
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,022 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5985 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
(R)-Carvedilol
CAS:(R)-Carvedilol is a non-selective blocker of β/α-1. (R)-Carvedilol exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).Formula:C24H26N2O4Purity:98%Color and Shape:SolidMolecular weight:406.47Zimelidine dihydrochloride
CAS:5-HT re-uptake inhibitorFormula:C16H18BrClN2Purity:98%Color and Shape:SolidMolecular weight:353.69GSK-215083
CAS:GSK-215083: a PET quinoline-based 5-HT6 antagonist radioligand, binds 5HT6 in striatum and 5HT2A in frontal cortex.Formula:C20H20FN3O2SColor and Shape:SolidMolecular weight:385.46JHW 007 hydrochloride
CAS:JHW 007 hydrochloride is a Dopamine uptake inhibitor.Formula:C24H30ClF2NOPurity:98%Color and Shape:SolidMolecular weight:421.95BMS-457
CAS:BMS-457 is a potent, CCR1-selective antagonist.Formula:C24H35ClN2O4Purity:98%Color and Shape:SolidMolecular weight:451BKM-570
CAS:BKM-570, a bradykinin antagonist, causes impressive growth inhibition of lung and prostate tumors.Formula:C34H34Cl2F5N3O3Purity:98%Color and Shape:SolidMolecular weight:698.55Antiplatelet agent 2
CAS:Antiplatelet agent 2 is a ticagrelor analogue that exhibits anti-platelet effects and can be used in platelet agglutination studies.Formula:C21H24F2N6O4SColor and Shape:SolidMolecular weight:494.51SB269652
CAS:SB269652 is the first drug-like allosteric modulator of the dopamine D2 receptor.Formula:C27H30N4OPurity:98%Color and Shape:SolidMolecular weight:426.55Apadenoson
CAS:Apadenoson: potent A2 agonist, A3 inhibitor (IC 45 nM), anti-inflammatory, for neurological research.Formula:C23H30N6O6Purity:98%Color and Shape:SolidMolecular weight:486.52VSN-16
CAS:VSN-16, a cannabinoid receptor agonist, is used potentially for the treatment of spasticity in multiple sclerosis.Formula:C18H26N2O3Color and Shape:SolidMolecular weight:318.41Indatraline hydrochloride
CAS:Inhibits transporters for 5-HT (SERT), dopamine (DAT) and noradrenalin (NET)Formula:C16H16Cl3NPurity:98%Color and Shape:SolidMolecular weight:328.66UR-PI376
CAS:UR-PI376 is a selective histamine H4 receptor agonist with low H1/H2 activity and moderate H3 affinity.Formula:C17H22N6SColor and Shape:SolidMolecular weight:342.46Cirazoline hydrochloride
CAS:Cirazoline hydrochloride is a synthetic competitive full agonist of α1A-AR (Ki 120 nM) and partial agonist at α1B-AR and α1D-AR.Formula:C13H17ClN2OPurity:99.863%Color and Shape:SolidMolecular weight:252.74Radioprotectin-1
CAS:Radioprotectin-1 is a selective agonist of LPA2 with EC50 of 25 nM for murine LPA2 GPCR and exerts radioprotective and radiomitigative action.Formula:C23H19ClN2O6SPurity:98.63% - 99.27%Color and Shape:SolidMolecular weight:486.92Ref: TM-T12684
1mg81.00€5mg170.00€1mL*10mM (DMSO)187.00€10mg259.00€25mg425.00€50mg562.00€100mg775.00€BAY-27-9955
CAS:BAY-27-9955 is a glucagon receptor antagonist.Formula:C23H31FOColor and Shape:SolidMolecular weight:342.49Alclofenac lysinate
CAS:Alclofenac is an anti-inflammatory agent used in the treatment of rheumatoid arthritis. It also used as an analgesic and an antipyretic.Formula:C17H25ClN2O5Purity:98%Color and Shape:SolidMolecular weight:372.84Dopamine D2 receptor antagonist-1
CAS:Dopamine D2 Receptor Antagonist-1 functions as a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R), demonstrating sub-millimolar affinity.Formula:C14H17N3SPurity:99.86%Color and Shape:SolidMolecular weight:259.37Ref: TM-T11077
1mg57.00€5mg120.00€1mL*10mM (DMSO)133.00€10mg178.00€25mg334.00€50mg492.00€100mg692.00€SB-226552
CAS:SB-226552 is an aryloxypropanolamine selective beta3AR agonist.Formula:C25H36NO5PColor and Shape:SolidMolecular weight:461.53NSC12404
CAS:NSC-12404 is a selective non-lipid LPA2/3 agonist.Formula:C21H13NO4Color and Shape:SolidMolecular weight:343.33B 4148
CAS:B 4148 is a bradykinin inhibitor.Formula:C62H95N19O14S2Color and Shape:SolidMolecular weight:1394.67
