GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,004 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(155 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(192 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5971 products of "GPCR/G-Protein"
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Apadenoson TFA
Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.
Formula:C25H31F3N6O8Purity:98.08%Color and Shape:SoildMolecular weight:600.55Teprotumumab
CAS:Teprotumumab: human antibody, inhibits IGF-1R, used for thyroid eye diseases.
Purity:SDS-PAGE:95.2%;SEC-HPLC:99.6%Color and Shape:LiquidMolecular weight:145.62 kDa(R)-(+)-Atenolol
CAS:(R)-(+)-Atenolol ((R)-Atenolol) is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.Formula:C14H22N2O3Purity:98.72%Color and Shape:SolidMolecular weight:266.34Peptide 401
CAS:Peptide 401: AMP from bee/wasp venom, triggers histamine release, reduces paw swelling.Formula:C110H192N40O24S4Purity:98%Color and Shape:SolidMolecular weight:2587.22Adrenomedullin (11-50), rat
CAS:Adrenomedullin 11-50 rat is a peptide, stimulates CGRP1 receptor for vasodilation, used in bone growth research.Formula:C194H304N58O59S4Purity:98%Color and Shape:SolidMolecular weight:4521.17Des-Arg9-[Leu8]-Bradykinin acetate
CAS:Des-Arg9-[Leu8]-Bradykinin acetate is a potent antagonist of the bradykinin receptor 1 (B1R), utilized in renal fibrosis research [1].Formula:C43H67N11O12Purity:98%Color and Shape:SolidMolecular weight:930.06AC-263093
CAS:AC-263093 is an NPFFR2 agonist with anxiolytic activity that increases c-Fos protein expression in the paraventricular nucleus of the hypothalamus.
Formula:C8H8Br2N4Purity:99.78%Color and Shape:SoildMolecular weight:319.98Substance P (alligator)
CAS:Substance P from alligator: a neuropeptide with structure Arg-Pro-Arg-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH2.Formula:C63H98N20O13SColor and Shape:SolidMolecular weight:1375.64PF-9184
CAS:PF-9184 inhibits human mPGES-1 selectively, with an IC50 of 16.5 nM, and reduces IL-1β-stimulated PGE2 production in vitro.Formula:C21H14Cl2N2O4SPurity:97.43%Color and Shape:SolidMolecular weight:461.32(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
CAS:(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].Formula:C52H76N14O11S2Purity:98%Color and Shape:SolidMolecular weight:1137.38TT-OAD2
CAS:TT-OAD2 is a non-peptide agonist of glucagon-like peptide-1 (GLP-1) receptor (EC50: 5 nM), with the potential for diabetes treatment.
Formula:C50H49Cl4N3O6Purity:98%Color and Shape:SolidMolecular weight:929.75LTB4-IN-2
LTB4-IN-2 (Compound 6x) is a selective inhibitor of Leukotriene B4 (LTB4), acting by specifically targeting the 5-Lipoxygenase-activating protein (FLAP) with anFormula:C24H17N5S2Purity:98%Color and Shape:SolidMolecular weight:439.56Cortistatin-8
CAS:ghrelin receptor antagonistFormula:C47H68N12O9S2Purity:98%Color and Shape:SolidMolecular weight:1009.25tBPC
CAS:Enhances Y4R response to PP, NPY & PYY with EC50 of 0.03, 0.4, 0.5 nM; selective for Y4R over Y1R, Y2R, Y5R.Formula:C16H24O2Color and Shape:SolidMolecular weight:248.36Pancreatic Polypeptide, human
CAS:Endogenous high affinity agonist for human NPY Y4 receptor (Ki = 0.056 nM). Believed to play an important role in the function of the gastrointestinal tract.Formula:C185H287N53O54S2Purity:98%Color and Shape:SolidMolecular weight:4181.71G-Protein antagonist peptide
CAS:Peptide inhibits G protein-receptor binding; competitively blocks M2 and β-adrenoceptor-induced Gs/Gi/Go activation.Formula:C57H64N12O9SPurity:98%Color and Shape:SolidMolecular weight:1093.27OXA(17-33)
CAS:Potent and selective peptide orexin OX1 receptor agonist (EC50 values are 8.29 and 187 nM for OX1 and OX2 receptors respectively). Truncated form of orexin A.Formula:C79H125N23O22Purity:98%Color and Shape:SolidMolecular weight:1749(±)5(6)-EET
CAS:5(6)-EET is a fully racemic version of the enantiomeric forms biosynthesized from arachidonic acid by cytochrome P450 enzymes.Formula:C20H32O3Color and Shape:SolidMolecular weight:320.473MCL0129
CAS:MCL0129, a selective and non-peptidergic melanocortin 4 (MC4) receptor antagonist, is a potential treatment for cachexia.Formula:C34H47FN4OPurity:98%Color and Shape:SolidMolecular weight:546.76M617
CAS:Galanin GAL1 agonist, Ki: GAL1 0.23 nM, GAL2 5.71 nM; boosts rat appetite, lessens inflammation pain.Formula:C112H161N29O28Purity:98%Color and Shape:SolidMolecular weight:2361.68
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