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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5985 products of "GPCR/G-Protein"

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  • (R)-Carvedilol

    CAS:
    (R)-Carvedilol is a non-selective blocker of β/α-1. (R)-Carvedilol exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).
    Formula:C24H26N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:406.47

    Ref: TM-T12615

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Zimelidine dihydrochloride

    CAS:
    5-HT re-uptake inhibitor
    Formula:C16H18BrClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:353.69

    Ref: TM-T23560

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GSK-215083

    CAS:
    GSK-215083: a PET quinoline-based 5-HT6 antagonist radioligand, binds 5HT6 in striatum and 5HT2A in frontal cortex.
    Formula:C20H20FN3O2S
    Color and Shape:Solid
    Molecular weight:385.46

    Ref: TM-T27455

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • JHW 007 hydrochloride

    CAS:
    JHW 007 hydrochloride is a Dopamine uptake inhibitor.
    Formula:C24H30ClF2NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:421.95

    Ref: TM-T22877

    10mg
    770.00€
  • BMS-457

    CAS:
    BMS-457 is a potent, CCR1-selective antagonist.
    Formula:C24H35ClN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:451

    Ref: TM-T26849

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BKM-570

    CAS:
    BKM-570, a bradykinin antagonist, causes impressive growth inhibition of lung and prostate tumors.
    Formula:C34H34Cl2F5N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:698.55

    Ref: TM-T26833

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Antiplatelet agent 2

    CAS:
    Antiplatelet agent 2 is a ticagrelor analogue that exhibits anti-platelet effects and can be used in platelet agglutination studies.
    Formula:C21H24F2N6O4S
    Color and Shape:Solid
    Molecular weight:494.51

    Ref: TM-T63335

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • SB269652

    CAS:
    SB269652 is the first drug-like allosteric modulator of the dopamine D2 receptor.
    Formula:C27H30N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:426.55

    Ref: TM-T16857

    25mg
    1,288.00€
    50mg
    1,674.00€
    100mg
    2,250.00€
  • Apadenoson

    CAS:
    Apadenoson: potent A2 agonist, A3 inhibitor (IC 45 nM), anti-inflammatory, for neurological research.
    Formula:C23H30N6O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:486.52

    Ref: TM-T26641

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • VSN-16

    CAS:
    VSN-16, a cannabinoid receptor agonist, is used potentially for the treatment of spasticity in multiple sclerosis.
    Formula:C18H26N2O3
    Color and Shape:Solid
    Molecular weight:318.41

    Ref: TM-T29117

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Indatraline hydrochloride

    CAS:
    Inhibits transporters for 5-HT (SERT), dopamine (DAT) and noradrenalin (NET)
    Formula:C16H16Cl3N
    Purity:98%
    Color and Shape:Solid
    Molecular weight:328.66

    Ref: TM-T22867

    10mg
    567.00€
    50mg
    2,358.00€
  • UR-PI376

    CAS:
    UR-PI376 is a selective histamine H4 receptor agonist with low H1/H2 activity and moderate H3 affinity.
    Formula:C17H22N6S
    Color and Shape:Solid
    Molecular weight:342.46

    Ref: TM-T35003

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Cirazoline hydrochloride

    CAS:
    Cirazoline hydrochloride is a synthetic competitive full agonist of α1A-AR (Ki 120 nM) and partial agonist at α1B-AR and α1D-AR.
    Formula:C13H17ClN2O
    Purity:99.863%
    Color and Shape:Solid
    Molecular weight:252.74

    Ref: TM-T14972

    1mg
    60.00€
    5mg
    130.00€
    10mg
    192.00€
    25mg
    324.00€
    50mg
    480.00€
    100mg
    683.00€
    200mg
    888.00€
  • Radioprotectin-1

    CAS:
    Radioprotectin-1 is a selective agonist of LPA2 with EC50 of 25 nM for murine LPA2 GPCR and exerts radioprotective and radiomitigative action.
    Formula:C23H19ClN2O6S
    Purity:98.63% - 99.27%
    Color and Shape:Solid
    Molecular weight:486.92

    Ref: TM-T12684

    1mg
    81.00€
    5mg
    170.00€
    1mL*10mM (DMSO)
    187.00€
    10mg
    259.00€
    25mg
    425.00€
    50mg
    562.00€
    100mg
    775.00€
  • BAY-27-9955

    CAS:
    BAY-27-9955 is a glucagon receptor antagonist.
    Formula:C23H31FO
    Color and Shape:Solid
    Molecular weight:342.49

    Ref: TM-T30299

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • Alclofenac lysinate

    CAS:
    Alclofenac is an anti-inflammatory agent used in the treatment of rheumatoid arthritis. It also used as an analgesic and an antipyretic.
    Formula:C17H25ClN2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:372.84

    Ref: TM-T25035

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Dopamine D2 receptor antagonist-1

    CAS:
    Dopamine D2 Receptor Antagonist-1 functions as a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R), demonstrating sub-millimolar affinity.
    Formula:C14H17N3S
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:259.37

    Ref: TM-T11077

    1mg
    57.00€
    5mg
    120.00€
    1mL*10mM (DMSO)
    133.00€
    10mg
    178.00€
    25mg
    334.00€
    50mg
    492.00€
    100mg
    692.00€
  • SB-226552

    CAS:
    SB-226552 is an aryloxypropanolamine selective beta3AR agonist.
    Formula:C25H36NO5P
    Color and Shape:Solid
    Molecular weight:461.53

    Ref: TM-T28682

    25mg
    1,369.00€
  • NSC12404

    CAS:
    NSC-12404 is a selective non-lipid LPA2/3 agonist.
    Formula:C21H13NO4
    Color and Shape:Solid
    Molecular weight:343.33

    Ref: TM-T25885

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • B 4148

    CAS:
    B 4148 is a bradykinin inhibitor.
    Formula:C62H95N19O14S2
    Color and Shape:Solid
    Molecular weight:1394.67

    Ref: TM-T71571

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€