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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5838 products of "GPCR/G-Protein"

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  • Tilisolol HCl

    CAS:
    Tilisolol, a nonselective beta-blocker, dilates dog coronary arteries via ATP-sensitive K(+) channels.
    Formula:C17H25ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:340.85
  • LY 344864 S-enantiomer

    CAS:
    LY 344864 S-enantiomer, the S-enantiomer of LY344864, serves as a 5-HT1F receptor agonist.
    Formula:C21H22FN3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:351.42
  • Bopindolol fumarate

    CAS:
    <p>Bopindolol fumarate: non-selective β1/β2-adrenoceptor blocker, partial agonist, low β3 affinity, treats hypertension.</p>
    Formula:C27H32N2O7
    Color and Shape:Solid
    Molecular weight:496.56
  • VNA-932

    CAS:
    <p>VNA-932 is an agonist of the vasopressin V2-receptor (IC50: 80.3 nM and 778 nM in human-V2 binding and V1a binding assay).</p>
    Formula:C23H19ClN4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:402.88
  • I-SAP

    CAS:
    <p>I-SAP: TP receptor blocker, alters platelet shape without causing clumping, EC50 9.7 nM, max binding pH 6.5-7.4, Kd 468-490 pM.</p>
    Formula:C22H30INO4S
    Color and Shape:Solid
    Molecular weight:531.45
  • PD-89211

    CAS:
    PD 89211 selectively blocks dopamine D4.2 receptor >800x vs. other subtypes; reverses quinpirole effect in vitro (IC50 = 2.1 nM).
    Formula:C19H21ClN4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.85
  • MK-0249

    CAS:
    <p>MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).</p>
    Formula:C23H24F3N3O2
    Purity:99.90%
    Color and Shape:Solid
    Molecular weight:431.45
  • 5-HT6/5-HT2A receptor ligand-1

    CAS:
    <p>Compound 33 is a dual 5-HT6/5-HT2A antagonist with Ki values of 2 nM and 11 nM, respectively, useful in neuro/psychiatric research.</p>
    Formula:C21H19FN2O2
    Color and Shape:Solid
    Molecular weight:350.39
  • H3 receptor-MO-1

    CAS:
    H3 receptor-MO-1 is a potent modulator of the histamine H3 receptor (H3 receptor) and can be used to study neurodegeneration and cognitive disorders.
    Formula:C20H27N3O2
    Purity:99.11%
    Color and Shape:Solid
    Molecular weight:341.45
  • Rocastine

    CAS:
    <p>Rocastine (AHR-11325) is a selective and potent non-sedating H1 receptor antagonist.</p>
    Formula:C13H19N3OS
    Purity:98.26%
    Color and Shape:Solid
    Molecular weight:265.37
  • QF0301B

    CAS:
    QF0301B is a potent α1-adrenergic receptor antagonist with inhibitory effects on α2-adrenergic receptors, 5-HT2A and histamine H1 receptors.
    Formula:C23H28N2O2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:364.48
  • Tulopafant

    CAS:
    Tulopafant (RP 59227) is a potent platelet-activating factor (PAF) antagonist that increases capillary patency and prolongs allograft heart survival.
    Formula:C25H19N3O2S
    Purity:99.38%
    Color and Shape:Solid
    Molecular weight:425.5
  • CL-216303 HCl

    CAS:
    CL-216303 HCl, a dopamine transporter inhibitor and a 5-HT inhibitor, is used potentially for the treatment of depression.
    Formula:C11H12Cl3N
    Purity:98%
    Color and Shape:Solid
    Molecular weight:264.58
  • Oxiperomide

    CAS:
    Oxiperomide is a dopamine D2 and muscarinic M1 receptor ligand. It also has putative antipsychotic and pro-cognitive potential.
    Formula:C20H23N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:337.42
  • T-0509

    CAS:
    <p>T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle and selectively down-regulates rat cardiac beta 1-</p>
    Formula:C18H23NO5
    Purity:97.52% - 98.43%
    Color and Shape:Solid
    Molecular weight:333.38
  • Glucagon receptor antagonists-2

    CAS:
    Glucagon receptor antagonist -2 is a highly effective glucagon receptor antagonist.
    Formula:C22H30FNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:359.48
  • JNJ-10191584

    CAS:
    JNJ-10191584, a potent and selective antagonist at the histamine H4 receptor, has antiinflammatory and analgesic effects in animal studies of acute inflammation
    Formula:C13H15ClN4O
    Color and Shape:Solid
    Molecular weight:278.74
  • Alimemazine

    CAS:
    Alimemazine, an antipruritic and HA-receptor antagonist, also partially activates H1R and other GPCRs.
    Formula:C18H22N2S
    Purity:98%
    Color and Shape:Crystals Solid
    Molecular weight:298.45
  • NGB 2904 hydrochloride

    CAS:
    dopamine D3 receptor antagonist
    Formula:C28H30Cl3N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:530.92
  • Isoproterenol-d7 HCl

    CAS:
    Isoproterenol-d7: internal standard for GC/LC-MS. β1-/β2-AR agonist, not for β3. Lowers blood pressure, tackles bradydysrhythmias, asthma.
    Formula:C11H18ClNO3
    Molecular weight:254.76
  • Aminopotentidine

    CAS:
    H2 antagonist
    Formula:C26H35N7O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:477.6
  • TC-C 14G

    CAS:
    CB1 receptor inverse agonist
    Formula:C24H17Cl2F2NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:492.3
  • RS 64459-193

    CAS:
    RS 64459-193 has a high affinity for the 5-HT1A binding site.
    Formula:C26H36Cl2N2O2
    Color and Shape:Solid
    Molecular weight:479.48
  • CCK-A receptor inhibitor 1

