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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5983 products of "GPCR/G-Protein"

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  • ORM-10921

    CAS:
    ORM-10921 is an α2C-adrenoceptor antagonist that has shown antipsychotic and antidepressant activity in animal studies.
    Formula:C18H23NO2
    Purity:99.46% - 99.98%
    Color and Shape:Solid
    Molecular weight:285.38

    Ref: TM-T28267

    1mg
    358.00€
    5mg
    873.00€
    10mg
    1,161.00€
    25mg
    1,755.00€
    50mg
    2,358.00€
  • Milenperone

    CAS:
    Milenperone (R 34009) is a novel anti-invasive compound for the control of behavioral disorders in patients with epilepsy and alcoholism.
    Formula:C22H23ClFN3O2
    Purity:98.09% - 99.84%
    Color and Shape:Solid
    Molecular weight:415.89

    Ref: TM-T25813

    1mg
    264.00€
    5mg
    650.00€
    10mg
    888.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
  • Egis-11150

    CAS:
    Egis-11150 is a potent inhibitor of adrenergic alpha1, alpha2c, 5-HT2a, 5HT7 receptors.
    Formula:C19H21ClFN5O2
    Purity:97.49% - >99.99%
    Color and Shape:Solid
    Molecular weight:405.85

    Ref: TM-T27248

    1mg
    164.00€
    5mg
    389.00€
    10mg
    532.00€
    25mg
    820.00€
  • Thiethylperazine dimaleate

    CAS:
    Thiethylperazine dimaleate (Thiethylperazine maleate) is an antagonist of the D2 receptor and H1 receptor.
    Formula:C30H37N3O8S2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:631.76

    Ref: TM-T17072

    5mg
    50.00€
    10mg
    75.00€
    25mg
    124.00€
    50mg
    200.00€
    100mg
    309.00€
    500mg
    To inquire
  • LY 272015 hydrochloride

    CAS:
    LY 272015 hydrochloride is a 5-HT2B receptor antagonist.
    Formula:C21H25ClN2O2
    Purity:99.47%
    Color and Shape:Solid
    Molecular weight:372.89

    Ref: TM-T22948

    1mg
    47.00€
    5mg
    92.00€
    10mg
    152.00€
    25mg
    304.00€
    50mg
    497.00€
    100mg
    802.00€
  • 7-Hydroxy-DPAT hydrobromide

    CAS:
    7-Hydroxy-DPAT hydrobromide is a D3 dopamine receptor agonist that blocks dopamine reuptake, used in research on neurological diseases.
    Formula:C16H26BrNO
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:328.29

    Ref: TM-T22531

    1mg
    49.00€
    5mg
    94.00€
    10mg
    153.00€
    25mg
    246.00€
    50mg
    370.00€
  • JTE-907

    CAS:
    JTE-907 是一种具有高度选择性和口服活性的 CB2 受体反向激动剂。JTE-907在体内展现出抗炎活性。
    Formula:C24H26N2O6
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:438.47

    Ref: TM-T19705

    1mg
    52.00€
    5mg
    119.00€
    10mg
    177.00€
    25mg
    313.00€
    50mg
    465.00€
    100mg
    662.00€
    1mL*10mM (DMSO)
    142.00€
  • Seridopidine

    CAS:
    Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy for schizophrenia, Parkinson's disease, and Tourette's syndrome.
    Formula:C14H20FNO2S
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:285.38

    Ref: TM-T34616

    1mg
    132.00€
    5mg
    315.00€
    10mg
    477.00€
    25mg
    773.00€
    50mg
    1,063.00€
    100mg
    1,431.00€
    500mg
    2,872.00€
  • N 0861

    CAS:
    N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.
    Formula:C13H17N5
    Purity:98.78%
    Color and Shape:Solid
    Molecular weight:243.31

    Ref: TM-T70722

    1mg
    164.00€
    2mg
    234.00€
    5mg
    389.00€
    10mg
    532.00€
    25mg
    820.00€
    50mg
    1,063.00€
    100mg
    1,423.00€
    200mg
    1,945.00€
  • OPC-51803

    CAS:
    OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of urinary incontinence and nocturia.
    Formula:C26H32ClN3O2
    Purity:98.93% - >99.99%
    Color and Shape:Solid
    Molecular weight:454

    Ref: TM-T28257

    1mg
    213.00€
    5mg
    533.00€
    10mg
    858.00€
    25mg
    1,251.00€
  • CyPPA

