
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(985 products)
- Adenosine Receptor(244 products)
- Adrenergic Receptor(2,991 products)
- Bombesin Receptor(32 products)
- Bradykinin Receptor(59 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(209 products)
- Dopamine Receptor(433 products)
- Endothelin Receptor(79 products)
- GNRH Receptor(77 products)
- GPCR19(32 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(181 products)
- Hedgehog/Smoothened(46 products)
- Histamine Receptor(380 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(309 products)
- PAFR(12 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5696 products of "GPCR/G-Protein"
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Protease-Activated Receptor-1 antagonist 2
CAS:<p>Orally active PAR-1 antagonist with 7 nM IC50; potential for CVD research.</p>Formula:C24H23F2N3O2Color and Shape:SolidMolecular weight:423.46Human growth hormone-releasing factor
CAS:<p>GHRH from the hypothalamus prompts the pituitary to produce/release GH by attaching to the GHRHR.</p>Formula:C215H358N72O66SPurity:98%Color and Shape:SolidMolecular weight:5039.65CB2R probe 1
CAS:<p>CB2R Probe 1, a cannabinoid 2 receptor (CB2R) fluorescent probe, exhibits both safety and environmental friendliness, boasting a dissociation constant (K i) of</p>Formula:C36H42N4O4Color and Shape:SolidMolecular weight:594.7415(S)-15-methyl Prostaglandin E2
CAS:15(S)-15-methyl PGE2: A stable PGE2 analog; strong antiulcer with double PGE2 affinity; excels PGE1 in uterine contraction.Formula:C21H34O5Color and Shape:SolidMolecular weight:366.49Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin
CAS:Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin, a synthetic analog of vasopressin (AVP), acts as a weak agonist at the antidiuretic receptor but is a potentFormula:C45H63N15O11S2Color and Shape:SolidMolecular weight:1054.21HAEGTFTSDVS
CAS:HAEGTFTSDVS is the first N-terminal 1-11 residues of GLP-1 peptide.Formula:C48H71N13O20Purity:98%Color and Shape:SolidMolecular weight:1150.18MrgprX2 antagonist-5
CAS:MrgprX2 antagonist-5 from patent WO2020223255A1 inhibits MrgprX2, useful for inflammatory skin disorder studies.Formula:C19H13ClF2N4O2SColor and Shape:SolidMolecular weight:434.85d[Cha4]-AVP
CAS:Potent human V1B vasopressin receptor agonist; Ki: V1B=1.2 nM; increases ACTH, corticosterone; low vasopressor effect.Formula:C50H71N13O11S2Purity:98%Color and Shape:SolidMolecular weight:1094.31GHRF, bovine
CAS:<p>bGRF(1-44)-NH2 is a bovine GH-releasing factor that stimulates GH release and synergizes with Hydrocortisone.</p>Formula:C220H366N72O66SColor and Shape:SolidMolecular weight:5104.72Cortistatin-29 (rat) (trifluoroacetate salt)
CAS:<p>Cortistatin-29, similar to somatostatin-28, derives from preprocortistatin and binds to SST receptors 1-5 with varying IC50 values.</p>Formula:C161H240N46O41S2Color and Shape:SolidMolecular weight:3540.09Scyliorhinin II
CAS:Scyliorhinin II, a cyclic Tachykinin peptide, is a potent NK3 receptor agonist.Formula:C77H119N21O26S3Purity:98%Color and Shape:SolidMolecular weight:1851.09Phoenixin-14 TFA
Phoenixin-14 TFA (PNX-14 TFA) is an endogenous neuropeptide that can modulate GnRH receptor expression and exerts anxiolytic effects.Formula:C75H110N18O20·xC2HF3O2Purity:99.11%Color and Shape:SolidMolecular weight:1583.78 (free base)CH 275
CAS:Potent sst1 agonist with 30.9 nM IC50; selective over sst2-5; inhibits somatostatin in rat nucleus accumbens.Formula:C74H96N14O15S2Purity:98%Color and Shape:SolidMolecular weight:1485.8(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
CAS:V1A receptor antagonist; blocks vasopressin & oxytocin, lowers Ca²⁺ levels (IC50: 5/30 nM); long-acting antivasopressor; anxiolytic in dorsal hippocampus.Formula:C52H74N14O12S2Purity:98%Color and Shape:White Lyophilized PowderMolecular weight:1151.38Proglumide hemicalcium
CAS:Proglumide hemicalcium is a antagonist of nonpeptide and orally active cholecystokinin (CCK)-A/B receptors, has antiepileptic and antioxidant activities.Formula:C18H28CaN2O4Purity:98%Color and Shape:SolidMolecular weight:376.51Dapiglutide
CAS:<p>Dapiglutide (ZP7570) is a long-acting GLP-1R & GLP-2R dual agonist for SBS research.</p>Color and Shape:SolidRelaxin H3 (human)
CAS:Relaxin H3 (human) is a relaxin peptide that exhibits antifibrotic effects through activation of RXFP1 [1].Color and Shape:SolidTHX-B
CAS:THX-B, a potent non-peptidic p75 NTR antagonist, aids in researching diabetic kidney disease and neurodegenerative and inflammatory disorders.Formula:C16H24N6O4Color and Shape:SolidMolecular weight:364.4O-Desmethyl Mebeverine alcohol
CAS:Mebeverine metabolite O-desmethyl alcohol inhibits α1 receptors, relaxing the gut.Formula:C15H25NO2Purity:98%Color and Shape:SolidMolecular weight:251.36GLP-1(7-36), amide acetate
CAS:<p>GLP-1(7-36), amide acetate is a derivative of GLP-1 peptide , activate the GLP-1 receptor, promote insulin secretion,Type 2 diabetes mellitus and obesity.</p>Formula:C151H230N40O47Purity:99.89%Color and Shape:SolidMolecular weight:3357.68