    CAS:
    <p>CCK-A receptor inhibitor 1 is a potent inhibitor of the cholecystokinin A (CCK-A) receptor (IC50: 340 nM).CCK-A receptor inhibitor 1 can be used for the study</p>
    Formula:C25H35NO6S
    Purity:99.47%
    Color and Shape:Solid
    Molecular weight:477.61
  • Pamatolol

    CAS:
    Pamatolol is a selective and potent beta-adrenoceptor antagonist that has not shown sympathomimetic activity in ex vivo experiments.
    Formula:C16H26N2O4
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:310.39
  • Cicloprolol hydrochloride

    CAS:
    Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.
    Formula:C18H30ClNO4
    Purity:97.26%
    Color and Shape:Solid
    Molecular weight:359.89
  • Bamirastine

    CAS:
    Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect on
    Formula:C31H37N5O3
    Purity:96.68%
    Color and Shape:Solid
    Molecular weight:527.66
  • LEI-101

    CAS:
    LEI-101: potent CB2 agonist, pEC50=8, bioavailable, >100x selective over CB1, potential for inflammatory diseases.
    Formula:C23H25FN4O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:472.53
  • (4E)-SUN9221

    CAS:
    (4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity in
    Formula:C25H31FN4O3
    Purity:97.79%
    Color and Shape:Solid
    Molecular weight:454.54
  • L-771688

    CAS:
    L-771688 (SNAP 6383) is a novel potent and selective α1A-adrenoceptor antagonist with a Ki value of 0.43±0.02 nM.L-771688 KE is used for the treatment of benign
    Formula:C28H33F2N5O5
    Purity:94.15%
    Color and Shape:Solid
    Molecular weight:557.59
  • GSK-894490A

    CAS:
    GSK-894490A is an agonist of ghrelin receptor. GSK-894490A crosses the blood/brain barrier and elicit pro-cognitive effects.
    Formula:C24H30ClN3O4S
    Color and Shape:Solid
    Molecular weight:492.03
  • Zolantidine dimaleate

    CAS:
    H2 receptor antagonist
    Formula:C26H31N3O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:497.61
  • ONO4057

    CAS:
    ONO4057 is a potent and orally active Leukotriene B4 receptor antagonist with an IC50 value of 0.7±0.3 μM.
    Formula:C27H34O7
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:470.55
  • PAF-AN-1

    CAS:
    <p>PAF-AN-1 is a novel potent platelet-activating factor receptor (PAF) antagonist involved in the study of anaphylactic death.</p>
    Formula:C28H28N2O3
    Purity:98.06%
    Color and Shape:Solid
    Molecular weight:440.53
  • L-803087

    CAS:
    L-803087: potent sst4 receptor agonist, 0.7 nM Ki, 280x selectivity, boosts AMPA responses & seizures in mice.
    Formula:C25H29F2N5O3
    Purity:99.37%
    Color and Shape:Solid
    Molecular weight:485.53
  • CP-66948

    CAS:
    CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion and can be used to protect gastric and intestinal mucosa.
    Formula:C13H20N6S
    Purity:99.14%
    Color and Shape:Solid
    Molecular weight:292.4
  • Indanidine

    CAS:
    Indanidine is a highly selective and potent α-adrenergic agonist with antihypertensive activity.Indanidine is an α-adrenergic antagonist that can be used in the
    Formula:C11H13N5
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:215.25
  • RS-601

    CAS:
    RS-601 is a potent dual leukotriene D4/thromboxane A2 inhibitor that inhibits antigen-induced airway hyperresponsiveness (AHR) and shows asthmatic effects in a
    Formula:C22H23F6NO4S
    Purity:99.31%
    Color and Shape:Solid
    Molecular weight:511.48
  • TD-5471 hydrochloride

    CAS:
    TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment of chronic obstructive pulmonary disease (
    Formula:C32H32ClN3O4
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:558.07
  • Masupirdine mesylate

    CAS:
    Masupirdine mesylate (SUVN-502 mesylate) is a 5-HT6 receptor antagonist.Masupirdine mesylate is used to study neurological disorders such as Alzheimer's disease
    Formula:C23H32BrN3O9S3
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:670.61
  • Odapipam

    CAS:
    Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).
    Formula:C19H20ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.82
  • SLM6031434 HCl

    CAS:
    SLM6031434 HCl (SLM-6031434 HCl) is a SphK2 inhibitor that reduces LPS-induced TNF伪 and IL-1尾 production.
    Formula:C22H31ClF3N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:489.96
  • p-MPPF dihydrochloride

    CAS:
    p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.
    Formula:C25H29Cl2FN4O2
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:507.43
  • ABT-239

    CAS:
    ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists.
    Formula:C22H22N2O
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:330.42
  • PF-03654764

    CAS:
    <p>PF-03654764, an oral H3 receptor blocker, Ki: human 1.2 nM, rat 7.9 nM, used with Fexofenadine for allergic rhinitis.</p>
    Formula:C20H28F2N2O
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:350.45
  • Napitane

    CAS:
    <p>napitane (A 75200) is a novel catecholamine uptake inhibitor with inhibitory effects on α-adrenergic receptors and potential antidepressant activity for the</p>
    Formula:C22H25NO2
    Purity:99.77% - 99.89%
    Color and Shape:Solid
    Molecular weight:335.44
  • Methdilazine Hydrochloride

    CAS:
    Methdilazine Hydrochloride (Bristaline) is a histamine H1 receptor antagonist for dermatologic conditions and relief of itching by allergies or rhinitis.
    Formula:C18H21ClN2S
    Color and Shape:Light-Tan Crystalline Powder 4 8-6 (Ntp 1992)
    Molecular weight:332.89
  • GB83

    CAS:
    GB83 is a selective human protease activated receptor 2 (PAR2) antagonist.
    Formula:C32H44N4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:548.72
  • WS 009A

