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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5983 products of "GPCR/G-Protein"

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  • ANR 94

    CAS:
    ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.
    Formula:C9H13N5O
    Purity:98.9%
    Color and Shape:Solid
    Molecular weight:207.23

    Ref: TM-T22031

    5mg
    46.00€
    10mg
    71.00€
    25mg
    130.00€
    50mg
    219.00€
    100mg
    309.00€
    200mg
    434.00€
    1mL*10mM (DMSO)
    46.00€
  • Neldazosin

    CAS:
    Neldazosin is used as a potent α1-adrenoceptor antagonist.
    Formula:C18H25N5O4
    Purity:99.76% - 99.97%
    Color and Shape:Solid
    Molecular weight:375.42

    Ref: TM-T61535

    1mg
    117.00€
    5mg
    286.00€
    10mg
    414.00€
    25mg
    637.00€
    1mL*10mM (DMSO)
    299.00€
  • Milveterol HCl

    CAS:
    Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).
    Formula:C25H30ClN3O4
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:471.98

    Ref: TM-T33386

    1mg
    105.00€
    5mg
    249.00€
    10mg
    358.00€
    25mg
    605.00€
    50mg
    848.00€
    100mg
    1,099.00€
    200mg
    1,485.00€
  • Ecopipam

    CAS:
    Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over D2/D4/5-HT/α2a. For schizophrenia, obesity research.
    Formula:C19H20ClNO
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:313.82

    Ref: TM-T31602

    1mg
    50.00€
    5mg
    105.00€
    10mg
    172.00€
    25mg
    334.00€
    50mg
    537.00€
  • 4-PPBP maleate

    CAS:
    4-PPBP maleate: potent σ1 agonist, selective NR1a/2B NMDA antagonist, neuroprotective.
    Formula:C25H31NO4
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:409.52

    Ref: TM-T22513

    5mg
    35.00€
    10mg
    52.00€
    25mg
    95.00€
    50mg
    153.00€
    100mg
    219.00€
    200mg
    309.00€
    1mL*10mM (DMSO)
    43.00€
  • Impromidine hydrochloride

    CAS:
    Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.
    Formula:C14H26Cl3N7S
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:430.83

    Ref: TM-T68921

    1mg
    153.00€
    5mg
    365.00€
    10mg
    520.00€
    25mg
    780.00€
  • AM-1235

    CAS:
    AM-1235 is a potent and selective cannabinoid receptor CB1 agonist.
    Formula:C24H21FN2O3
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:404.43

    Ref: TM-T29930

    1mg
    315.00€
    5mg
    745.00€
    10mg
    1,018.00€
    25mg
    1,431.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Evodenoson

    CAS:
    Evodenoson (ATL313), a potent A2aR agonist, treats eye diseases, tumors, and immune disorders; potential for glaucoma and blood cancer studies.
    Formula:C23H29N7O6
    Purity:99.75% - 99.83%
    Color and Shape:Solid
    Molecular weight:499.52

    Ref: TM-T31731

    1mg
    225.00€
    5mg
    567.00€
    10mg
    855.00€
    25mg
    1,645.00€
    50mg
    2,215.00€
    100mg
    3,348.00€
  • GSK299115A

    CAS:
    GSK299115A (GSK-299115A) is a selective ROCK1 Inhibitor. GSK299115A exhibits IC50 of 8nM, 620nM, 560nM for ROCK1, RSK1, p70S6K, respectively.
    Formula:C20H16Cl2N4O2
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:415.27

    Ref: TM-T27471

    1mg
    303.00€
    5mg
    732.00€
    10mg
    1,018.00€
    25mg
    1,513.00€
    50mg
    2,035.00€
    100mg
    2,673.00€
    1mL*10mM (DMSO)
    895.00€
  • Ronacaleret HCl

    CAS:
    Ronacaleret HCl (SB-751689) is a small molecule CaSR antagonist for the treatment of endocrine and metabolic diseases, skin and musculoskeletal disorders.
    Formula:C25H32ClF2NO4
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:483.98

    Ref: TM-T34385

    1mg
    261.00€
    5mg
    642.00€
    10mg
    888.00€
    25mg
    1,333.00€
    50mg
    1,783.00€
    100mg
    2,457.00€
  • Pipoxazole

