
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,018 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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ORM-10921
CAS:ORM-10921 is an α2C-adrenoceptor antagonist that has shown antipsychotic and antidepressant activity in animal studies.Formula:C18H23NO2Purity:99.46% - 99.98%Color and Shape:SolidMolecular weight:285.38Milenperone
CAS:Milenperone (R 34009) is a novel anti-invasive compound for the control of behavioral disorders in patients with epilepsy and alcoholism.Formula:C22H23ClFN3O2Purity:98.09% - 99.84%Color and Shape:SolidMolecular weight:415.89Egis-11150
CAS:Egis-11150 is a potent inhibitor of adrenergic alpha1, alpha2c, 5-HT2a, 5HT7 receptors.Formula:C19H21ClFN5O2Purity:97.49% - >99.99%Color and Shape:SolidMolecular weight:405.85Thiethylperazine dimaleate
CAS:Thiethylperazine dimaleate (Thiethylperazine maleate) is an antagonist of the D2 receptor and H1 receptor.Formula:C30H37N3O8S2Purity:99.88%Color and Shape:SolidMolecular weight:631.76LY 272015 hydrochloride
CAS:LY 272015 hydrochloride is a 5-HT2B receptor antagonist.Formula:C21H25ClN2O2Purity:99.47%Color and Shape:SolidMolecular weight:372.897-Hydroxy-DPAT hydrobromide
CAS:7-Hydroxy-DPAT hydrobromide is a D3 dopamine receptor agonist that blocks dopamine reuptake, used in research on neurological diseases.Formula:C16H26BrNOPurity:99.73%Color and Shape:SolidMolecular weight:328.29JTE-907
CAS:JTE-907 是一种具有高度选择性和口服活性的 CB2 受体反向激动剂。JTE-907在体内展现出抗炎活性。Formula:C24H26N2O6Purity:99.93%Color and Shape:SolidMolecular weight:438.47Ref: TM-T19705
1mg52.00€5mg119.00€10mg177.00€25mg313.00€50mg465.00€100mg662.00€1mL*10mM (DMSO)142.00€Seridopidine
CAS:Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy for schizophrenia, Parkinson's disease, and Tourette's syndrome.Formula:C14H20FNO2SPurity:99.77%Color and Shape:SolidMolecular weight:285.38N 0861
CAS:N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.Formula:C13H17N5Purity:98.78%Color and Shape:SolidMolecular weight:243.31Ref: TM-T70722
1mg164.00€2mg234.00€5mg389.00€10mg532.00€25mg820.00€50mg1,063.00€100mg1,423.00€200mg1,945.00€OPC-51803
CAS:OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of urinary incontinence and nocturia.Formula:C26H32ClN3O2Purity:98.93% - >99.99%Color and Shape:SolidMolecular weight:454CyPPA
CAS:CyPPA enhances SK channels, reducing firing rate and extending apamin-sensitive afterhyperpolarization.Formula:C16H23N5Purity:99.88%Color and Shape:SolidMolecular weight:285.39Ref: TM-T20968
2mg42.00€5mg62.00€10mg87.00€25mg166.00€50mg266.00€100mg442.00€500mg973.00€1mL*10mM (DMSO)66.00€BMS CCR2 22
CAS:BMS CCR2 22 is a potent and selective antagonist of CCR2 with calcium flux IC50 of 18 nM, chemotaxis IC50 of 1 nM, and binding IC50 of 5.1 nM.Formula:C28H34F3N5O4SPurity:99.65%Color and Shape:SolidMolecular weight:593.66Ref: TM-T14688
1mg55.00€5mg110.00€10mg173.00€25mg349.00€50mg532.00€100mg718.00€200mg964.00€1mL*10mM (DMSO)147.00€DF-1111301
CAS:DF-1111301 is a novel anti-allergic compound with anti-histamine H1 and anti-PAF activity.Formula:C15H25Cl2N3OPurity:99.17%Color and Shape:SolidMolecular weight:334.29Halopemide
CAS:Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).Formula:C21H22ClFN4O2Purity:96.57%Color and Shape:SolidMolecular weight:416.88Regrelor disodium
CAS:Regrelor disodium (INS 50589) is a p2y12 receptor antagonist that prevents thrombosis, effectively inhibits vascular smooth muscle cell contraction, inhibitsFormula:C22H23N6Na2O8PPurity:99.89%Color and Shape:SolidMolecular weight:576.41Ecastolol
CAS:Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.Formula:C26H33N3O6Purity:99.89%Color and Shape:SolidMolecular weight:483.56Ref: TM-T11148
1mg349.00€5mg697.00€10mg888.00€25mg1,395.00€50mg1,783.00€100mg2,530.00€1mL*10mM (DMSO)880.00€N6-(2-Phenylethyl)adenosine
CAS:N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM forFormula:C18H21N5O4Purity:99.83%Color and Shape:SolidMolecular weight:371.39Besipirdine
CAS:Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic activity and cardiovascular activity.Formula:C16H17N3Purity:97.15% - 98.85%Color and Shape:SolidMolecular weight:251.33LY-2624803
CAS:LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.Formula:C22H25N3O3Purity:99.78% - 99.97%Color and Shape:SolidMolecular weight:379.45K6PC-5
CAS:K6PC-5 is a ceramide derivative that acts as an activator of sphingosine kinase 1 (SPHK1), inducing a swift and temporary rise in intracellular calcium levels.Formula:C19H37NO4Purity:99.9%Color and Shape:SolidMolecular weight:343.5
