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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5983 products of "GPCR/G-Protein"

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  • L-168049

    CAS:
    L-168049: Human glucagon receptor antagonist, IC50 - 3.7 nM human, 63 nM murine, 60 nM canine.
    Formula:C24H20BrClN2O
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:467.79

    Ref: TM-T22893

    1mg
    50.00€
    5mg
    105.00€
    10mg
    170.00€
    25mg
    358.00€
    50mg
    530.00€
    100mg
    758.00€
    500mg
    1,558.00€
    1mL*10mM (DMSO)
    116.00€
  • Remogliflozin etabonate

    CAS:
    Remogliflozin etabonate is a prodrug SGLT2 inhibitor; Ki for hSGLT2: 1.95μM, rSGLT2: 2.14μM, rSGLT1: 8.57μM, hSGLT1: 43.1μM.
    Formula:C26H38N2O9
    Purity:98.98%
    Color and Shape:Solid
    Molecular weight:522.59

    Ref: TM-T34286

    2mg
    34.00€
    5mg
    50.00€
    10mg
    92.00€
    25mg
    156.00€
    50mg
    231.00€
    100mg
    323.00€
    200mg
    447.00€
    1mL*10mM (DMSO)
    58.00€
  • Ensaculin

    CAS:
    Ensaculin, a benzopyrone-piperazine compound, enhances memory, protects neurons, and may treat dementia.
    Formula:C26H32N2O5
    Purity:99.56% - 99.81%
    Color and Shape:Solid
    Molecular weight:452.54

    Ref: TM-T67955

    1mg
    126.00€
    5mg
    304.00€
    10mg
    447.00€
    25mg
    733.00€
    50mg
    1,026.00€
    100mg
    1,388.00€
    500mg
    2,775.00€
  • ADR-851 free base

    CAS:
    ADR-851 free base is an antagonist of the HT3 receptor.
    Formula:C14H18ClN3O2
    Purity:97.88% - 98.39%
    Color and Shape:Solid
    Molecular weight:295.77

    Ref: TM-T23642

    1mg
    164.00€
    5mg
    389.00€
    10mg
    532.00€
    25mg
    820.00€
    50mg
    1,063.00€
    100mg
    1,423.00€
  • RS 67333 hydrochloride

    CAS:
    RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.
    Formula:C19H30Cl2N2O2
    Purity:98.78%
    Color and Shape:Solid
    Molecular weight:389.36

    Ref: TM-T23265

    10mg
    48.00€
    25mg
    96.00€
    50mg
    159.00€
    1mL*10mM (DMSO)
    34.00€
  • Lensiprazine

    CAS:
    Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder and
    Formula:C24H27FN4O2
    Purity:97.86%
    Color and Shape:Solid
    Molecular weight:422.5

    Ref: TM-T32633

    1mg
    84.00€
    5mg
    182.00€
    10mg
    259.00€
    25mg
    408.00€
    50mg
    580.00€
    100mg
    793.00€
    200mg
    1,063.00€
  • Dimethindene maleate

    CAS:
    Dimethindene maleate (SU 6518) is a histamine H1 antagonist and can be used in studies about the treatment of hypersensitivity reactions, pruritus and rhinitis.
    Formula:C24H28N2O4
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:408.49

    Ref: TM-T21472

    1mg
    34.00€
    5mg
    71.00€
    10mg
    105.00€
    25mg
    236.00€
    50mg
    313.00€
    100mg
    409.00€
    200mg
    582.00€
    1mL*10mM (DMSO)
    82.00€
  • A2A receptor antagonist 1

    CAS:
    A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
    Formula:C16H12FN5O
    Purity:99.52% - 99.93%
    Color and Shape:Solid
    Molecular weight:309.3

    Ref: TM-T37792

    2mg
    To inquire
    5mg
    62.00€
    10mg
    87.00€
    25mg
    183.00€
    50mg
    280.00€
    100mg
    416.00€
    200mg
    To inquire
    1mL*10mM (DMSO)
    47.00€
  • SC 19220

    CAS:
    SC 19220 is a prostaglandin E2 receptor EP1 antagonist that inhibits RANKL-induced osteoclastogenesis.
    Formula:C16H14ClN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:331.75

    Ref: TM-T23330

    1mg
    43.00€
    5mg
    93.00€
    10mg
    152.00€
    25mg
    298.00€
    50mg
    440.00€
    100mg
    627.00€
    200mg
    845.00€
    1mL*10mM (DMSO)
    92.00€
  • Pitolisant