    CAS:
    WS 009A is an antagonist of the endothelin receptor.
    Formula:C24H25NO10S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:519.52
  • Norfenefrine HCl

    CAS:
    <p>Norfenefrine HCl is an α1-adrenergic receptor agonist, an endogenous neurotransmitter and sympathomimetic drug for hypotension,glycerol adipose.</p>
    Formula:C8H12ClNO2
    Purity:99.44%
    Color and Shape:Solid
    Molecular weight:189.64
  • Arvanil

    CAS:
    Arvanil (N-Vanillylarachidonamide) is a synthetic capsaicin-amphetamine hybrid that acts as a ligand for VR1 and CB1, offering neuroprotective effects.
    Formula:C28H41NO3
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:439.63
  • PGN-9856

    CAS:
    PGN-9856 is an EP2 receptor ligand and EP2 receptor agonist with anti-inflammatory and intraocular pressure-lowering properties, useful for glaucoma research.
    Formula:C21H15F2NO4
    Purity:99.27%
    Color and Shape:Solid
    Molecular weight:383.35
  • CCK-B Receptor Antagonist 1

    CAS:
    CCK-B Receptor Antagonist 1 is a cholecystokinin B (CCK-B) receptor agonist and has the potential of reducing the secretion of gastric acid.
    Formula:C28H30N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:498.58
  • Propiomazine HCl

    CAS:
    Propiomazine HCl is an analgesia adjunct.
    Formula:C20H25ClN2OS
    Color and Shape:Solid
    Molecular weight:376.94
  • RP73870

    CAS:
    RP73870 is a gastrin/cholecystokinin-B receptor antagonist and H2 receptor antagonist with potent anti-ulcer activity.
    Formula:C27H30N4O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:554.61
  • Trimopam

    CAS:
    Trimopam is a dopamine receptor agonist of the benzazepine group.
    Formula:C19H23NO2
    Color and Shape:Solid
    Molecular weight:297.39
  • Daledalin tosylate

    CAS:
    Daledalin tosylate is an antidepressant.
    Formula:C26H32N2O3S
    Color and Shape:Solid
    Molecular weight:452.61
  • PD 118717

    CAS:
    PD 118717: a piperazinyl benzopyranone dopamine agonist with potential antipsychotic properties and no neurological side effects in tests.
    Formula:C20H22N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:366.41
  • Bucumarol (HCl)

    CAS:
    Bucumarol is a beta-adrenergic blocking agent.
    Formula:C17H24ClNO4
    Color and Shape:Solid
    Molecular weight:341.83
  • MHP 133

    CAS:
    <p>MHP 133 is a drug with multiple CNS targets(AChE with Ki of 69 μM).</p>
    Formula:C17H20ClN5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:377.83
  • SKF-80723 HBr

    CAS:
    SKF-80723 HBr is a potent D1 agonist enhancing quinpirole-induced circling in 6-OHDA lesioned rats.
    Formula:C16H16BrNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:334.21
  • Trebenzomine

    CAS:
    Trebenzomine is apsychotropic agent with potential as an antidepressant and an antipsychotic.
    Formula:C12H17NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:191.27
  • VK-II-86

    CAS:
    VK-II-86 is a non-β-blocking carvedilol analog. It prevents ouabain-Induced cardiotoxicity
    Formula:C25H28N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:420.5
  • LPA2 antagonist 1

    CAS:
    LPA2 antagonist 1 is a potent LPA2 antagonist.
    Formula:C20H23Cl2N5O2S2
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:500.47
  • (R)-Viloxazine Hydrochloride

    CAS:
    (R)-Viloxazine Hydrochloride, the R-isomer of Viloxazine.
    Formula:C13H20ClNO3
    Purity:99.88% - 99.94%
    Color and Shape:Solid
    Molecular weight:273.76
  • Ro 363

    CAS:
    RO 363: Potent β1-adrenoceptor agonist, boosts heart contractility, lowers diastolic pressure.
    Formula:C19H25NO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:363.4
  • A1AR antagonist 3

    CAS:
    Compound 13: selective A1AR antagonist, Ki human A1: 9.69 nM, rat A1: 0.529 nM, useful for neurological research.
    Formula:C25H20N2O3S
    Color and Shape:Solid
    Molecular weight:428.5
  • Argiprestocin

    CAS:
    Argiprestocin: antidiuretic, regulates osmolality, neurohypophysial hormone, vasoconstrictor.
    Formula:C43H67N15O12S2
    Purity:99.34%
    Color and Shape:Solid
    Molecular weight:1050.22
  • RWJ 52353

    CAS:
    α2D adrenergic receptor agonist
    Formula:C11H10N2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:202.28
  • AF40431

    CAS:
    AF40431 is the first reported small-molecule ligand of sortilin (IC50: 4.4 μM; Kd: 0.7 μM). AF40431 is bound in the neurotensin-binding site of sortilin.
    Formula:C17H21NO5
    Color and Shape:Solid
    Molecular weight:319.35
  • VL-0395

    CAS:
    VL-0395 is an antagonist of CCK1 receptor.
    Formula:C25H21N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:427.45
  • Iloperidone hydrochloride

    CAS:
    Iloperidone hydrochloride is a D(2)/5-HT(2) receptor antagonist. It is also an atypical antipsychotic for the treatment of schizophrenia symptoms.
    Formula:C24H28ClFN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:462.95
  • A1AR antagonist 5

    CAS:
    <p>A1AR antagonist 5 (compound 20) is a potent and selective antagonist of A1 adenosine receptor (A1AR) with a pKi of 6.11 and a pIC 50 of 5.83 [1].</p>
    Formula:C17H15ClN4O
    Color and Shape:Solid
    Molecular weight:326.78
  • SB-269970