    CAS:
    Pipoxazole, an adrenergic receptor antagonist, is used potentially for the treatment of depression.
    Formula:C14H20N4O
    Purity:98.58% - 99.53%
    Color and Shape:Solid
    Molecular weight:260.33

    Ref: TM-T28419

    1mg
    164.00€
    5mg
    388.00€
    10mg
    532.00€
    25mg
    803.00€
  • Rezatomidine

    CAS:
    Rezatomidine (AGN203818) is a selective antagonist of α2-adrenergic receptor and can be used in studies about chronic pain, including neuropathic pain.
    Formula:C13H16N2S
    Purity:98.34%
    Color and Shape:Solid
    Molecular weight:232.34

    Ref: TM-T34308

    1mg
    175.00€
    2mg
    264.00€
    5mg
    404.00€
    10mg
    592.00€
    25mg
    888.00€
    50mg
    1,243.00€
    100mg
    1,701.00€
  • Nemazoline Free Base

    CAS:
    Nemazoline Free Base: a long-lasting nasal decongestant, better than oxymetazoline, with no systemic effects or toxicity in dogs and rats.
    Formula:C10H11Cl2N3
    Purity:98.06% - 98.83%
    Color and Shape:Solid
    Molecular weight:244.12

    Ref: TM-T71012

    1mg
    164.00€
    2mg
    234.00€
    5mg
    389.00€
    10mg
    532.00€
    25mg
    820.00€
  • Remogliflozin etabonate

    CAS:
    Remogliflozin etabonate is a prodrug SGLT2 inhibitor; Ki for hSGLT2: 1.95μM, rSGLT2: 2.14μM, rSGLT1: 8.57μM, hSGLT1: 43.1μM.
    Formula:C26H38N2O9
    Purity:98.98%
    Color and Shape:Solid
    Molecular weight:522.59

    Ref: TM-T34286

    2mg
    34.00€
    5mg
    50.00€
    10mg
    92.00€
    25mg
    156.00€
    50mg
    231.00€
    100mg
    323.00€
    200mg
    447.00€
    1mL*10mM (DMSO)
    58.00€
  • Egis-11150

    CAS:
    Egis-11150 is a potent inhibitor of adrenergic alpha1, alpha2c, 5-HT2a, 5HT7 receptors.
    Formula:C19H21ClFN5O2
    Purity:97.49% - >99.99%
    Color and Shape:Solid
    Molecular weight:405.85

    Ref: TM-T27248

    1mg
    164.00€
    5mg
    389.00€
    10mg
    532.00€
    25mg
    820.00€
  • Cilansetron

    CAS:
    Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.
    Formula:C20H21N3O
    Purity:99.82% - 99.98%
    Color and Shape:Solid
    Molecular weight:319.4

    Ref: TM-T27020

    1mg
    175.00€
    5mg
    434.00€
    10mg
    622.00€
    25mg
    973.00€
    50mg
    1,341.00€
    100mg
    1,773.00€
  • 5-HT6/7 antagonist 1

    CAS:

    5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.

    Formula:C22H20FN3O3
    Purity:98.78% - 99.26%
    Color and Shape:Solid
    Molecular weight:393.41

    Ref: TM-T61807

    1mg
    665.00€
    5mg
    1,681.00€
  • Quinupramine

    CAS:
    Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.
    Formula:C21H24N2
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:304.43

    Ref: TM-T60707

    1mg
    415.00€
    5mg
    964.00€
    25mg
    1,918.00€
    50mg
    2,502.00€
  • MRS1220

    CAS:
    MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeutic
    Formula:C21H14ClN5O2
    Purity:98.43%
    Color and Shape:Solid
    Molecular weight:403.82

    Ref: TM-T23016

    1mg
    50.00€
    5mg
    110.00€
    10mg
    168.00€
    25mg
    288.00€
    50mg
    414.00€
    100mg
    583.00€
    500mg
    To inquire
  • Nexopamil

    CAS:

    Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.

    Formula:C24H40N2O3
    Purity:97.87% - >99.99%
    Color and Shape:Solid
    Molecular weight:404.59

    Ref: TM-T28164

    1mg
    79.00€
    5mg
    170.00€
    10mg
    250.00€
    25mg
    415.00€
    50mg
    613.00€
    100mg
    873.00€
    200mg
    1,188.00€