GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,025 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Cortistatin-8 acetate
Cortistatin-8 acetate: synthetic corticosteroid analog, GHS-R antagonist; doesn't affect acyl GH release or hesperidin response.
Formula:C49H72N12O11S2Purity:99.01%Color and Shape:SoildMolecular weight:1069.3Ref: TM-TP2236L
1mg229.00€5mg560.00€10mg800.00€25mg1,216.00€50mg1,644.00€100mg2,213.00€500mg4,436.00€Neuropeptide W-23 (human) (TFA)
Neuropeptide W-23 (human) (NPW-23) TFA, representing the active form of Neuropeptide W, functions as an endogenous agonist for both NPBW1 (GPR7) and NPBW2 (GPR8Color and Shape:Odour SolidVIP(6-28)(human, rat, porcine, bovine)
CAS:VIP(6-28) blocks VIP-induced cAMP signaling in humans, rats, pigs, and cows.Formula:C126H207N37O34SPurity:98%Color and Shape:SolidMolecular weight:2816.2815(S)-Latanoprost
CAS:15(S)-Latanoprost, a latanoprost analog with inverted hydroxyl at C-15, has an IC50 of 24 nM and reduces IOP by 1 mmHg at 3 μg.Formula:C26H40O5Color and Shape:SolidMolecular weight:432.59INCB3344 R-isomer
INCB3344 is a potent CCR2 antagonist. INCB3344 R-isomer is the R-isomer of INCB3344.Formula:C29H34F3N3O6Purity:98%Color and Shape:SolidMolecular weight:577.595-OMe-UDP trisodium salt
CAS:Potent P2Y6 agonistFormula:C10H16N2O13P2Purity:98%Color and Shape:SolidMolecular weight:434.19Apraglutide
CAS:Apraglutide (FE 203799 is a synthetic 33-amino acid peptide and long-acting glp-2 analogue.Formula:C172H263N43O52Purity:98%Color and Shape:SolidMolecular weight:3765.25VU0453379 hydrochloride
VU0453379 hydrochloride: selective CNS-penetrant GLP-1R PAM, EC50 1.3 μM.Formula:C26H35ClN4O2Color and Shape:SolidMolecular weight:471.03Dapoxetine
CAS:Dapoxetine (Dapoxetina) is a selective serotonin reuptake inhibitor, for the treatment of premature ejaculation.Formula:C21H23NOPurity:99.73%Color and Shape:White To Off-White Crystalline PowderMolecular weight:305.42ent-8-iso Prostaglandin F2α
CAS:ent-8-iso Prostaglandin F2α is a potent vasoconstrictor of porcine retinal and cerebral microvessels with EC50 values of 30.6 and 53.5 nM, respectively.Formula:C20H34O5Color and Shape:SolidMolecular weight:354.487Antidepressant agent 4
Antidepressant agent 4: orally active, has antidepressant, anxiolytic, and nootropic effects.Formula:C19H38ClN5O2SColor and Shape:SolidMolecular weight:436.06FSLLRY-NH2
CAS:PAR2 antagonist; counters taxol effects, PKC in mice; inhibits ERK, collagen in fibroblasts; lessens dermatophyte itch in mice.Formula:C39H60N10O8Purity:98%Color and Shape:SolidMolecular weight:796.97(±)5(6)-EET
CAS:5(6)-EET is a fully racemic version of the enantiomeric forms biosynthesized from arachidonic acid by cytochrome P450 enzymes.Formula:C20H32O3Color and Shape:SolidMolecular weight:320.47315-keto-17-phenyl trinor Prostaglandin F2α ethyl amide
CAS:Bimatoprost is the Allergan trade name for 17-phenyl trinor prostaglandin F2α ethyl amide (17-phenyl trinor PGF2α ethyl amide), an F-series PG analog which hasFormula:C25H35NO4Color and Shape:SolidMolecular weight:413.558Pancreatic Polypeptide, human
CAS:Endogenous high affinity agonist for human NPY Y4 receptor (Ki = 0.056 nM). Believed to play an important role in the function of the gastrointestinal tract.Formula:C185H287N53O54S2Purity:98%Color and Shape:SolidMolecular weight:4181.71O-Desmethyl-N-deschlorobenzoyl Indomethacin
CAS:O-Desmethyl-N-deschlorobenzoyl indomethacin, a metabolite of indomethacin, reduces HL-60 cell viability and aids in synthesizing PGD2 receptor antagonists.Formula:C11H11NO3Color and Shape:SolidMolecular weight:205.213Pemvidutide TFA
Pemvidutide (TFA), a GLP-1R/GCGR dual agonist, effectively reduces body weight, liver fat, and serum lipid levels, and is utilized in research on non-alcoholicFormula:C182H275N39O54·xC2HF3O2Color and Shape:SolidMolecular weight:3873.35 (free base)Thielocin B1
CAS:Thielocin B1, a PAC3 inhibitor and novel PLA2 blocker, is derived from Thielavia terricola RF-143's culture.Formula:C53H58O17Color and Shape:SolidMolecular weight:967.02Hemopressin(rat)
CAS:Peptide inhibitor for ep24.15, neurolysin & ACE with Ki 27.76, 3.43, 1.87 μM. Lowers blood pressure, modulates CB1 receptor, reduces pain & food intake.Formula:C53H77N13O12Purity:98%Color and Shape:SolidMolecular weight:1088.27Cannabigerorcin
CAS:Cannabigerorcin, a phytocannabinoid, serves as an analytical reference standard. It is designated for research and forensic applications.Formula:C17H24O2Color and Shape:SolidMolecular weight:260.377
