
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,018 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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FR-181157
CAS:FR-181157, a novel prostaglandin (PG) mimetic, shows high potency and agonist efficacy at the IP receptor and has good bioavailability.Formula:C30H27NNaO4Purity:98%Color and Shape:SolidMolecular weight:488.539APJ receptor agonist 6
CAS:APJ receptor agonist 6 is a potent agonist of the APJ (apelin receptor) (Ki: 0.059 μM). (EC50: 6.22 μM).Formula:C29H34FN3O5Color and Shape:SolidMolecular weight:523.6Velusetrag
CAS:Velusetrag(TD-5108), a potent 5-HT4 agonist, is in development for gastroparesis, constipation, and IBS.Formula:C25H36N4O5SColor and Shape:SolidMolecular weight:504.64Cipralisant maleate
CAS:Cipralisant maleate is a potent, selective Histamine H3 receptor antagonist.Formula:C18H24N2O4Color and Shape:SolidMolecular weight:332.39Aganepag isopropyl
CAS:Aganepag isopropyl can be used to treat Glaucoma.Formula:C27H37NO4SColor and Shape:SolidMolecular weight:471.65TA-1887
CAS:TA-1887: Selective SGLT2 inhibitor, treats type 2 diabetes, lowers glucose in high-fat diet mice, boosts UGE, has good pharmacokinetics.Formula:C24H26FNO5Color and Shape:SolidMolecular weight:427.47Satigrel
CAS:Satigrel is a new antiplatelet agent. It also inhibits platelet accumulation in prosthetic arterial grafts.Formula:C20H19NO4Purity:98%Color and Shape:SolidMolecular weight:337.37Pecavaptan
CAS:Pecavaptan is a vasopressin receptor antagonist.Formula:C22H19Cl2F3N6O3Color and Shape:SolidMolecular weight:543.33TASP0376377
CAS:TASP0376377 is a potent antagonist of CRTH2.Formula:C25H16Cl2N2O4Color and Shape:SolidMolecular weight:479.31GSK2263167
CAS:GSK2263167 is an agonist of S1P1 receptor.Formula:C25H26N4O4Color and Shape:SolidMolecular weight:446.5CP 154,526
CAS:CP 154,526 is a selective CRF1 receptor antagonist (Ki = 2.7 nM). CP 154,526 blocks CRF-induced activation of adenylate cyclase and the HPA axis.Formula:C23H32N4Color and Shape:SolidMolecular weight:364.53NBI-35965
CAS:NBI-35965 is a CRF1 receptor antagonist.
Formula:C21H22Cl2N4Color and Shape:SolidMolecular weight:401.33(R)-Casopitant
CAS:(R)-Casopitant ((R)-GW679769), an NK1-receptor antagonist, is used in chemotherapy-induced nausea research.Formula:C30H35F7N4O2Color and Shape:SolidMolecular weight:616.61Hedgehog IN-2
CAS:Hedgehog IN-2 (Compound 20) functions as an inhibitor of the Hedgehog signaling pathway, exhibiting an IC50 of <0.003 μM in C3H10T1/2 cells [1].Formula:C24H22N4O2Color and Shape:SolidMolecular weight:398.46RXFP1 receptor agonist-7
CAS:RXFP1 receptor agonist-7 (Example 2) serves as an RXFP1 receptor agonist, effectively inhibiting cAMP production in HEK293 cells that stably express the humanFormula:C40H32F5N3O7Color and Shape:SolidMolecular weight:761.69Y1R probe-1
CAS:Compound 39, or Y1R probe-1, is a fluorescent probe for Neuropeptide Y Y1 Receptor used in cancer research.Formula:C64H71F3N10O12Color and Shape:SolidMolecular weight:1229.3CCR4 antagonist 4
CAS:CCR4 Antagonist 4 (Compound 22) is a potent and selective antagonist of the CC chemokine receptor-4 (CCR4), displaying an IC50 value of 0.02 μM. It also inhibits MDC-mediated chemotaxis and Ca2+ mobilization, with IC50 values of 0.007 μM and 0.003 μM, respectively. This compound is utilized in research on allergic inflammation [1].Formula:C24H27Cl2N7OColor and Shape:SolidMolecular weight:500.42ABT-702 hydrochloride
CAS:ABT-702 hydrochloride effectively inhibits adenosine kinase, exhibiting an IC50 value of 1.7 nM [1] [2].Formula:C22H20BrClN6OColor and Shape:SolidMolecular weight:499.79COR659
CAS:COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.Formula:C16H16ClNO3SPurity:99.75%Color and Shape:SolidMolecular weight:337.82Ref: TM-T36520
1mg38.00€5mg86.00€10mg123.00€25mg215.00€50mg299.00€100mg411.00€200mg560.00€1mL*10mM (DMSO)94.00€Macimorelin acetate
CAS:Macimorelin acetate (EP-1572) is an oral GHSR agonist for AGHD and CACS research.Formula:C28H34N6O5Color and Shape:SolidMolecular weight:534.61