    CAS:
    SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).
    Formula:C18H28N2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.49
  • Mabuterol, (S)-

    CAS:
    Mabuterol, a β2 adrenoreceptor agonist, lowers rat blood pressure and boosts guinea pig heart rate/force, not affecting other receptors.
    Formula:C13H18ClF3N2O
    Color and Shape:Solid
    Molecular weight:310.74
  • MRS1097

    CAS:
    MRS1097 is a selective antagonist A3 adenosine receptor.
    Formula:C26H27NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:417.5
  • CBK289001

    CAS:
    <p>CBK289001 inhibits TRAP 5b MV, 5b OX &amp; 5a OX with IC50s: 125μM, 4.21μM, 14.2μM.</p>
    Formula:C19H20N6O4
    Color and Shape:Solid
    Molecular weight:396.4
  • SB 258719 hydrochloride

    CAS:
    Selective 5-HT7 receptor antagonist
    Formula:C18H31ClN2O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:374.97
  • Colterol HCl

    CAS:
    Colterol HCl, a β2-adrenoceptor agonist salt, is used for bronchospasm in asthma and COPD.
    Formula:C12H20ClNO3
    Color and Shape:Solid
    Molecular weight:261.75
  • Dacemazine

    CAS:
    Dacemazine is used to treat depression.
    Formula:C16H16N2OS
    Color and Shape:Solid
    Molecular weight:284.38
  • Fulimetibant

    CAS:
    Fulimetibant is a bradykinin receptor antagonist.
    Formula:C25H21F4N3O3
    Color and Shape:Solid
    Molecular weight:487.45
  • TBC3711

    CAS:
    TBC3711 is an endothelin receptor modulator. It is used for the research of endothelin-mediated disorders.
    Formula:C20H21N3O5S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:447.53
  • Ambenoxan hydrochloride

    CAS:
    Ambenoxan hydrochloride is a centrally acting skeletal muscle relaxant.
    Formula:C14H22ClNO4
    Color and Shape:Solid
    Molecular weight:303.78
  • Ambucetamide

    CAS:
    Ambucetamide is an antispasmodic, it may inhibit or diminish the spontaneous rhythmical activity of the human myometrium.
    Formula:C17H28N2O2
    Color and Shape:Solid
    Molecular weight:292.42
  • BAY-386

    CAS:
    BAY-386 is a PAR1 receptor inhibitor which suppresses activation of thrombin and platelet activity.
    Formula:C22H25F3N4O5S
    Color and Shape:Solid
    Molecular weight:514.52
  • Ranitidine bismuth citrate

    CAS:
    Ranitidine bismuth citrate, oral H2 blocker, IC50 3.3 µM, targets SARS-CoV-2 cells, treats H. pylori; MIC90 16 ng/L.
    Formula:C19H27BiN4O10S
    Color and Shape:Solid
    Molecular weight:712.48
  • F-15599 tosylate

    CAS:
    F-15599 tosylate is a selective 5-HT(1A) agonist.
    Formula:C26H29ClF2N4O4S
    Color and Shape:Solid
    Molecular weight:567.05
  • VUF14738

    CAS:
    VUF14738 is a robust and fatigue-resistant photoswitchable GPCR antagonist.
    Formula:C25H32N4O2
    Color and Shape:Solid
    Molecular weight:420.55
  • OPC-14523 free base

    CAS:
    OPC-14523, a 5-HT1A receptor agonist, is used potentially for the treatment of depression and neuropathic pain.
    Formula:C23H28ClN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:413.94
  • LY320135

    CAS:
    CB1 receptor antagonist/inverse agonist
    Formula:C24H17NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:383.4
  • Cyclazosin HCl

    CAS:
    Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.
    Formula:C23H28ClN5O4
    Purity:99.10%
    Color and Shape:Solid
    Molecular weight:473.95
  • Albuterol adipate

    CAS:
    Albuterol adipate, a β2-AR agonist salt, treats asthma/COPD, with high selectivity for pulmonary over cardiac receptors.
    Formula:C32H52N2O10
    Color and Shape:Solid
    Molecular weight:624.77
  • Levomepromazine Maleate

    CAS:
    Levomepromazine Maleate: TCA and SNRI with antihistamine, antiadrenergic, and anticholinergic properties.
    Formula:C23H28N2O5S
    Color and Shape:Solid
    Molecular weight:444.546
  • ZD7114 free base

    CAS:
    ZD7114 (ICI-D7114) selectively activates brown fat, boosts thermogenesis, and aids in obesity and metabolic disorders.
    Formula:C22H30N2O6
    Color and Shape:Solid
    Molecular weight:418.48
  • L-694,247

    CAS:
    L-694,247 is a 5-HT receptor agonist with affinity for 5-HT1D, 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1E receptors, and can be used to study neurological diseases.
    Formula:C20H21N5O3S
    Purity:98.36%
    Color and Shape:White Solid
    Molecular weight:411.48
  • Aceprometazine

    CAS:
    Aceprometazine (1664CB) is an antipsychotic which is orally active. Aceprometazine can be used in psychiatric disorders research, for example, depression [1].
    Formula:C19H22N2OS
    Color and Shape:Solid
    Molecular weight:326.46
  • Ricinelaidic Acid

    CAS:
    Ricinelaidic acid blocks LTB4 receptors; hampers human neutrophil responses; reduces rat bronchoconstriction by 46% at 1 mg/kg i.v.
    Formula:C18H34O3
    Color and Shape:Solid
    Molecular weight:298.46
  • Darbufelone

    CAS:
    <p>Darbufelone (CI-1004) is a non-competitive dual inhibitor of PGF2α and LTB4.</p>
    Formula:C18H24N2O2S
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:332.46
  • GBR-12935 maleate

