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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5983 products of "GPCR/G-Protein"

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  • FR-181157

    CAS:
    FR-181157, a novel prostaglandin (PG) mimetic, shows high potency and agonist efficacy at the IP receptor and has good bioavailability.
    Formula:C30H27NNaO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:488.539

    Ref: TM-T27373

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€
  • APJ receptor agonist 6

    CAS:
    APJ receptor agonist 6 is a potent agonist of the APJ (apelin receptor) (Ki: 0.059 μM). (EC50: 6.22 μM).
    Formula:C29H34FN3O5
    Color and Shape:Solid
    Molecular weight:523.6

    Ref: TM-T63669

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • Velusetrag

    CAS:
    Velusetrag(TD-5108), a potent 5-HT4 agonist, is in development for gastroparesis, constipation, and IBS.
    Formula:C25H36N4O5S
    Color and Shape:Solid
    Molecular weight:504.64

    Ref: TM-T35046

    25mg
    1,026.00€
    50mg
    1,341.00€
    100mg
    2,025.00€
  • Cipralisant maleate

    CAS:
    Cipralisant maleate is a potent, selective Histamine H3 receptor antagonist.
    Formula:C18H24N2O4
    Color and Shape:Solid
    Molecular weight:332.39

    Ref: TM-T27022

    25mg
    1,773.00€
    50mg
    2,322.00€
    100mg
    3,060.00€
  • Aganepag isopropyl

    CAS:
    Aganepag isopropyl can be used to treat Glaucoma.
    Formula:C27H37NO4S
    Color and Shape:Solid
    Molecular weight:471.65

    Ref: TM-T29708

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€
  • TA-1887

    CAS:
    TA-1887: Selective SGLT2 inhibitor, treats type 2 diabetes, lowers glucose in high-fat diet mice, boosts UGE, has good pharmacokinetics.
    Formula:C24H26FNO5
    Color and Shape:Solid
    Molecular weight:427.47

    Ref: TM-T34767

    25mg
    1,773.00€
    50mg
    2,322.00€
    100mg
    3,060.00€
  • Satigrel

    CAS:
    Satigrel is a new antiplatelet agent. It also inhibits platelet accumulation in prosthetic arterial grafts.
    Formula:C20H19NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:337.37

    Ref: TM-T24760

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€
  • Pecavaptan

    CAS:
    Pecavaptan is a vasopressin receptor antagonist.
    Formula:C22H19Cl2F3N6O3
    Color and Shape:Solid
    Molecular weight:543.33

    Ref: TM-T70066

    25mg
    3,970.00€
    50mg
    5,518.00€
    100mg
    7,444.00€
  • TASP0376377

    CAS:
    TASP0376377 is a potent antagonist of CRTH2.
    Formula:C25H16Cl2N2O4
    Color and Shape:Solid
    Molecular weight:479.31

    Ref: TM-T28925

    25mg
    1,773.00€
    50mg
    2,322.00€
    100mg
    3,060.00€
  • GSK2263167

    CAS:
    GSK2263167 is an agonist of S1P1 receptor.
    Formula:C25H26N4O4
    Color and Shape:Solid
    Molecular weight:446.5

    Ref: TM-T27459

    25mg
    1,908.00€
    50mg
    2,502.00€
    100mg
    3,330.00€
  • CP 154,526

    CAS:
    CP 154,526 is a selective CRF1 receptor antagonist (Ki = 2.7 nM). CP 154,526 blocks CRF-induced activation of adenylate cyclase and the HPA axis.
    Formula:C23H32N4
    Color and Shape:Solid
    Molecular weight:364.53

    Ref: TM-T27057

    25mg
    1,639.00€
    50mg
    2,142.00€
    100mg
    2,790.00€
  • NBI-35965

    CAS:

    NBI-35965 is a CRF1 receptor antagonist.

    Formula:C21H22Cl2N4
    Color and Shape:Solid
    Molecular weight:401.33

    Ref: TM-T69544

    25mg
    2,015.00€
    50mg
    2,642.00€
    100mg
    3,515.00€
  • (R)-Casopitant

    CAS:
    (R)-Casopitant ((R)-GW679769), an NK1-receptor antagonist, is used in chemotherapy-induced nausea research.
    Formula:C30H35F7N4O2
    Color and Shape:Solid
    Molecular weight:616.61

    Ref: TM-T72820

    25mg
    1,198.00€
    50mg
    1,566.00€
    100mg
    2,502.00€
  • Hedgehog IN-2

    CAS:
    Hedgehog IN-2 (Compound 20) functions as an inhibitor of the Hedgehog signaling pathway, exhibiting an IC50 of <0.003 μM in C3H10T1/2 cells [1].
    Formula:C24H22N4O2
    Color and Shape:Solid
    Molecular weight:398.46

    Ref: TM-T79055

    5mg
    To inquire
    50mg
    To inquire
  • RXFP1 receptor agonist-7

    CAS:
    RXFP1 receptor agonist-7 (Example 2) serves as an RXFP1 receptor agonist, effectively inhibiting cAMP production in HEK293 cells that stably express the human
    Formula:C40H32F5N3O7
    Color and Shape:Solid
    Molecular weight:761.69

    Ref: TM-T81240

    5mg
    To inquire
    50mg
    To inquire
  • Y1R probe-1

    CAS:
    Compound 39, or Y1R probe-1, is a fluorescent probe for Neuropeptide Y Y1 Receptor used in cancer research.
    Formula:C64H71F3N10O12
    Color and Shape:Solid
    Molecular weight:1229.3

    Ref: TM-T74459

    5mg
    To inquire
    50mg
    To inquire
  • CCR4 antagonist 4

    CAS:
    CCR4 Antagonist 4 (Compound 22) is a potent and selective antagonist of the CC chemokine receptor-4 (CCR4), displaying an IC50 value of 0.02 μM. It also inhibits MDC-mediated chemotaxis and Ca2+ mobilization, with IC50 values of 0.007 μM and 0.003 μM, respectively. This compound is utilized in research on allergic inflammation [1].
    Formula:C24H27Cl2N7O
    Color and Shape:Solid
    Molecular weight:500.42

    Ref: TM-T84701

    10mg
    To inquire
    50mg
    To inquire
  • ABT-702 hydrochloride

    CAS:
    ABT-702 hydrochloride effectively inhibits adenosine kinase, exhibiting an IC50 value of 1.7 nM [1] [2].
    Formula:C22H20BrClN6O
    Color and Shape:Solid
    Molecular weight:499.79

    Ref: TM-T84880

    10mg
    To inquire
    50mg
    To inquire
  • COR659

    CAS:
    COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.
    Formula:C16H16ClNO3S
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:337.82

    Ref: TM-T36520

    1mg
    38.00€
    5mg
    86.00€
    10mg
    123.00€
    25mg
    215.00€
    50mg
    299.00€
    100mg
    411.00€
    200mg
    560.00€
    1mL*10mM (DMSO)
    94.00€
  • Macimorelin acetate

    CAS:
    Macimorelin acetate (EP-1572) is an oral GHSR agonist for AGHD and CACS research.
    Formula:C28H34N6O5
    Color and Shape:Solid
    Molecular weight:534.61

    Ref: TM-T68276

    25mg
    475.00€
    50mg
    765.00€
    100mg
    1,223.00€