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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5745 products of "GPCR/G-Protein"

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  • Losulazine
    Targetmol
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    Losulazine

    CAS:
    <p>Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.</p>
    Formula:C27H22F4N4O3S
    Purity:98.83%
    Color and Shape:Solid
    Molecular weight:558.55

    Ref: TM-T68095

  • 16-phenoxy tetranor Prostaglandin F2α methyl ester
    Targetmol
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    16-phenoxy tetranor Prostaglandin F2α methyl ester

    CAS:
    <p>Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor.</p>
    Formula:C23H32O6
    Color and Shape:Solid
    Molecular weight:404.503

    Ref: TM-T37937

  • Cloprostenol isopropyl ester
    Targetmol
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    Cloprostenol isopropyl ester

    CAS:
    (+)-Chloprostol is a PGF2α agonist, mimics prostaglandin F2α, induces luteal dissolution in mares without side effects or stress.
    Formula:C25H35ClO6
    Color and Shape:Solid
    Molecular weight:466.99

    Ref: TM-T29246

  • INCB3344 R-isomer
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    INCB3344 R-isomer

    <p>INCB3344 is a potent CCR2 antagonist. INCB3344 R-isomer is the R-isomer of INCB3344.</p>
    Formula:C29H34F3N3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:577.59

    Ref: TM-T11650

  • Apelin-36(human)
    Targetmol
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    Apelin-36(human)

    CAS:
    Endogenous APJ agonist, EC50=20nM, regulates cardiovascular function, fluid balance, and feeding; blocks certain HIV strains.
    Formula:C184H297N69O43S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4195.87

    Ref: TM-TP2093

  • Dipentylone hydrochloride
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    Dipentylone hydrochloride

    CAS:
    Dipentylone hydrochloride (Bk-dmbdp HCl) is a psychoactive synthetic cathinone and sympathomimetic stimulant. Its inhibitory activity towards the dopamine transporter (IC50=0.233µM) is tenfold higher than that towards NET and SERT, inhibiting dopamine uptake and stimulating locomotor activity in mice.
    Formula:C14H20ClNO3
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:285.77

    Ref: TM-T205977

  • (R)-CJ 11974
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    (R)-CJ 11974

    CAS:
    (R)-CJ 11974: non-peptide NK1 receptor antagonist, may relieve pain and prevent chemo-induced vomiting.
    Formula:C31H38N2O
    Purity:97.15%
    Color and Shape:Soild
    Molecular weight:454.65

    Ref: TM-T68068L

  • Preclamol hydrochloride
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    Preclamol hydrochloride

    CAS:
    Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.
    Formula:C14H22ClNO
    Color and Shape:Solid
    Molecular weight:255.78

    Ref: TM-T73684

  • Hemokinin 1, human
    Targetmol
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    Hemokinin 1, human

    CAS:
    Endogenous P-like compound, NK1 receptor agonist; IC50: NK1-1.8 nM, NK3-370 nM, NK2-480 nM; boosts B-cell growth, antiapoptotic, lowers blood pressure in vivo.
    Formula:C54H84N14O14S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1185.4

    Ref: TM-TP1899

  • I-BOP
    Targetmol
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    I-BOP

    CAS:
    I-BOP is an agonist (KD=0.61 nM) at the thromboxane A2 receptor (TP).
    Formula:C23H29IO5
    Color and Shape:Solid
    Molecular weight:512.384

    Ref: TM-T35585

  • 15(S)-15-methyl Prostaglandin E2
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    15(S)-15-methyl Prostaglandin E2

    CAS:
    15(S)-15-methyl PGE2: A stable PGE2 analog; strong antiulcer with double PGE2 affinity; excels PGE1 in uterine contraction.
    Formula:C21H34O5
    Color and Shape:Solid
    Molecular weight:366.49

    Ref: TM-T36154

  • CymitQuimica logo
    Targetmol
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    CAP-100

    <p>CAP-100 is a monoclonal antibody targeting CCR7. It neutralizes the ligand binding site and signaling of CCR7. This compound effectively inhibits migration, extravasation, homing, and survival in chronic lymphocytic leukemia (CLL) samples induced by CCR7. CAP-100 can mediate potent tumor cell killing through host immune mechanisms and exhibits favorable toxicity profiles in related hematopoietic cell subsets. It is involved in research on antitumor activity and diseases like chronic lymphocytic leukemia (CLL).</p>
    Color and Shape:Odour Liquid

    Ref: TM-T9901A-961

  • NF157
    Targetmol
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    NF157

    CAS:
    <p>NF157, a selective P2Y11 antagonist with pKi 7.35, lowers MMP-3/MMP-13, aiding OA treatment; IC50s: P2Y11 463 nM, P2Y1 1811 μM, P2Y2 170 μM.</p>
    Formula:C49H28F2N6Na6O23S6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1437.1

    Ref: TM-T16291

  • 15-keto Latanoprost
    Targetmol
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    15-keto Latanoprost

    CAS:
    Latanoprost, a PG analog for ocular pressure, metabolizes into 15-keto latanoprost, a less potent variant reducing intraocular pressure and pupil size.
    Formula:C26H38O5
    Color and Shape:Solid
    Molecular weight:430.58

    Ref: TM-T37932

  • AB21 HCl
    Targetmol
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    AB21 HCl

    AB21 HCl: σ1 receptor antagonist, Ki 13 nM; less potent at σ2 (102 nM). Reduces mechanical hypersensitivity.
    Formula:C23H29ClN2O
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:384.2

    Ref: TM-T77340L

  • CAY10580
    Targetmol
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    CAY10580

    CAS:
    CAY10580 is a potent and selective prostaglandin EP 4 receptor agonist ( K i =35 nM).
    Formula:C19H35NO4
    Color and Shape:Solid
    Molecular weight:341.49

    Ref: TM-T40738

  • Neuropeptide Y 13-36 (porcine)
    Targetmol
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    Neuropeptide Y 13-36 (porcine)

    CAS:
    Neuropeptide Y 13-36 (porcine) is a selective neuropeptide Y2 receptor agonist.
    Formula:C135H209N41O36
    Color and Shape:Solid
    Molecular weight:2982.408

    Ref: TM-T36447

  • Eletriptan
    Targetmol
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    Eletriptan

    CAS:
    <p>Eletriptan, second-generation triptans used to treat migraines, is used as an abortion drug.</p>
    Formula:C22H26N2O2S
    Color and Shape:Solid
    Molecular weight:382.52

    Ref: TM-T0216L

  • Xanthine amine congener trihydrochloride
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    Xanthine amine congener trihydrochloride

    CAS:
    Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.
    Formula:C21H29ClN6O4
    Purity:98.81%
    Color and Shape:Solid
    Molecular weight:464.95

    Ref: TM-T23535L

  • GLP-1R Antagonist 1
    Targetmol
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    GLP-1R Antagonist 1

    CAS:
    <p>GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).</p>
    Formula:C16H11ClF6N4O2
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:440.73

    Ref: TM-T15387