GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,027 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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BGC-20-1531 free base
CAS:BGC-20-1531 (PGN 1531) free base is a selective and potent prostaglandin EP4 receptor antagonist (pKB: 7.6) that exhibits potential for migraine research.Formula:C26H24N2O6SColor and Shape:SolidMolecular weight:492.54DuP 734
CAS:DuP 734 is a potent and selective sigma receptor antagonist, functioning as a ligand for both sigma and 5-HT2 receptors, and exhibiting weak affinity towards D2 receptors. It possesses potential antipsychotic activity, potentially devoid of the motor side effects commonly observed with neuroleptics[1][2][3].Formula:C17H23BrFNOColor and Shape:SolidMolecular weight:356.279Donitriptan
CAS:Donitriptan 是一种 5-HT 受体激动剂，对 5-HT1B 和 5-HT1D 的 pKi 分别为 9.4 和 9.3。
Formula:C23H25N5O2Purity:98.76%Color and Shape:SolidMolecular weight:403.48CGP 35949
CAS:CGP 35949 is an LTD4 antagonist with phospholipase inhibitory activity.Formula:C23H25ClN5NaO5Purity:99.62%Color and Shape:SolidMolecular weight:509.92Ref: TM-T30828
1mg73.00€5mg149.00€1mL*10mM (DMSO)177.00€10mg213.00€25mg319.00€50mg447.00€100mg610.00€200mg823.00€PD 120697
CAS:PD 120697 is a dopamine antagonist with central dopamine agonist properties.Formula:C11H15N3SPurity:98%Color and Shape:SolidMolecular weight:221.32RG-12915
CAS:RG-12915 is a selective antagonist of 5-HT3(IC50 value of 0.16 nM).Formula:C20H25ClN2O2Purity:98%Color and Shape:SolidMolecular weight:360.88Nelonicline
CAS:Nelonicline is a selective agonist of neuronal nicotinic receptors.Formula:C17H19N3OSPurity:98%Color and Shape:SolidMolecular weight:313.42CB2 modulator 1
CAS:CB2 modulator 1 is a potent CB2 modulator. It can be used for the research for immune disorders, osteoporosis, inflammation, renal ischemia.Formula:C18H19F3N4O2Purity:99.6%Color and Shape:SolidMolecular weight:380.36Pridefine
CAS:Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.Formula:C19H21NPurity:99.15% - 99.66%Color and Shape:SolidMolecular weight:263.38Tedatioxetine hydrobromide
CAS:Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.Formula:C18H22BrNSPurity:99.65%Color and Shape:SolidMolecular weight:364.34UR-PI376
CAS:UR-PI376 is a selective histamine H4 receptor agonist with low H1/H2 activity and moderate H3 affinity.Formula:C17H22N6SColor and Shape:SolidMolecular weight:342.46VSN-16
CAS:VSN-16, a cannabinoid receptor agonist, is used potentially for the treatment of spasticity in multiple sclerosis.Formula:C18H26N2O3Color and Shape:SolidMolecular weight:318.41Way 100289
CAS:Way 100289 is a selective 5-HT3 receptor antagonist.Formula:C20H27N3O3Color and Shape:SolidMolecular weight:357.45PF-3246799
CAS:PF-3246799 is an effective and selective agonist of the 5-HT2C receptor.Formula:C15H17N3Purity:98%Color and Shape:SolidMolecular weight:239.32Impromidine
CAS:Impromidine is a highly potent and specific agonist of the histamine H2 receptor.Formula:C14H23N7SPurity:98%Color and Shape:SolidMolecular weight:321.44Vestipitant
CAS:Vestipitant (GW597599): a potent NK1 antagonist, may treat anxiety, depression, nausea, tinnitus, insomnia.Formula:C23H24F7N3OColor and Shape:SolidMolecular weight:491.45Avosentan
CAS:Avosentan（Ro 67-0565; SPP-301） is a potent endothelin receptor (ETA) antagonist.Cost-effective and quality-assured.Formula:C23H21N5O5SPurity:98.31% - 99.47%Color and Shape:SolidMolecular weight:479.51Tetrahydrozoline nitrate
CAS:Tetrahydrozoline, an imidazoline derivative, is an α-adrenergic agonist for nasal and eye congestion studies.Formula:C13H17N3O3Color and Shape:SolidMolecular weight:263.297A1AR antagonist 2
CAS:Compound 18h is a potent A1 adenosine receptor blocker with Ki of 1.49 nM for hA1, 10.2 nM for hA2A, 50.1 nM for hA2B.Formula:C17H12N4OColor and Shape:SolidMolecular weight:288.3Roxindole hydrochloride
CAS:Dopamine D2 autoreceptor agonistFormula:C23H27ClN2OPurity:98%Color and Shape:SolidMolecular weight:382.93
