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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5985 products of "GPCR/G-Protein"

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  • SB-423562

    CAS:
    SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.
    Formula:C26H32N2O4
    Purity:99.22%
    Color and Shape:Solid
    Molecular weight:436.54

    Ref: TM-T12846

    1mg
    37.00€
    5mg
    80.00€
    10mg
    119.00€
    25mg
    210.00€
    50mg
    319.00€
    100mg
    442.00€
    200mg
    605.00€
    1mL*10mM (DMSO)
    89.00€
  • AZD5462

    CAS:
    AZD5462 is a potent orally available relaxin receptor RXFP1 agonist for the study of heart failure and cancer.
    Formula:C30H41FN2O6
    Purity:98.32% - 99.63%
    Color and Shape:Solid
    Molecular weight:544.65

    Ref: TM-T63838

    1mg
    354.00€
    5mg
    850.00€
    10mg
    1,206.00€
    25mg
    1,882.00€
    50mg
    2,642.00€
    100mg
    3,345.00€
  • LSN3318839

    CAS:
    <p>LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can</p>
    Formula:C26H23Cl2N3O2
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:480.39

    Ref: TM-T63166

    1mg
    202.00€
    5mg
    512.00€
    10mg
    738.00€
    25mg
    1,121.00€
    50mg
    1,510.00€
    100mg
    2,062.00€
  • Vofopitant

    CAS:
    Vofopitant (GR 205171) is a potent NK1 receptor antagonist with anxiolytic and antiemetic activity for the study of post-traumatic stress disorder (PTSD).
    Formula:C21H23F3N6O
    Purity:97.86%
    Color and Shape:Solid
    Molecular weight:432.44

    Ref: TM-T13329

    1mg
    99.00€
    5mg
    235.00€
    10mg
    349.00€
    25mg
    565.00€
    50mg
    818.00€
    100mg
    1,103.00€
    500mg
    2,205.00€
  • Vofopitant dihydrochloride

    CAS:
    Vofopitant dihydrochloride (GR 205171A) is a tachykinin NK1 receptor antagonist and a potential compound for the treatment of pathologic vomiting.
    Formula:C21H25Cl2F3N6O
    Purity:98.99%
    Color and Shape:Solid
    Molecular weight:505.36

    Ref: TM-T13329L

    1mg
    99.00€
    5mg
    235.00€
    10mg
    376.00€
    25mg
    712.00€
    50mg
    1,064.00€
    100mg
    1,454.00€
    500mg
    2,822.00€
    1mL*10mM (DMSO)
    261.00€
  • PF-07258669

    CAS:
    PF-07258669 is a selective melanocortin 4 receptor (MC4) antagonist used in the study of cachexia and loss of appetite.
    Formula:C25H27FN6O2
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:462.52

    Ref: TM-T69526

    1mg
    802.00€
    5mg
    1,605.00€
    10mg
    2,612.00€
    25mg
    5,159.00€
    50mg
    8,255.00€
  • Dersimelagon

    CAS:
    Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist.Cost-effective and quality-assured.
    Formula:C36H45F4N3O5
    Purity:97.35% - 98.23%
    Color and Shape:Solid
    Molecular weight:675.75

    Ref: TM-T25310

    1mg
    79.00€
    5mg
    180.00€
    10mg
    264.00€
    25mg
    452.00€
    50mg
    647.00€
  • BMS-986141

    CAS:
    BMS-986141(UDM-003183) is a selective and potent protease-activated receptor-4 (PAR-4) antagonist with oral activity and an IC50 value of 0.4 nM.BMS-98614
    Formula:C27H23N5O5S2
    Purity:98.43% - 99.26%
    Color and Shape:Solid
    Molecular weight:561.63

    Ref: TM-T63966

    1mg
    612.00€
    5mg
    1,216.00€
    10mg
    1,549.00€
    25mg
    2,213.00€
  • SB-224289 hydrochloride

    CAS:
    SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.
    Formula:C32H33ClN4O3
    Purity:98.99% - 99.96%
    Color and Shape:Solid
    Molecular weight:557.08

    Ref: TM-T12841

    1mg
    42.00€
    5mg
    88.00€
    10mg
    115.00€
    25mg
    To inquire
    50mg
    To inquire
    1mL*10mM (DMSO)
    101.00€
  • BQ-788