    CAS:
    GBR-12935: dopamine reuptake inhibitor, used in research for Parkinson's and brain's dopamine pathways.
    Formula:C32H38N2O5
    Color and Shape:Solid
    Molecular weight:530.665
  • 6-Chloromelatonin

    CAS:
    6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.
    Formula:C13H15ClN2O2
    Purity:97.26% - 99.25%
    Color and Shape:Solid
    Molecular weight:266.72
  • (R)-Mequitazine

    CAS:
    <p>(R)-Mequitazine, a muscarinic acetylcholine receptor (M-AChRs) antagonist, is used potentially for the treatment of asthma.</p>
    Formula:C20H22N2S
    Color and Shape:Solid
    Molecular weight:322.47
  • VRX 03011 Potassium salt

    CAS:
    VRX 03011, a 5-HT4 partial agonist, is used potentially for the treatment of Alzheimer's disease.
    Formula:C19H27KN3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:416.6
  • Quinpirole

    CAS:
    Quinpirole is a dopamine D2/D3 receptor agonist.
    Formula:C13H21N3
    Color and Shape:Solid
    Molecular weight:219.33
  • KUL-7211 racemate

    CAS:
    KUL 7211, a selective β-adrenoceptor agonist, exists as a racemate, referred to as KUL 7211 racemate, which is the mixture of its enantiomers.
    Formula:C19H23NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:345.39
  • Thiothixene hydrochloride

    CAS:
    Thiothixene hydrochloride is an antipsychotic agent that can be used in the study of schizophrenia and bipolar mania.
    Formula:C23H30ClN3O2S2
    Color and Shape:Solid
    Molecular weight:480.08
  • Isoetharine hydrochloride

    CAS:
    Isoetharine HCl, a selective, short-acting oral β-agonist, is used as a bronchodilator for inhalation therapy.
    Formula:C13H22ClNO3
    Color and Shape:Solid
    Molecular weight:275.77
  • A-304121

    CAS:
    A-304121 is a histamine H(3) receptor.
    Formula:C20H29N3O3
    Color and Shape:Solid
    Molecular weight:359.46
  • Trimethaphan camsylate

    CAS:
    Trimethaphan camsylate is a nicotinic antagonist that has been used as a ganglionic blocker in hypertension.
    Formula:C32H40N2O5S2
    Color and Shape:Solid
    Molecular weight:596.801
  • Ro 23-3423

    CAS:
    Ro 23-3423 is a specific inhibitor of thromboxane synthetase.
    Formula:C23H22N4O2
    Color and Shape:Solid
    Molecular weight:386.45
  • Glucagon receptor antagonists-5

    CAS:
    Oral indazole-based glucagon antagonist, Ki: 32 nM, may treat type 2 diabetes.
    Formula:C30H29ClF3N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:572.02
  • Proxodolol hydrochloride

    CAS:
    Proxodolol, a β-adrenergic receptor antagonist, is used potentially for the treatment of glaucoma, hypertension and angina.
    Formula:C17H26ClN3O4
    Color and Shape:Solid
    Molecular weight:371.86
  • Opaganib HCl

    CAS:
    ABC294640 (Opaganib) is an SK2 inhibitor with potential anti-cancer effects; it blocks S1P production to induce apoptosis.
    Formula:C23H26Cl2N2O
    Color and Shape:Solid
    Molecular weight:417.37
  • GSK466317A

    CAS:
    GSK466317A is a GRK2 inhibitor.
    Formula:C21H16ClF3N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:448.83
  • Dicentrine HCl

    CAS:
    Dicentrine HCl is the salt form of Dicentrine, an alpha 1-adrenoceptor antagonist effective against human hyperplastic prostates.
    Formula:C20H22ClNO4
    Color and Shape:Solid
    Molecular weight:375.85
  • Org-12962 hydrochloride

    CAS:
    Org-12962 hydrochloride is a 5-HT2C receptor agonist.
    Formula:C10H12Cl2F3N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:302.12
  • DH-97

    CAS:
    DH-97 is a potent MT2 melatonin receptor antagonist (pKi value = 8.03).
    Formula:C22H26N2O
    Color and Shape:Solid
    Molecular weight:334.45
  • Esreboxetine

    CAS:
    Esreboxetine( PNU-165442, (S,S) -reboxetine) is a selective inhibitor of norepinephrine reuptake.
    Formula:C19H23NO3
    Color and Shape:Solid
    Molecular weight:313.39
  • CGP 25454A

    CAS:
    CGP 25454A is a novel and selective antagonist of the presynaptic dopamine autoreceptor.
    Formula:C15H21Cl2N3O2
    Color and Shape:Solid
    Molecular weight:346.25
  • Bitolterol

    CAS:
    Bitolterol is a new beta 2-adrenergic agonist and classified as a pro-drug.
    Formula:C28H31NO5
    Color and Shape:Solid
    Molecular weight:461.55
  • R-SKF-38393A HCl

    CAS:
    R(+)-SKF-38393A is a D1 dopamine receptor agonist and also is a more active enantiomer of (±)-SKF-38393A.
    Formula:C16H18ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:291.77
  • A1AR antagonist 4

    CAS:
    Compound 22: A1AR antagonist, pIC50 5.51, pKi 6.29, potent and selective.
    Formula:C23H25N3O2
    Color and Shape:Solid
    Molecular weight:375.46
  • 5-Methylurapidil

    CAS:
    <p>5-Methylurapidil is an alpha1A-adrenoceptor antagonist.</p>
    Formula:C21H31N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:401.5
  • 5-HT4 antagonist 1

    CAS:
    5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).
    Formula:C23H36N4O5S
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:480.62
  • Glucagon Receptor Antagonist I

