GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(444 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(55 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5984 products of "GPCR/G-Protein"
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Molindone
CAS:Molindone: antipsychotic for schizophrenia; blocks dopamine, often paired with serotonin; dosage affects error/response rates.Formula:C16H24N2O2Purity:99.46% - 99.67%Color and Shape:Off-White SolidMolecular weight:276.37Landipirdine
CAS:Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders such as dementia.Formula:C18H19FN2O3SPurity:97.61% - 99.99%Color and Shape:SolidMolecular weight:362.422'-MeCCPA
CAS:2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.Formula:C16H22ClN5O4Purity:99.93%Color and Shape:SolidMolecular weight:383.83Felcisetrag
CAS:<p>Felcisetrag (TD-8954), an oral 5-HT4 agonist with GI prokinetic effects, has a high affinity (pKi 9.4) for h5-HT4(c) receptors.</p>Formula:C25H37N5O3Purity:99.99%Color and Shape:SolidMolecular weight:455.59Ticolubant
CAS:Ticolubant: Oral LTB4 antagonist, Ki=0.78 nM; blocks Ca2+ migration, IC50=6.6 nM; anti-inflammatory in mice.Formula:C23H19Cl2NO3SPurity:99.5%Color and Shape:SolidMolecular weight:460.37JTE-907
CAS:JTE-907 是一种具有高度选择性和口服活性的 CB2 受体反向激动剂。JTE-907在体内展现出抗炎活性。Formula:C24H26N2O6Purity:99.93%Color and Shape:SolidMolecular weight:438.47Ref: TM-T19705
1mg56.00€5mg126.00€10mg187.00€25mg329.00€50mg490.00€100mg700.00€1mL*10mM (DMSO)150.00€SB 699551 dihydrochloride
CAS:SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.Formula:C34H47Cl2N3OPurity:99.83%Color and Shape:SolidMolecular weight:584.66Ref: TM-T23325
1mg52.00€5mg111.00€10mg180.00€25mg311.00€50mg449.00€100mg615.00€1mL*10mM (DMSO)150.00€PSB-16133 sodium
CAS:PSB-16133 sodium is a selective P2Y purine receptor variant antagonist with an IC of 233 nM.Formula:C28H21N2NaO5S2Purity:98.03% - 98.93%Color and Shape:SolidMolecular weight:552.60Crinecerfont
CAS:Crinecerfont (SSR-125543) is a CRF1 antagonist, useful in congenital adrenal hyperplasia research.Formula:C27H28ClFN2OSPurity:97.79% - 98.55%Color and Shape:SolidMolecular weight:483.04Ecastolol
CAS:Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.Formula:C26H33N3O6Purity:99.89%Color and Shape:SolidMolecular weight:483.56Ref: TM-T11148
1mg369.00€5mg735.00€10mg938.00€25mg1,473.00€50mg1,882.00€100mg2,670.00€1mL*10mM (DMSO)929.00€Benperidol
CAS:Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.Formula:C22H24FN3O2Purity:99.91%Color and Shape:SolidMolecular weight:381.44Ref: TM-T26360
1mg116.00€5mg276.00€10mg410.00€25mg680.00€50mg938.00€100mg1,293.00€500mg2,593.00€1mL*10mM (DMSO)279.00€SB-209670
CAS:SB-209670 is a selective endothelin receptor antagonist that inhibits the activity of ET(B) receptors in rat vascular endothelium and vascular smooth muscle.Formula:C29H28O9Purity:98.29% - 99.40%Color and Shape:SolidMolecular weight:520.53Ref: TM-T34541
1mg333.00€5mg787.00€10mg1,074.00€25mg1,510.00€50mg1,882.00€100mg2,375.00€500mg4,655.00€1mL*10mM (DMSO)797.00€MLS1547
CAS:MLS1547 is a potent D2 receptor G protein-biased agonist (Ki=1.2 μM, EC50=0.37 μM in Ca2+ assay).Formula:C19H19ClN4OPurity:99.64%Color and Shape:SolidMolecular weight:354.83Enerisant hydrochloride
CAS:Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for P-gp, mediated by cytochrome P450 (CYP) and transporter proteinsFormula:C22H31ClN4O3Purity:99.95%Color and Shape:SolidMolecular weight:434.96L 651896
CAS:L 651896 is an inhibitor of 5-lipoxygenase.Formula:C18H18O3Purity:96.06% - 99.85%Color and Shape:SolidMolecular weight:282.33Lecozotan HCl
CAS:<p>Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.</p>Formula:C28H30ClN5O3Purity:99.04%Color and Shape:SolidMolecular weight:520.02BAY 60-6583
CAS:BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3Formula:C19H17N5O2SPurity:98.46% - 99.8%Color and Shape:SolidMolecular weight:379.44Ref: TM-T14506
1mg42.00€2mgTo inquire5mg88.00€10mg123.00€25mg245.00€50mg398.00€100mg597.00€200mg842.00€1mL*10mM (DMSO)106.00€LX-2931
CAS:LX-2931(LX-3305) is a sphingosine-1-phosphate cleavage enzyme (S1P) inhibitor for the treatment of rheumatoid arthritis.Formula:C9H15N3O5Purity:98.85% - 99.83%Color and Shape:SolidMolecular weight:245.23Egis-11150
CAS:Egis-11150 is a potent inhibitor of adrenergic alpha1, alpha2c, 5-HT2a, 5HT7 receptors.Formula:C19H21ClFN5O2Purity:97.49% - >99.99%Color and Shape:SolidMolecular weight:405.85Dabelotine
CAS:<p>Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.</p>Formula:C15H22N2O2Purity:98.55%Color and Shape:SolidMolecular weight:262.35