    CAS:
    BQ-788 is an ETB receptor antagonist with potential hypertensive activity that inhibits exogenous ET-1-induced elevation of coronary perfusion pressure.
    Formula:C34H51N5O7
    Purity:98.81%
    Color and Shape:Solid
    Molecular weight:641.8

    Ref: TM-T10595

    1mg
    137.00€
    2mg
    188.00€
    5mg
    329.00€
    10mg
    472.00€
    25mg
    753.00€
    50mg
    1,017.00€
    100mg
    1,378.00€
    500mg
    2,737.00€
    1mL*10mM (DMSO)
    360.00€
  • Rolapitant hydrochloride

    CAS:
    Rolapitant HCl is a potent NK1 antagonist, non-CYP3A4 interactive, with anti-emetic effects and a Ki of 0.66 nM.
    Formula:C25H27ClF6N2O2
    Purity:98.35% - 99.79%
    Color and Shape:Solid
    Molecular weight:536.94

    Ref: TM-T3724

    1mg
    153.00€
    5mg
    365.00€
    10mg
    520.00€
    25mg
    780.00€
    50mg
    1,054.00€
    100mg
    1,425.00€
    200mg
    1,882.00€
    1mL*10mM (DMSO)
    439.00€
  • Beraprost sodium

    CAS:
    Beraprost sodium is a stable and orally active prodrug of PGI2.
    Formula:C24H29NaO5
    Color and Shape:Solid
    Molecular weight:420.481

    Ref: TM-T13859

    1mg
    Discontinued
    Discontinued product
  • HOKU-81

    CAS:
    HOKU-81is a new bronchodilator and is one of the metabolites of tulobuterol.
    Formula:C12H18ClNO2
    Color and Shape:Solid
    Molecular weight:243.73

    Ref: TM-T15498

    1mg
    Discontinued
    Discontinued product
  • SHA 68

    CAS:
    SHA 68 is a potent and selective non-peptide antagonist of neuropeptide S receptor (NPSR) with IC50 values of 22.0 nM for NPSR Asn107 and 23.8 nM for NPSR Ile107.
    Formula:C26H24FN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:445.49

    Ref: TM-T12895

    1mg
    Discontinued
    Discontinued product
  • JMV 2959

    CAS:
    JMV 2959 is an antagonist of growth hormone secretagogue receptor type 1a (GHS-R1a) (IC50: 32 nM).
    Formula:C30H32N6O2
    Color and Shape:Solid
    Molecular weight:508.61

    Ref: TM-T11719L

    1mg
    Discontinued
    2mg
    Discontinued
    Discontinued product
  • ML-00253764 hydrochloride

    CAS:
    ML-00253764 hydrochloride is an antagonist of nonpeptidic melanocortin receptor 4 (MC4R) (Ki and IC50 of 0.16 µM and 0.103 µM, respectively).
    Formula:C18H19BrClFN2O
    Color and Shape:Solid
    Molecular weight:413.71

    Ref: TM-T12072

    1mg
    Discontinued
    Discontinued product
  • 7-Desmethyl-agomelatine

    CAS:
    7-Desmethyl-agomelatine, a metabolite of Agomelatine, exhibits lower activity than Agomelatine, which functions as a melatonergic (MT1 and MT2) agonist and 5-HT2C antagonist.
    Formula:C14H15NO2
    Color and Shape:Solid
    Molecular weight:229.27

    Ref: TM-T10193

    1mg
    Discontinued
    Discontinued product
  • SR 146131

    CAS:
    SR 146131 is a potent and selective agonist of the nonpeptide receptor.
    Formula:C32H36ClN3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:610.16

    Ref: TM-T16935

    1mg
    Discontinued
    Discontinued product
  • BIBP3226 TFA

    CAS:
    BIBP3226 TFA is an effective and selective antagonist of neuropeptide Y Y1 (NPY Y1) and neuropeptide FF (NPFF) receptor (Kis: 1.1, 79, and 108 nM for rNPY Y1, hNPFF2, and rNPFF).
    Formula:C29H32F3N5O5
    Color and Shape:Solid
    Molecular weight:587.59

    Ref: TM-T10540

    1mg
    Discontinued
    Discontinued product
  • CYM 9484

    CAS:
    CYM 9484 is a selective and potent neuropeptide Y (NPY) Y2 receptor antagonist with an IC50 value of 19 nM.
    Formula:C27H31N3O3S2
    Color and Shape:Solid
    Molecular weight:509.68

    Ref: TM-T10921

    1mg
    Discontinued
    2mg
    Discontinued
    Discontinued product