    CAS:
    Glucagon antagonist I blocks the GCGR (IC50=181 nM), stops glucagon-induced glycogenolysis, and lowers glucose in glucagon-treated humanized mice.
    Formula:C20H30N2OS
    Color and Shape:Solid
    Molecular weight:346.53
  • Sch 44643

    CAS:
    Sch 44643 is an antagonist of platelet activating factor with oral activity.
    Formula:C25H22ClN3O2
    Color and Shape:Solid
    Molecular weight:431.91
  • A2AR-agonist-1

    CAS:
    <p>A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).</p>
    Formula:C20H22N6O4
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:410.43
  • DR4485 hydrochloride

    CAS:
    5-HT7 antagonist
    Formula:C26H29Cl3N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:491.88
  • Iferanserin HCl

    CAS:
    Iferanserin HCl is a selective serotonin receptor antagonist.
    Formula:C23H29ClN2O
    Color and Shape:Solid
    Molecular weight:384.95
  • GYKI-13380

    CAS:
    GYKI-13380, also known as LS-79445, is a small molecule with potent bioactivity. Detail information has not been published yet.
    Formula:C16H22N2O3
    Color and Shape:Solid
    Molecular weight:290.36
  • Ksg 504

    CAS:
    Ksg 504 has superior selectivity and affinity to CCK-A receptors and derived from proglumide.
    Formula:C31H49N5O8S
    Color and Shape:Solid
    Molecular weight:651.81
  • VER-3323

    CAS:
    VER-3323 is a selective agonist for the 5-HT2B and 5-HT2C serotonin receptor with potent anorectic effects in animal studies.
    Formula:C11H15BrN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:255.15
  • Reproterol hydrochloride

    CAS:
    Reproterol hydrochloride, a β2 adrenoreceptor agonist, is used to treat asthma and chronic obstructive pulmonary disease (COPD).
    Formula:C18H24ClN5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:425.87
  • XCC

    CAS:
    XCC is an Adenosine receptor antagonist.
    Formula:C19H22N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:386.4
  • U 101958

    CAS:
    U 101958 is a putative antipsychotic agent It is also a highly selective dopamine D4 receptor antagonist.
    Formula:C20H27N3O
    Color and Shape:Solid
    Molecular weight:325.45
  • ZCZ011

    CAS:
    ZCZ011 enhances CB1 receptor effects, crosses blood-brain barrier, and potentiates cannabimimetic behaviors in mice.
    Formula:C21H18N2O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:362.44
  • Fonazine hydrochloride

    CAS:
    Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.
    Formula:C19H26ClN3O2S2
    Color and Shape:Solid
    Molecular weight:428.01
  • S1P1 Agonist III

    CAS:
    S1P1 Agonist III is an orally active S1P1 receptor agonist (EC₅₀ = 18 nM) with applications in inflammation, immunology, and receptor signaling studies.
    Formula:C21H16F3N3O3
    Purity:99.08%
    Color and Shape:Solid
    Molecular weight:415.37
  • HEAT hydrochloride

    CAS:
    HEAT hydrochloride is an α1-adrenoceptor antagonist.
    Formula:C19H22ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:331.84
  • Sch 40120

    CAS:
    Sch 40120 is an inhibitor of 5-lipoxygenase.
    Formula:C18H15ClN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:310.78
  • CAD031

    CAS:
    <p>CAD031, a more active derivative of the Alzheimer's disease (AD) targeting agent J147, exhibits neuroprotective and memory-enhancing properties.</p>
    Formula:C18H14F6N2O2
    Color and Shape:Solid
    Molecular weight:404.31
  • Denopamine

    CAS:
    Denopamine is an agonist of 1-Adrenoceptor.
    Formula:C18H23NO4
    Color and Shape:Solid
    Molecular weight:317.38
  • MRS2690

    CAS:
    MRS2690 is a potent P2Y14 receptor agonist (EC50 = 49 nM) that displays 7-fold higher potency than UDP-glucose.
    Formula:C15H24N2O16P2S
    Color and Shape:Solid
    Molecular weight:582.37
  • SEP-363856

    CAS:
    <p>SEP-363856, a non-D2/5-HT2A, orally active CNS psychotropic may treat schizophrenia.</p>
    Formula:C9H13NOS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:183.27
  • 5-trans-Prostaglandin E2

    CAS:
    5-trans-PGE2 speeds up fibrinolysis, boosts tissue-PA mediated plasminogen activation, and blocks platelet clumping in human PRP.
    Formula:C20H32O5
    Color and Shape:Solid
    Molecular weight:352.47
  • Toreforant

    CAS:
    Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).
    Formula:C23H32N6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.54
  • TISCH

    CAS:
    TISCH is a potent and selective iodinated ligand for CNS D1 dopamine receptor.
    Formula:C17H17ClINO
    Color and Shape:Solid
    Molecular weight:413.68
  • JTC-017

    CAS:
    JTC-017 is an antagonist of Corticotropin-releasing hormone receptor 1.
    Formula:C20H25Cl2N3O5S
    Color and Shape:Solid
    Molecular weight:490.4
  • Fonazine mesylate

    CAS:
    Fonazine mesylate is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.
    Formula:C20H29N3O5S3
    Color and Shape:Solid
    Molecular weight:487.65
  • Flerobuterol HCl

    CAS:
    "Flerobuterol, a β adrenergic agonist, may treat depression by boosting serotonin synthesis and Trp in the brain."
    Formula:C12H19ClFNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:247.74
  • Zimelidine

    CAS:
    Zimelidine, a withdrawn antidepressant, posed Guillain-Barre risk.
    Formula:C16H17BrN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:317.22
  • RP-72540

    CAS:
    RP-72540: CCKB receptor blocker, 200x more selective for CCKA, binds to stomach gastrin, limits [3H]pCCK-8 in mouse brain, <0.01% reaches forebrain.
    Formula:C28H30N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:518.56
  • hBChE-IN-2

