GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,998 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5959 products of "GPCR/G-Protein"
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CTP-amiodarone
CTP-amiodarone, a cellular-penetrating conjugate of myocardial cell-targeting peptide and Amiodarone, exhibits anti-arrhythmic activity by blocking Na+, K+, and Ca2+ channels as well as β-adrenergic receptors.Formula:C97H131F3I2N20O25S2Color and Shape:SolidMolecular weight:2352.13[Gln8]-C517 (LH-RH), chicken
CAS:[Gln8] LH-RH: Avian hypothalamic peptide; prompts anterior pituitary to release gonadotropins, controlling reproduction.Formula:C54H71N15O14Purity:98%Color and Shape:SolidMolecular weight:1154.23rGHRH(1-29)NH2
RGHRH (1-29)NH2 is a synthetic peptide that stimulates the secretion of growth hormone (GH).Formula:C155H251N49O40SPurity:98%Color and Shape:SolidMolecular weight:3473.02Desglymidodrine
CAS:Desglymidodrine (ST 1059) is an α1-adrenoceptor agonist and vasoconstrictor, used in cardiovascular research and neurocardiogenic syncope studies.Formula:C10H15NO3Purity:99.56%Color and Shape:SolidMolecular weight:197.23Liraglutide acetate
CAS:Liraglutide acetate is the acetate salt form of Liraglutide, which is a glucagon-like peptide-1 (GLP-1) receptor agonist, utilized in the study of type 2 diabetes.Formula:C172H265N43O51·xC2H4O2Color and Shape:SolidMolecular weight:3751.20 (free base)(Des-Bromo)-Neuropeptide B (1-23) (human)
CAS:'(Des-Bromo)-Neuropeptide B (1-23) (human)' is an agonist for orphan G-protein-coupled receptors, exhibiting a K i of 1.2 nM for GPR7 (NPBW1) and 341 nM forFormula:C107H162N30O30Color and Shape:SolidMolecular weight:2348.61[Tyr0] Corticotropin Releasing Factor, ovine
CAS:[Tyr^0] Corticotropin Releasing Factor, ovine, is a hypothalamic hormone sourced from sheep that prompts the secretion of adrenocorticotropic hormone (ACTH) andColor and Shape:Solid[Tyr11]-Somatostatin
CAS:[Tyr11]-Somatostatin, a neuroactive peptide, aids proteomics research and modulates retinal function.Formula:C76H104N18O20S2Color and Shape:SolidMolecular weight:1653.8913,14-dihydro-15-keto Prostaglandin F1α
CAS:13,14-dihydro-15-keto Prostaglandin F1α (13,14-dihydro-15-keto PGF1α) is a metabolite of PGF1α that has been reported in the rat stomach.Formula:C20H36O5Color and Shape:SolidMolecular weight:356.5Galanin (1-29)(rat, mouse)
CAS:Non-selective galanin agonist; Ki: GAL1-0.98, GAL2-1.48, GAL3-1.47 nM. Anticonvulsant, stops full seizures in rats.Formula:C141H211N43O41Purity:98%Color and Shape:White Lyophilized PowderMolecular weight:3164.499Ebiratide
CAS:Ebiratide is an analog of ACTH 4-9.Formula:C48H73N11O10SPurity:98%Color and Shape:SolidMolecular weight:996.23Crustacean Cardioactive Peptide (CCAP)
CAS:Crustacean Cardioactive Peptide (CCAP) is a conserved modified cyclic nonapeptide primary structure of PFCNAFTGC-NH2, a disulfide bridge between Cys3 and Cys9.Formula:C42H58N10O12S2Purity:95.40%Color and Shape:SolidMolecular weight:959.1[D-Arg25]-Neuropeptide Y (human)
[D-Arg25] NPY: human Y1 receptor agonist; linked to AD; shields rat neurons from β-Amyloid.Formula:C189H285N55O57SMolecular weight:4271.68Lipoxin B4 methyl ester
CAS:Lipoxin B4 methyl ester is a lipid-soluble prodrug of LXB4, inhibiting PMN migration/adhesion by LTB4 with IC50 of 0.3 nM.Formula:C21H34O5Color and Shape:SolidMolecular weight:366.498[D-His26]-Neuropeptide Y, human, rat
[D-His26]-Neuropeptide Y, human, rat is a synthetic variant of neuropeptide Y (NPY). This compound acts as a Y1R agonist and may help prevent the development of anxiety, social disorders, and depressive symptoms. It has potential as an early intervention treatment for post-traumatic stress responses.Formula:C180H276N54O55SMolecular weight:4106.01808(+)-5-trans Cloprostenol
CAS:Cloprostenol, a synthetic PGF2α derivative, induces estrus and treats reproductive issues in livestock; its minor impurity, (+)-5-trans, is less effective.Formula:C22H29ClO6Color and Shape:SolidMolecular weight:424.92Pindolol
CAS:Pindolol is an effective, non-selective, and specific beta-receptor blocker that acts as a partial beta-adrenergic receptor agonist and a localized 5-HT1A receptor antagonist (Ki=33nM). Pindolol has intrinsic sympathetic activity (ISA) and is primarily used to treat high blood pressure and certain heart conditions. Exhaustion.Formula:C14H20N2O2Color and Shape:Crystals From Ethanol SolidMolecular weight:248.32Thrombostatin cont-1
CAS:Thrombostatin cont-1, an analogue of the bradykinin metabolite thrombostatin, has been shown to reduce platelet activation in the canine carotid arteryFormula:C87H142N34O29S2Molecular weight:2192.4Mitemcinal fumarate
CAS:Mitemcinal fumarate is a erythromycin derivative that is used to treat gastroesophageal reflux disease.Formula:C84H142N2O28Color and Shape:SolidMolecular weight:1628.02Endothelin 1 (swine, human) (TFA)
CAS:Synthetic human/swine Endothelin 1 (TFA) peptide; a potent vasoconstrictor acting on ET A and ET B receptors.Formula:C111H160F3N25O34S5Molecular weight:2605.93
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