
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,018 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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L-168049
CAS:L-168049: Human glucagon receptor antagonist, IC50 - 3.7 nM human, 63 nM murine, 60 nM canine.Formula:C24H20BrClN2OPurity:>99.99%Color and Shape:SolidMolecular weight:467.79Ref: TM-T22893
1mg50.00€5mg105.00€10mg170.00€25mg358.00€50mg530.00€100mg758.00€500mg1,558.00€1mL*10mM (DMSO)116.00€Remogliflozin etabonate
CAS:Remogliflozin etabonate is a prodrug SGLT2 inhibitor; Ki for hSGLT2: 1.95μM, rSGLT2: 2.14μM, rSGLT1: 8.57μM, hSGLT1: 43.1μM.Formula:C26H38N2O9Purity:98.98%Color and Shape:SolidMolecular weight:522.59Ref: TM-T34286
2mg34.00€5mg50.00€10mg92.00€25mg156.00€50mg231.00€100mg323.00€200mg447.00€1mL*10mM (DMSO)58.00€Ensaculin
CAS:Ensaculin, a benzopyrone-piperazine compound, enhances memory, protects neurons, and may treat dementia.Formula:C26H32N2O5Purity:99.56% - 99.81%Color and Shape:SolidMolecular weight:452.54ADR-851 free base
CAS:ADR-851 free base is an antagonist of the HT3 receptor.Formula:C14H18ClN3O2Purity:97.88% - 98.39%Color and Shape:SolidMolecular weight:295.77RS 67333 hydrochloride
CAS:RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.Formula:C19H30Cl2N2O2Purity:98.78%Color and Shape:SolidMolecular weight:389.36Lensiprazine
CAS:Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder andFormula:C24H27FN4O2Purity:97.86%Color and Shape:SolidMolecular weight:422.5Dimethindene maleate
CAS:Dimethindene maleate (SU 6518) is a histamine H1 antagonist and can be used in studies about the treatment of hypersensitivity reactions, pruritus and rhinitis.Formula:C24H28N2O4Purity:99.79%Color and Shape:SolidMolecular weight:408.49Ref: TM-T21472
1mg34.00€5mg71.00€10mg105.00€25mg236.00€50mg313.00€100mg409.00€200mg582.00€1mL*10mM (DMSO)82.00€A2A receptor antagonist 1
CAS:A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.Formula:C16H12FN5OPurity:99.52% - 99.93%Color and Shape:SolidMolecular weight:309.3Ref: TM-T37792
2mgTo inquire5mg62.00€10mg87.00€25mg183.00€50mg280.00€100mg416.00€200mgTo inquire1mL*10mM (DMSO)47.00€SC 19220
CAS:SC 19220 is a prostaglandin E2 receptor EP1 antagonist that inhibits RANKL-induced osteoclastogenesis.Formula:C16H14ClN3O3Purity:98%Color and Shape:SolidMolecular weight:331.75Ref: TM-T23330
1mg43.00€5mg93.00€10mg152.00€25mg298.00€50mg440.00€100mg627.00€200mg845.00€1mL*10mM (DMSO)92.00€Pitolisant
CAS:Pitolisant is a potent and selective nonimidazole inverse agonist that acts on the recombinant human histamine H3 receptor with Ki of 0.16 nM.Formula:C17H26ClNOPurity:99.84%Color and Shape:SolidMolecular weight:295.85Ref: TM-T60636
5mg46.00€10mg66.00€25mg114.00€50mg178.00€100mg295.00€500mg708.00€1mL*10mM (DMSO)49.00€Agomelatine hydrochloride
CAS:Agomelatine HCl is a MT1/MT2 receptor agonist (Ki: 0.1-0.27 nM) and a 5-HT2C antagonist (pKi: 6.2-6.4).Formula:C15H18ClNO2Purity:99.57%Color and Shape:SolidMolecular weight:279.76PPTN hydrochloride
CAS:PPTN hydrochloride is a potent, high-affinity, competitive, highly selective P2Y14 receptor antagonist (KB: 434 pM), but no agonist or antagonist activity atFormula:C29H25ClF3NO2Purity:99.80%Color and Shape:SolidMolecular weight:511.96BMY-14802 hydrochloride
CAS:BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.Formula:C18H23ClF2N4OPurity:99.97%Color and Shape:SolidMolecular weight:384.85Compound C108
CAS:Compound C108 is an inhibitor of GTPase-activating protein SH3 domain-binding protein 2 (G3BP2).
Formula:C15H14N2O3Purity:99.77%Color and Shape:SolidMolecular weight:270.28DA-6886
CAS:DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.Formula:C19H28Cl2N6O2Purity:99.91% - 99.99%Color and Shape:SolidMolecular weight:443.37Besipirdine
CAS:Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic activity and cardiovascular activity.Formula:C16H17N3Purity:97.15% - 98.85%Color and Shape:SolidMolecular weight:251.33MRS1220
CAS:MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeuticFormula:C21H14ClN5O2Purity:98.43%Color and Shape:SolidMolecular weight:403.82RLX-33
CAS:RLX-33 blocks RXFP3 and relaxin 3 effects, controls food intake in rats, and may help study metabolic syndrome.Formula:C24H19ClN4O4Purity:99.89%Color and Shape:SolidMolecular weight:462.89SPD-473 citrate
CAS:SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.Formula:C23H31Cl2NO8SPurity:99.37%Color and Shape:SolidMolecular weight:552.472'-MeCCPA
CAS:2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.Formula:C16H22ClN5O4Purity:99.93%Color and Shape:SolidMolecular weight:383.83