    CAS:
    CyPPA enhances SK channels, reducing firing rate and extending apamin-sensitive afterhyperpolarization.
    Formula:C16H23N5
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:285.39

    Ref: TM-T20968

    2mg
    42.00€
    5mg
    62.00€
    10mg
    87.00€
    25mg
    166.00€
    50mg
    266.00€
    100mg
    442.00€
    500mg
    973.00€
    1mL*10mM (DMSO)
    66.00€
  • BMS CCR2 22

    CAS:
    BMS CCR2 22 is a potent and selective antagonist of CCR2 with calcium flux IC50 of 18 nM, chemotaxis IC50 of 1 nM, and binding IC50 of 5.1 nM.
    Formula:C28H34F3N5O4S
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:593.66

    Ref: TM-T14688

    1mg
    55.00€
    5mg
    110.00€
    10mg
    173.00€
    25mg
    349.00€
    50mg
    532.00€
    100mg
    718.00€
    200mg
    964.00€
    1mL*10mM (DMSO)
    147.00€
  • DF-1111301

    CAS:
    DF-1111301 is a novel anti-allergic compound with anti-histamine H1 and anti-PAF activity.
    Formula:C15H25Cl2N3O
    Purity:99.17%
    Color and Shape:Solid
    Molecular weight:334.29

    Ref: TM-T27159

    1mg
    164.00€
    2mg
    234.00€
    5mg
    389.00€
    10mg
    532.00€
    25mg
    820.00€
  • Halopemide

    CAS:
    Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).
    Formula:C21H22ClFN4O2
    Purity:96.57%
    Color and Shape:Solid
    Molecular weight:416.88

    Ref: TM-T15461

    1mg
    34.00€
    5mg
    85.00€
    10mg
    126.00€
    25mg
    245.00€
    50mg
    364.00€
    100mg
    530.00€
    1mL*10mM (DMSO)
    94.00€
  • Regrelor disodium

    CAS:
    Regrelor disodium (INS 50589) is a p2y12 receptor antagonist that prevents thrombosis, effectively inhibits vascular smooth muscle cell contraction, inhibits
    Formula:C22H23N6Na2O8P
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:576.41

    Ref: TM-T34280

    1mg
    85.00€
    5mg
    168.00€
    10mg
    240.00€
    25mg
    371.00€
    50mg
    513.00€
    100mg
    687.00€
    200mg
    928.00€
  • Ecastolol

    CAS:
    Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.
    Formula:C26H33N3O6
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:483.56

    Ref: TM-T11148

    1mg
    349.00€
    5mg
    697.00€
    10mg
    888.00€
    25mg
    1,395.00€
    50mg
    1,783.00€
    100mg
    2,530.00€
    1mL*10mM (DMSO)
    880.00€
  • N6-(2-Phenylethyl)adenosine

    CAS:
    N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for
    Formula:C18H21N5O4
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:371.39

    Ref: TM-T12163

    10mg
    33.00€
    25mg
    59.00€
    50mg
    104.00€
    100mg
    177.00€
    200mg
    316.00€
    1mL*10mM (DMSO)
    33.00€
  • Besipirdine

    CAS:
    Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic activity and cardiovascular activity.
    Formula:C16H17N3
    Purity:97.15% - 98.85%
    Color and Shape:Solid
    Molecular weight:251.33

    Ref: TM-T26778

    1mg
    164.00€
    5mg
    389.00€
    10mg
    532.00€
    25mg
    820.00€
  • LY-2624803

    CAS:
    LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.
    Formula:C22H25N3O3
    Purity:99.78% - 99.97%
    Color and Shape:Solid
    Molecular weight:379.45

    Ref: TM-T24421

    1mg
    133.00€
    5mg
    324.00€
    10mg
    477.00€
    25mg
    773.00€
    50mg
    1,063.00€
    100mg
    1,431.00€
    500mg
    2,872.00€
  • K6PC-5

    CAS:
    K6PC-5 is a ceramide derivative that acts as an activator of sphingosine kinase 1 (SPHK1), inducing a swift and temporary rise in intracellular calcium levels.
    Formula:C19H37NO4
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:343.5

    Ref: TM-T27710

    1mg
    38.00€
    5mg
    84.00€
    10mg
    119.00€
    25mg
    260.00€
    50mg
    424.00€
    100mg
    623.00€
    1mL*10mM (DMSO)
    93.00€