
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(993 products)
- Adenosine Receptor(246 products)
- Adrenergic Receptor(3,004 products)
- Bombesin Receptor(33 products)
- Bradykinin Receptor(59 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(212 products)
- Dopamine Receptor(433 products)
- Endothelin Receptor(79 products)
- GNRH Receptor(77 products)
- GPCR19(32 products)
- GRK(32 products)
- GTPase(22 products)
- Glucagon Receptor(182 products)
- Hedgehog/Smoothened(47 products)
- Histamine Receptor(381 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(310 products)
- PAFR(12 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5745 products of "GPCR/G-Protein"
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Beraprost
CAS:Beraprost is a stable prostacyclin analog.Formula:C24H30O5Color and Shape:SolidMolecular weight:398.49Desglymidodrine
CAS:Desglymidodrine (ST 1059) is an α1-adrenoceptor agonist and vasoconstrictor, used in cardiovascular research and neurocardiogenic syncope studies.Formula:C10H15NO3Purity:99.56%Color and Shape:SolidMolecular weight:197.23Pasireotide ditrifluoroacetate
Pasireotide is a stable cyclohexapeptide somatostatin mimic.Formula:C62H68F6N10O13Purity:98%Color and Shape:SolidMolecular weight:1275.25PSEM 308 hydrochloride
PSAM agonist targeting PSAML141F-GlyR and related ion channels in mice; ideal concentration ≤5 mg/kg; plasmids at Addgene.Color and Shape:SolidCB1R antagonist 2
<p>CB1R antagonist 2 (Compound 11g) functions as an antagonist of the cannabinoid receptor 1 (CB1R), inhibiting the MAPK/NF-κB signaling pathway and exhibiting anti-inflammatory properties. In RAW264.7 cells, it suppresses LPS-induced expression of IL-6, IL-1β, and TNF-α. In murine models, it improves OVA-induced allergic rhinitis.</p>Formula:C24H26N4OColor and Shape:SolidMolecular weight:386.49Parstatin(human)
CAS:Cell-permeable PAR1-derived peptide; inhibits endothelial migration, proliferation (IC50 ~3μM), induces apoptosis, and has cardioprotective effects.Formula:C191H330N64O53S3Purity:98%Color and Shape:SolidMolecular weight:4467.29Luprostiol
CAS:Luprostiol is a prostaglandin analog.Formula:C21H29ClO6SColor and Shape:SolidMolecular weight:444.976β-Prostaglandin I1
CAS:6β-PGI1 is a stable PGI2 analog resistant to hydrolysis in aqueous solutions.Formula:C20H34O5Color and Shape:SolidMolecular weight:354.487SLP7111228
CAS:SLP7111228 is an effective and selective SphK1 inhibitor (Ki = 48 nM).Formula:C22H33N5OColor and Shape:SolidMolecular weight:383.53AR-C126313
CAS:<p>AR-C126313 is a thiouracil derivative.</p>Formula:C28H23N7O3SColor and Shape:SolidMolecular weight:537.59Navafenterol
CAS:AZD-8871, a potential COPD and asthma treatment, may work well with ICS.Formula:C38H42N6O6S2Color and Shape:SolidMolecular weight:742.91BA 1
CAS:<p>Potent BB1, BB2, and BB3 agonist; IC50: 0.26, 1.55, 2.52 nM. Boosts glucose transport in myocytes, promotes cancer cell growth in vitro.</p>Formula:C57H76N14O11Purity:98%Color and Shape:SolidMolecular weight:1133.32AM-0466
CAS:AM-0466 has a wide range of applications in life science related research.Formula:C27H19F3N4O4SColor and Shape:SolidMolecular weight:552.52Piperulin A
CAS:Piperulin A effectively inhibits platelet-activating factor receptor (PAFR) by specifically blocking its binding to isolated rabbit platelet plasma membranes,Formula:C23H28O6Color and Shape:SolidMolecular weight:400.46Neuropeptide S(Rat)
CAS:Potent endogenous neuropeptide S receptor (NSPR) agonist (EC50 = 3.2 nM).Formula:C95H160N34O27Purity:98%Color and Shape:SolidMolecular weight:2210.5211β-Prostaglandin E2
CAS:11β-PGE2 is the C-11 epimer of PGE2.Formula:C20H32O5Color and Shape:SolidMolecular weight:352.47Zovaglutide
CAS:Zovaglutide is a GLP-1 receptor agonist that is utilized in diabetes research.Color and Shape:SolidAntibiotic Sch 60057
CAS:Antibiotic Sch 60057 is a useful organic compound for research related to life sciences. The catalog number is T125403 and the CAS number is 203061-35-2.Formula:C45H84O6Color and Shape:SolidMolecular weight:721.161RFRP-3(human)
CAS:<p>NPFF1 receptor agonist, IC50 0.7 nM, blocks cAMP by forskolin. A GnIH homolog, it inhibits GnRH neuron activity.</p>Formula:C45H72N14O10Purity:98%Color and Shape:SolidMolecular weight:969.15L-703606 oxalate hydrate
L-703606 oxalate hydrate is an effective, selective NK1 receptor antagonist. It is utilized in research related to gastric acid secretion.