    CAS:
    <p>hBChE-IN-2 is a BChE inhibitor and CB2R agonist with neuroprotective activity for the study of Alzheimer's disease-like neurological disorders.</p>
    Formula:C27H36N4O3
    Purity:99.60% - 99.83%
    Color and Shape:Soild
    Molecular weight:464.6
  • Usmarapride free base

    CAS:
    Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.
    Formula:C21H29N5O2
    Purity:99.91% - 99.91%
    Color and Shape:Solid
    Molecular weight:383.49
  • Sulfisoxazole diethanolamine

    CAS:
    Sulfisoxazole diethanolamine: a sulfonamide antibacterial, endothelin receptors A and B antagonist, inhibits breast cancer exosomes.
    Formula:C15H24N4O5S
    Color and Shape:Solid
    Molecular weight:372.44
  • A-971432

    CAS:
    A-971432: selective S1P5 agonist, IC50 = 0.006 µM. Enhances blood-brain barrier, reduces Huntington’s symptoms in mice at 0.1 mg/kg.
    Formula:C18H17Cl2NO3
    Color and Shape:Solid
    Molecular weight:366.24
  • Brl 22321

    CAS:
    Brl 22321 is a mast cell stabilizer.
    Formula:C12H9N3O2
    Color and Shape:Solid
    Molecular weight:227.22
  • Isoetharine

    CAS:
    Isoetharine is a selective agonist of β2-adrenergic receptor used as a bronchodilator for emphysema, bronchitis, and asthma.
    Formula:C13H21NO3
    Color and Shape:Solid
    Molecular weight:239.31
  • Imnopitant

    CAS:
    Imnopitant is an antagonist of the NK1 receptor [1].
    Formula:C28H28F6N4O
    Color and Shape:Solid
    Molecular weight:550.54
  • (R)-Bambuterol

    CAS:
    Bambuterol is a β2-agonist prodrug for asthma and COPD, taken daily, with a good safety profile and reduces plasma LDL-C and cholesterol.
    Formula:C18H29N3O5
    Color and Shape:Solid
    Molecular weight:367.44
  • AZD-2207

    CAS:
    AZD-2207 is a cannabinoid receptor CB1 antagonist and highly lipophilic compound for the treatment of type 2 diabetes mellitus and obesity.
    Formula:C25H25Cl2F3N4O4S
    Color and Shape:Solid
    Molecular weight:605.46
  • Cannabicitran

    CAS:
    Cannabicitran is a cannabinoid that can decrease rabbits intraocular pressure [1] [2].
    Formula:C21H30O2
    Color and Shape:Solid
    Molecular weight:314.46
  • FR-171113

    CAS:
    Protease-activated receptor 1 antagonist
    Formula:C19H11Cl3N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:469.73
  • Atrasentan hydrochloride

    CAS:
    Atrasentan hydrochloride (ABT-627 hydrochloride) is an antagonist of the endothelin receptor(IC50 = 55.1 μM for ETA).
    Formula:C29H39ClN2O6
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:547.08
  • ADR-851 HCl

    CAS:
    ADR-851 HCl is an HT3 receptor antagonist. It works against mechanical, acute thermal, and formalin-induced inflammatory pain.
    Formula:C14H19Cl2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:332.23
  • VUF8504

    CAS:
    VUF8504 is a novel ligand of adenosine A3 receptor.
    Formula:C22H17N3O2
    Color and Shape:Solid
    Molecular weight:355.39
  • E2508

    CAS:
    E2508 is a selective antagonist of corticotropin-releasing factor 1 receptor.
    Formula:C36H47N3O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:665.84
  • Trimipramine

    CAS:
    Trimipramine is an antidepressant with an anxiety-reducing sedative component to its action.
    Formula:C20H26N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:294.43
  • BL 6341A

    CAS:
    BL 6341A is related to Tumor data and H2-antagonists or anti-histamins
    Formula:C9H14N8OS3
    Color and Shape:Solid
    Molecular weight:346.46
  • FR 139317

    CAS:
    highly potent and selective ETA endothelin receptor antagonist
    Formula:C33H44N6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:604.74
  • Carbuterol hydrochloride

    CAS:
    Carbuterol hydrochloride is a short-acting β2 adrenoreceptor agonist.
    Formula:C13H22ClN3O3
    Color and Shape:Solid
    Molecular weight:303.79
  • S-22153

    CAS:
    <p>S22153 is an antagonist of melatonin receptor.</p>
    Formula:C14H17NOS
    Color and Shape:Solid
    Molecular weight:247.36
  • GR 128107

    CAS:
    GR 128107 is an antagonist of melatonin receptor.
    Formula:C16H20N2O2
    Color and Shape:Solid
    Molecular weight:272.34
  • Cgp 52608

    CAS:
    CGP 52608 is a selective ligand for RAR-associated orphan receptor alpha.
    Formula:C8H12N4OS2
    Color and Shape:Solid
    Molecular weight:244.34
  • HAMI 3379

    CAS:
    HAMI 3379 (HAMI3379) is a CysLT2 antagonist that attenuates brain damage and inhibits microglia inflammation following focal cerebral ischemia in rats.
    Formula:C34H45NO8
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:595.72
  • PF-06412154 HCl

    CAS:
    PF-06412154 HCl is a glucagon receptor antagonist.
    Formula:C24H28ClN3O3
    Color and Shape:Solid
    Molecular weight:441.96
  • Thromboxane B2

    CAS:
    Thromboxane B2 is a prostaglandin derivative that is released during anaphylaxis. Thromboxane B2 induces platelet aggregation and arterial contraction.
    Formula:C20H34O6
    Color and Shape:Solid
    Molecular weight:370.48
  • Benzamide Derivative 1