    CAS:
    Pitolisant is a potent and selective nonimidazole inverse agonist that acts on the recombinant human histamine H3 receptor with Ki of 0.16 nM.
    Formula:C17H26ClNO
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:295.85

    Ref: TM-T60636

    5mg
    46.00€
    10mg
    66.00€
    25mg
    114.00€
    50mg
    178.00€
    100mg
    295.00€
    500mg
    708.00€
    1mL*10mM (DMSO)
    49.00€
  • Agomelatine hydrochloride

    CAS:
    Agomelatine HCl is a MT1/MT2 receptor agonist (Ki: 0.1-0.27 nM) and a 5-HT2C antagonist (pKi: 6.2-6.4).
    Formula:C15H18ClNO2
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:279.76

    Ref: TM-T60523

    10mg
    43.00€
    25mg
    70.00€
    50mg
    105.00€
    100mg
    135.00€
    500mg
    329.00€
    1mL*10mM (DMSO)
    34.00€
  • PPTN hydrochloride

    CAS:
    PPTN hydrochloride is a potent, high-affinity, competitive, highly selective P2Y14 receptor antagonist (KB: 434 pM), but no agonist or antagonist activity at
    Formula:C29H25ClF3NO2
    Purity:99.80%
    Color and Shape:Solid
    Molecular weight:511.96

    Ref: TM-T63534

    1mg
    46.00€
    5mg
    90.00€
    10mg
    152.00€
    25mg
    289.00€
    50mg
    447.00€
    100mg
    650.00€
    500mg
    1,369.00€
  • BMY-14802 hydrochloride

    CAS:
    BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.
    Formula:C18H23ClF2N4O
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:384.85

    Ref: TM-T22612

    5mg
    34.00€
    10mg
    50.00€
    25mg
    95.00€
    50mg
    161.00€
    100mg
    235.00€
    200mg
    333.00€
  • Compound C108

    CAS:

    Compound C108 is an inhibitor of GTPase-activating protein SH3 domain-binding protein 2 (G3BP2).

    Formula:C15H14N2O3
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:270.28

    Ref: TM-T38387

    1mg
    44.00€
    5mg
    89.00€
    10mg
    130.00€
    25mg
    251.00€
    50mg
    401.00€
    100mg
    597.00€
    200mg
    848.00€
  • DA-6886

    CAS:
    DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.
    Formula:C19H28Cl2N6O2
    Purity:99.91% - 99.99%
    Color and Shape:Solid
    Molecular weight:443.37

    Ref: TM-T27117

    1mg
    62.00€
    5mg
    132.00€
    10mg
    192.00€
    25mg
    314.00€
    50mg
    455.00€
    100mg
    622.00€
    200mg
    869.00€
  • Besipirdine

    CAS:
    Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic activity and cardiovascular activity.
    Formula:C16H17N3
    Purity:97.15% - 98.85%
    Color and Shape:Solid
    Molecular weight:251.33

    Ref: TM-T26778

    1mg
    164.00€
    5mg
    389.00€
    10mg
    532.00€
    25mg
    820.00€
  • MRS1220

    CAS:
    MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeutic
    Formula:C21H14ClN5O2
    Purity:98.43%
    Color and Shape:Solid
    Molecular weight:403.82

    Ref: TM-T23016

    1mg
    50.00€
    5mg
    110.00€
    10mg
    168.00€
    25mg
    288.00€
    50mg
    414.00€
    100mg
    583.00€
    500mg
    To inquire
  • RLX-33

    CAS:
    RLX-33 blocks RXFP3 and relaxin 3 effects, controls food intake in rats, and may help study metabolic syndrome.
    Formula:C24H19ClN4O4
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:462.89

    Ref: TM-T62929

    1mg
    78.00€
    5mg
    168.00€
    10mg
    269.00€
    25mg
    427.00€
    50mg
    610.00€
    100mg
    820.00€
    500mg
    1,603.00€
  • SPD-473 citrate

    CAS:
    SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.
    Formula:C23H31Cl2NO8S
    Purity:99.37%
    Color and Shape:Solid
    Molecular weight:552.47

    Ref: TM-T13898

    1mg
    138.00€
    5mg
    334.00€
    10mg
    469.00€
    25mg
    750.00€
    50mg
    1,009.00€
    100mg
    1,359.00€
  • 2'-MeCCPA

    CAS:
    2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.
    Formula:C16H22ClN5O4
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:383.83

    Ref: TM-T22489

    1mg
    35.00€
    5mg
    71.00€
    10mg
    123.00€
    25mg
    197.00€
    50mg
    301.00€
    100mg
    434.00€
    200mg
    615.00€