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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5984 products of "GPCR/G-Protein"

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  • Methyldopate hydrochloride

    CAS:
    Methyldopate HCl is an agent of antihypertensive.
    Formula:C12H18ClNO4
    Color and Shape:Solid
    Molecular weight:275.73

    Ref: TM-T20133

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SDZ NKT 343

    CAS:
    human tachykinin NK1 receptor antagonist
    Formula:C33H33N5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:579.65

    Ref: TM-T23345

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A2AR-antagonist-1

    CAS:
    Oral A2AR-antagonist-1, IC50 29 nM; anti-tumor, stable in mice (t1/2 86.1 min), boosts T cells, impedes LAG-3/TIM-3.
    Formula:C27H25N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:451.52

    Ref: TM-T72626

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Glucagon receptor antagonists-5

    CAS:
    Oral indazole-based glucagon antagonist, Ki: 32 nM, may treat type 2 diabetes.
    Formula:C30H29ClF3N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:572.02

    Ref: TM-T11416

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • RS 56812 hydrochloride

    CAS:
    5-HT3 partial agonist
    Formula:C18H22ClN3O2
    Purity:98.62%
    Color and Shape:Solid
    Molecular weight:347.84

    Ref: TM-T23264

    1mg
    62.00€
    2mg
    86.00€
    5mg
    127.00€
    10mg
    178.00€
    25mg
    416.00€
  • Cyclazosin HCl

    CAS:
    Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.
    Formula:C23H28ClN5O4
    Purity:99.10%
    Color and Shape:Solid
    Molecular weight:473.95

    Ref: TM-T70585

    1mg
    264.00€
    5mg
    650.00€
    10mg
    888.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
  • LY288513

    CAS:
    Selective CCK2 receptor antagonist
    Formula:C22H18BrN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:436.3

    Ref: TM-T22949

    10mg
    1,288.00€
    50mg
    5,544.00€
  • Guanfacine

    CAS:
    Guanfacine is a selective agonist of the α2A receptor.
    Formula:C9H9Cl2N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:246.09

    Ref: TM-T22824

    25mg
    103.00€
    50mg
    170.00€
    100mg
    261.00€
  • GSK-269984B

    CAS:
    GSK-269984B is a novel antagonist of EP1 receptor.
    Formula:C20H14Cl2FNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:406.23

    Ref: TM-T27466

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 2-CMDO

    CAS:
    2-CMDO is a Dopamine D2-like receptor antagonist.
    Formula:C23H23ClN2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:442.89

    Ref: TM-T22493

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Esreboxetine

    CAS:
    Esreboxetine( PNU-165442, (S,S) -reboxetine) is a selective inhibitor of norepinephrine reuptake.
    Formula:C19H23NO3
    Color and Shape:Solid
    Molecular weight:313.39

    Ref: TM-T31679

    25mg
    3,150.00€
    50mg
    4,725.00€
    100mg
    7,087.00€
  • Carbuterol hydrochloride

    CAS:
    Carbuterol hydrochloride is a short-acting β2 adrenoreceptor agonist.
    Formula:C13H22ClN3O3
    Color and Shape:Solid
    Molecular weight:303.79

    Ref: TM-T69394

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ranitidine bismuth citrate

    CAS:
    Ranitidine bismuth citrate, oral H2 blocker, IC50 3.3 µM, targets SARS-CoV-2 cells, treats H. pylori; MIC90 16 ng/L.
    Formula:C19H27BiN4O10S
    Color and Shape:Solid
    Molecular weight:712.48

    Ref: TM-T71059

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A 55453

    CAS:
    A 55453 is a radiated ionophore used as a reversibl, high-affinity alpha 1-adrenergic receptor probe.
    Formula:C25H32N6O3
    Color and Shape:Solid
    Molecular weight:464.56

    Ref: TM-T26421

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (Rac)-SEP-363856

    CAS:
    (Rac)-SEP-363856 is the racemate of SEP-363856. SEP-363856 is an orally active and CNS active psychotropic agent with a unique
    Formula:C9H13NOS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:183.27

    Ref: TM-T12677

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • FRG8701

    CAS:
    FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.
    Formula:C22H30N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:418.55

    Ref: TM-T11324

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • C-021 dihydrochloride

    CAS:
    C-021 dihydrochloride is a potent CCR4 antagonist. It potently inhibits functional chemotaxis in human and mouse with IC50s of 140 nM and 39 nM.
    Formula:C27H43Cl2N5O2
    Purity:98.67%
    Color and Shape:Solid
    Molecular weight:540.57

    Ref: TM-T10639

    1mg
    52.00€
    5mg
    97.00€
    1mL*10mM (DMSO)
    115.00€
    10mg
    154.00€
    25mg
    249.00€
    50mg
    374.00€
  • PD-135666

    CAS:
    PD-135666 is an antagonist of CCK receptor.
    Formula:C33H39N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:557.68

    Ref: TM-T28340

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • ADRA1D receptor antagonist 1 free base

    CAS:
    ADRA1D antagonist blocks bladder contractions; Ki=1.6 nM, IC30=15 nM, useful in overactive bladder research.
    Formula:C15H13ClN4O
    Color and Shape:Solid
    Molecular weight:300.74

    Ref: TM-T72091

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GAT228

    CAS:
    GAT228, an allosteric ligand for the cannabinoid receptor 1 (CB1), functions as the enantiomer of GAT211 [1].
    Formula:C22H18N2O2
    Color and Shape:Solid
    Molecular weight:342.39

    Ref: TM-T61105

    1mg
    118.00€
    10mg
    673.00€