
    Color and Shape:Solid
    Molecular weight:375.85

    Ref: TM-T69075

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • DH-97

    CAS:
    DH-97 is a potent MT2 melatonin receptor antagonist (pKi value = 8.03).
    Formula:C22H26N2O
    Color and Shape:Solid
    Molecular weight:334.45

    Ref: TM-T69409

    1mg
    124.00€
  • Esreboxetine

    CAS:
    Esreboxetine( PNU-165442, (S,S) -reboxetine) is a selective inhibitor of norepinephrine reuptake.
    Formula:C19H23NO3
    Color and Shape:Solid
    Molecular weight:313.39

    Ref: TM-T31679

    25mg
    3,150.00€
    50mg
    4,725.00€
    100mg
    7,087.00€
  • Bitolterol

    CAS:
    Bitolterol is a new beta 2-adrenergic agonist and classified as a pro-drug.
    Formula:C28H31NO5
    Color and Shape:Solid
    Molecular weight:461.55

    Ref: TM-T69485

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 5-HT4 antagonist 1

    CAS:
    5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).
    Formula:C23H36N4O5S
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:480.62

    Ref: TM-T10169

    1mg
    60.00€
    5mg
    138.00€
    10mg
    200.00€
    25mg
    339.00€
    50mg
    484.00€
    100mg
    658.00€
    500mg
    1,324.00€
  • Glucagon Receptor Antagonist I

    CAS:
    Glucagon antagonist I blocks the GCGR (IC50=181 nM), stops glucagon-induced glycogenolysis, and lowers glucose in glucagon-treated humanized mice.
    Formula:C20H30N2OS
    Color and Shape:Solid
    Molecular weight:346.53

    Ref: TM-T37223

    1mg
    430.00€
    5mg
    1,549.00€
  • Sch 44643

    CAS:
    Sch 44643 is an antagonist of platelet activating factor with oral activity.
    Formula:C25H22ClN3O2
    Color and Shape:Solid
    Molecular weight:431.91

    Ref: TM-T28720

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Iferanserin HCl

    CAS:
    Iferanserin HCl is a selective serotonin receptor antagonist.
    Formula:C23H29ClN2O
    Color and Shape:Solid
    Molecular weight:384.95

    Ref: TM-T69905

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GYKI-13380

    CAS:
    GYKI-13380, also known as LS-79445, is a small molecule with potent bioactivity. Detail information has not been published yet.
    Formula:C16H22N2O3
    Color and Shape:Solid
    Molecular weight:290.36

    Ref: TM-T32027

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • VER-3323

    CAS:
    VER-3323 is a selective agonist for the 5-HT2B and 5-HT2C serotonin receptor with potent anorectic effects in animal studies.
    Formula:C11H15BrN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:255.15

    Ref: TM-T29103

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Reproterol hydrochloride

    CAS:
    Reproterol hydrochloride, a β2 adrenoreceptor agonist, is used to treat asthma and chronic obstructive pulmonary disease (COPD).
    Formula:C18H24ClN5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:425.87

    Ref: TM-T28519

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • U 101958

    CAS:
    U 101958 is a putative antipsychotic agent It is also a highly selective dopamine D4 receptor antagonist.
    Formula:C20H27N3O
    Color and Shape:Solid
    Molecular weight:325.45

    Ref: TM-T70263

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Fonazine hydrochloride

    CAS:
    Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.
    Formula:C19H26ClN3O2S2
    Color and Shape:Solid
    Molecular weight:428.01

    Ref: TM-T69407

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Sch 40120

    CAS:
    Sch 40120 is an inhibitor of 5-lipoxygenase.
    Formula:C18H15ClN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:310.78

    Ref: TM-T28718

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MRS2690

    CAS:
    MRS2690 is a potent P2Y14 receptor agonist (EC50 = 49 nM) that displays 7-fold higher potency than UDP-glucose.
    Formula:C15H24N2O16P2S
    Color and Shape:Solid
    Molecular weight:582.37

    Ref: TM-T68827

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€