    CAS:
    Benzamide Derivative 1 Benzamide derivative with gastrokinetic activity.Benzamide Derivative 1 can be used in the study of gastrointestinal diseases.
    Formula:C22H34ClN3O3
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:423.98
  • Clenproperol

    CAS:
    Clenproperol is a β2-adrenergic agonist.
    Formula:C11H16Cl2N2O
    Color and Shape:Solid
    Molecular weight:263.16
  • PF-04628935

    CAS:
    PF-04628935: potent GHS-R1a antagonist/inverse agonist, IC50=4.6 nM, orally bioavailable, brain penetrant.
    Formula:C24H26ClN7OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:496.03
  • OUP-186

    CAS:
    OUP-186 is a selective H3 receptor antagonist that suppresses breast cancer cell growth with an IC50 of ~50 μM and induces apoptosis.
    Formula:C19H30ClN3S
    Color and Shape:Solid
    Molecular weight:367.98
  • (2R,3R)-E1R

    CAS:
    (2R,3R)-E1R is an enantiomer of E1R. (2R,3R)-E1R is a sigma-1 receptor positive allosteric modulator for the treatment of cognition/memory disorders.
    Formula:C13H16N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:232.28
  • Prostaglandin D2

    CAS:
    <p>Prostaglandin D2 (PGD2) is one of the major PGs actively produced in the brain of various mammals,and is a potent endogenous sleep promoting substances.</p>
    Formula:C20H32O5
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:352.47
  • Amosulalol, (+)-

    CAS:
    Amosulalol, (+)-, is an adrenergic agent.
    Formula:C18H24N2O5S
    Color and Shape:Solid
    Molecular weight:380.46
  • CP-122721

    CAS:
    CP-122721: NK1 receptor blocker, has antidepressant, anti-anxiety, antiemetic effects, and selectively inhibits substance P receptors.
    Formula:C20H23F3N2O2
    Color and Shape:Solid
    Molecular weight:380.4
  • Zinterol

    CAS:
    <p>Zinterol is a potent and selective agonist of β2-adrenoceptor. Zinterol increases ICa in a concentration-dependent manner(EC50 of 2.2 nM).</p>
    Formula:C19H26N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:378.49
  • Z-335 sodium

    CAS:
    Z-335 Salt, a thromboxane A2 receptor antagonist, is used potentially for the treatment of arterial occlusive disease.
    Formula:C18H18ClNNaO4S
    Color and Shape:Solid
    Molecular weight:402.84
  • YM-430

    CAS:
    YM-430: β1 blocker & Ca²⁺ channel antagonist; antianginal & antihypertensive; IC50: 59.2 nM (rhythmic contractions), 36.6 mg/kg in rats (ST depression).
    Formula:C29H35N3O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:553.6
  • Pirepemat fumarate

    CAS:
    Pirepemat fumarate (IRL752), aids Parkinson's research, boosts cognition and cortical catecholamine transmission.
    Formula:C15H17F2NO5
    Color and Shape:Solid
    Molecular weight:329.3
  • U-101958 Maleate

    CAS:
    U-101958 Maleate binds to dopamine D4 and sigma1 receptors with high affinity in neuroblastoma cells and human cerebellum.
    Formula:C25H33N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:455.55
  • NGD 98-2

    CAS:
    NGD 98-2 is a new generation, topology 2 selective orally active corticotropin releasing factor-1 (CRF-1) receptor antagonist.
    Formula:C19H24F3N3O3
    Color and Shape:Solid
    Molecular weight:399.41
  • Trimazosin hydrochloride

    CAS:
    Trimazosin hydrochloride is used in the treatment of hypertensive patients failing to respond to thiazides.
    Formula:C20H32ClN5O7
    Color and Shape:Solid
    Molecular weight:489.95
  • mCPBG

    CAS:
    mCPBG is a potent high affinity agonist of 5-HT3 receptor.
    Formula:C8H10ClN5
    Color and Shape:Solid
    Molecular weight:211.65
  • ChemR23-IN-2

    CAS:
    ChemR23-IN-2 is a potent, orally active inhibitor of ChemR23 (IC50: 3.2 nM).
    Formula:C29H26N4O5
    Color and Shape:Solid
    Molecular weight:510.54
  • RX821002

    CAS:
    RX821002: potent α2-adrenoceptor antagonist, selective for α2D (pKd 9.7) over α2A (pKd 8.2), low affinity for imidazoline.
    Formula:C12H14N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:234.25
  • GTS-21

    CAS:
    GTS-21 (DMXB-A) is an α7 nAChR agonist. GTS-21 suppresses inflammation associated with rheumatoid arthritis by inhibiting RA Th1 cell differentiation.
    Formula:C19H20N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:308.37
  • (R)-Azelastine

    CAS:
    (R)-Azelastine, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.
    Formula:C22H24ClN3O
    Color and Shape:Solid
    Molecular weight:381.9
  • TP-680

    CAS:
    TP-680 is a antagonist of cholecystokininA receptor.
    Formula:C35H33N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:619.73
  • Eptapirone fumarate

    CAS:
    Eptapirone (F11440) is a strong 5HT1A agonist with high anxiolytic and antidepressant effects, more potent than buspirone and flesinoxan.
    Formula:C20H27N7O6
    Color and Shape:Solid
    Molecular weight:461.479
  • Abanoquil

    CAS:
    Abanoquil is an antagonist of alpha-1 adrenoceptor.
    Formula:C22H25N3O4
    Color and Shape:Solid
    Molecular weight:395.45
  • Metitepine

    CAS:
    Metitepine is a serotonin receptor antagonist in the CNS used as an antipsychotic.
    Formula:C20H24N2S2
    Color and Shape:Solid
    Molecular weight:356.55