
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,022 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5984 products of "GPCR/G-Protein"
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Methyldopate hydrochloride
CAS:Methyldopate HCl is an agent of antihypertensive.Formula:C12H18ClNO4Color and Shape:SolidMolecular weight:275.73SDZ NKT 343
CAS:human tachykinin NK1 receptor antagonistFormula:C33H33N5O5Purity:98%Color and Shape:SolidMolecular weight:579.65A2AR-antagonist-1
CAS:Oral A2AR-antagonist-1, IC50 29 nM; anti-tumor, stable in mice (t1/2 86.1 min), boosts T cells, impedes LAG-3/TIM-3.Formula:C27H25N5O2Purity:98%Color and Shape:SolidMolecular weight:451.52Glucagon receptor antagonists-5
CAS:Oral indazole-based glucagon antagonist, Ki: 32 nM, may treat type 2 diabetes.Formula:C30H29ClF3N3O3Purity:98%Color and Shape:SolidMolecular weight:572.02RS 56812 hydrochloride
CAS:5-HT3 partial agonistFormula:C18H22ClN3O2Purity:98.62%Color and Shape:SolidMolecular weight:347.84Cyclazosin HCl
CAS:Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.Formula:C23H28ClN5O4Purity:99.10%Color and Shape:SolidMolecular weight:473.95LY288513
CAS:Selective CCK2 receptor antagonistFormula:C22H18BrN3O2Purity:98%Color and Shape:SolidMolecular weight:436.3Guanfacine
CAS:Guanfacine is a selective agonist of the α2A receptor.Formula:C9H9Cl2N3OPurity:98%Color and Shape:SolidMolecular weight:246.09GSK-269984B
CAS:GSK-269984B is a novel antagonist of EP1 receptor.Formula:C20H14Cl2FNO3Purity:98%Color and Shape:SolidMolecular weight:406.232-CMDO
CAS:2-CMDO is a Dopamine D2-like receptor antagonist.Formula:C23H23ClN2O5Purity:98%Color and Shape:SolidMolecular weight:442.89Esreboxetine
CAS:Esreboxetine( PNU-165442, (S,S) -reboxetine) is a selective inhibitor of norepinephrine reuptake.Formula:C19H23NO3Color and Shape:SolidMolecular weight:313.39Carbuterol hydrochloride
CAS:Carbuterol hydrochloride is a short-acting β2 adrenoreceptor agonist.Formula:C13H22ClN3O3Color and Shape:SolidMolecular weight:303.79Ranitidine bismuth citrate
CAS:Ranitidine bismuth citrate, oral H2 blocker, IC50 3.3 µM, targets SARS-CoV-2 cells, treats H. pylori; MIC90 16 ng/L.Formula:C19H27BiN4O10SColor and Shape:SolidMolecular weight:712.48A 55453
CAS:A 55453 is a radiated ionophore used as a reversibl, high-affinity alpha 1-adrenergic receptor probe.Formula:C25H32N6O3Color and Shape:SolidMolecular weight:464.56(Rac)-SEP-363856
CAS:(Rac)-SEP-363856 is the racemate of SEP-363856. SEP-363856 is an orally active and CNS active psychotropic agent with a uniqueFormula:C9H13NOSPurity:98%Color and Shape:SolidMolecular weight:183.27FRG8701
CAS:FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.Formula:C22H30N2O4SPurity:98%Color and Shape:SolidMolecular weight:418.55C-021 dihydrochloride
CAS:C-021 dihydrochloride is a potent CCR4 antagonist. It potently inhibits functional chemotaxis in human and mouse with IC50s of 140 nM and 39 nM.Formula:C27H43Cl2N5O2Purity:98.67%Color and Shape:SolidMolecular weight:540.57PD-135666
CAS:PD-135666 is an antagonist of CCK receptor.Formula:C33H39N3O5Purity:98%Color and Shape:SolidMolecular weight:557.68ADRA1D receptor antagonist 1 free base
CAS:ADRA1D antagonist blocks bladder contractions; Ki=1.6 nM, IC30=15 nM, useful in overactive bladder research.Formula:C15H13ClN4OColor and Shape:SolidMolecular weight:300.74GAT228
CAS:GAT228, an allosteric ligand for the cannabinoid receptor 1 (CB1), functions as the enantiomer of GAT211 [1].Formula:C22H18N2O2Color and Shape:SolidMolecular weight:342.39
