GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

Show 18 more subcategories

Found 5745 products of "GPCR/G-Protein"

Purity (%)

100

products per page.

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Onvitrelin ucalontide
CAS:
- 1174415-90-7
Onvitrelin ucalontide is a LHRH analogue with anticancer effect; halts breast, ovarian, and prostate tumors in mice.
Formula:C₁₆₃H₂₄₃N₄₃O₃₂
Molecular weight:3316.94
Ref: TM-T76558
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(Ala13)-Apelin-13
CAS:
- 568565-11-7
(Ala13)-Apelin-13 is a useful organic compound for research related to life sciences. The catalog number is T35374 and the CAS number is 568565-11-7.
Formula:C₆₃H₁₀₇N₂₃O₁₆S
Purity:98%
Color and Shape:Solid
Molecular weight:1474.75
Ref: TM-T35374
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17-phenyl trinor Prostaglandin F2α cyclopropyl methyl amide
CAS:
- 1138395-10-4
Prostaglandin F2α (PGF2α) activates the FP receptor, promoting smooth muscle contraction and luteolysis.
Formula:C₂₇H₃₉NO₄
Color and Shape:Solid
Molecular weight:441.612
Ref: TM-T37941
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Glucagon (19-29), human
CAS:
- 64790-15-4
Glucagon, a 29-amino-acid hormone, is produced by alpha cells in the pancreas' islets of Langerhans.
Formula:C₆₁H₈₉N₁₅O₁₈S
Purity:98%
Color and Shape:Solid
Molecular weight:1352.53
Ref: TM-TP1863
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allo-Yohimbine
CAS:
- 522-94-1
allo-Yohimbine is a biochemical.
Formula:C₂₁H₂₆N₂O₃
Color and Shape:Solid
Molecular weight:354.44
Ref: TM-T29884
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17-phenyl trinor Prostaglandin E2 ethyl amide
CAS:
- 1219032-20-8
17-phenyl trinor PGE2 ethyl amide, an EP1/EP3 agonist (Ki: 14-54 nM), enhances lipid solubility and tissue uptake, is a potent antifertility agent.
Formula:C₂₅H₃₅NO₄
Color and Shape:Solid
Molecular weight:413.55
Ref: TM-T37996
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Bombinakinin M acetate
Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial smooth muscle bradykinin receptors and is
Formula:C₁₀₂H₁₆₃N₃₁O₂₆
Purity:99.80%
Color and Shape:Solid
Molecular weight:2239.58
Ref: TM-TP2075L
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Benzomalvin A
CAS:
- 157047-96-6
Benzomalvin A is a filamentous fungal secondary metabolite.
Formula:C₂₄H₁₉N₃O₂
Color and Shape:Solid
Molecular weight:381.43
Ref: TM-T30407
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4-Chloromethamphetamine hydrochloride
CAS:
- 30572-91-9
4-Chloromethamphetamine hydrochloride is a novel psychoactive substance belonging to the amphetamine class.
Formula:C₁₀H₁₅Cl₂N
Color and Shape:Solid
Molecular weight:220.14
Ref: TM-T203542
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Xaliproden
CAS:
- 135354-02-8
Xaliproden is a biochemical.
Formula:C₂₄H₂₂F₃N
Color and Shape:Solid
Molecular weight:381.43
Ref: TM-T35152
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[Leu31,Pro34]-Neuropeptide Y(human,rat)
CAS:
- 132699-73-1
High affinity neuropeptide Y Y1 receptor agonist (Ki = 0.39 nM). Also shows affinity for Y4 and Y5 receptors.
Formula:C₁₈₉H₂₈₄N₅₄O₅₆S
Purity:98%
Color and Shape:Solid
Molecular weight:4241
Ref: TM-TP1985
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LY83583
CAS:
- 91300-60-6
LY83583 is a soluble guanylate cyclase competitive inhibitor with IC50 of 2 µM.
Formula:C₁₅H₁₀N₂O₂
Purity:99.54% - 99.80%
Color and Shape:Solid
Molecular weight:250.25
Ref: TM-T21576
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Anti-TSHR Antibody (M22)
Anti-TSHR Antibody (M22) is a humanized IgG1 monoclonal antibody targeting the thyroid-stimulating hormone receptor (TSHR). This antibody is capable of inhibiting the interaction between TSH and TSHR.
Color and Shape:Odour Liquid
Ref: TM-T9901A-942
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Fabesetron
CAS:
- 129300-27-2
Fabesetron (FK1052): oral dual antagonist for 5-HT3/5-HT4 receptors. Aids in managing acute and delayed chemo-induced emesis.
Formula:C₁₈H₁₉N₃O
Color and Shape:Solid
Molecular weight:293.37
Ref: TM-T38692
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Dipivefrin
CAS:
- 52365-63-6
Dipivefrin is a prodrug of epinephrine, and is used to treat open-angle glaucoma.
Formula:C₁₉H₂₉NO₅
Color and Shape:Solid
Molecular weight:351.44
Ref: TM-T0103L
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Pellotine
CAS:
- 19622-05-0
Pellotine is an alkaloid isolated from Lophophora. It acts as an inverse agonist of the 5-HT7 receptor (5-HT7 receptor), with an EC50 of 291 nM. Pellotine shows strong affinity for the 5-HT1DR and 5-HT6R, with Ki values of 117 nM and 170 nM, respectively. Additionally, Pellotine reduces intracellular cAMP levels, thereby decreasing neuronal excitability and neurotransmitter release.
Formula:C₁₃H₁₉NO₃
Color and Shape:Solid
Molecular weight:237.295
Ref: TM-TN9164
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5-MeO-pyr-T
CAS:
- 3949-14-2
5-MeO-pyr-T (5-Methoxy pyrrolidinyltryptamine) acts as a 5-HT1AR agonist, exhibiting Ki values of 0.577 μM and 373 μM for 5-HT1AR and 5-HT2AR, respectively. It inhibits the reuptake of 5-HT and triggers its release. Additionally, 5-MeO-pyr-T can induce reduced motor activity.
Formula:C₁₅H₂₀N₂O
Color and Shape:Solid
Molecular weight:244.33
Ref: TM-T203568
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Urotensin I
CAS:
- 83930-33-0
Urotensin I, 41-aa neuropeptide, agonist for human/rat CRF receptors, lowers blood pressure in rats, isolated from white suckers.
Formula:C₂₁₀H₃₄₀N₆₂O₆₇S₂
Purity:98%
Color and Shape:Solid
Molecular weight:4869.46
Ref: TM-TP1199
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DSP-1053
CAS:
- 1176326-76-3
Dsp-1053 is a powerful SERT (Ki=1.02 nM) inhibitor with partial 5-HT1A receptor (Ki=5.05 nM) agonizing activity.
Formula:C₂₆H₃₂BrNO₄
Purity:98%
Color and Shape:Solid
Molecular weight:502.44
Ref: TM-T11107
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Benzoquinamide hydrochloride
CAS:
- 113-69-9
Benzoquinamide hydrochloride (3-carbamoyl-N,N-diethyl-1,3,4,6,7,11b-hexahydro-9,11-dimethoxy-2H-benzo[a]quinolizin-2-yl acetate hydrochloride) is an antiemetic
Formula:C₂₂H₃₃ClN₂O₅
Purity:97.13% - 99.56%
Color and Shape:Solid
Molecular weight:440.96
Ref: TM-T9881