GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5972 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
YM 16638
CAS:YM 16638 is an LT antagonist that can be used to study antigen-induced early and late airway responses in allergic sheep.Formula:C18H22N2O5S3Purity:99.18%Color and Shape:SolidMolecular weight:442.575-OMe-UDP trisodium salt
CAS:Potent P2Y6 agonistFormula:C10H16N2O13P2Purity:98%Color and Shape:SolidMolecular weight:434.19Neurokinin B acetate(86933-75-7 free base)
Neurokinin B acetate, a tachykinin, interacts with NK1R, NK2R, & NK3R receptors to exert biological effects.Formula:C57H83N13O16S2Purity:98.53%Color and Shape:SolidMolecular weight:1270.48Jmv 167
CAS:Jmv 167 is an antagonist of the Cholecystokinin receptor.Formula:C51H68N8O14SPurity:98%Color and Shape:SolidMolecular weight:1049.21Leukotriene B4 Ethanolamide
CAS:<p>LTB4 binds to BLT1 (high affinity) and BLT2. LTB4-EA, a metabolite, is a stronger BLT1 antagonist, suggesting anti-inflammatory properties.</p>Formula:C22H37NO4Color and Shape:SolidMolecular weight:379.541HAEGTFT
CAS:HAEGTFT is the first N-terminal 1-7 residues of GLP-1 peptide.Formula:C33H47N9O12Purity:98%Color and Shape:SolidMolecular weight:761.78CH 275
CAS:Potent sst1 agonist with 30.9 nM IC50; selective over sst2-5; inhibits somatostatin in rat nucleus accumbens.Formula:C74H96N14O15S2Purity:98%Color and Shape:SolidMolecular weight:1485.8HAEGTFTSD acetate(926018-45-3 free base)
HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is a product of the preproglucagon gene, which is secreted fromFormula:C42H61N11O19Purity:98%Color and Shape:SolidMolecular weight:1024.01LysoPalloT-NH-amide-C3-ph-m-O-C11
CAS:LysoPalloT-NH-amide-C3-ph-m-O-C11 is an agonist of the GPR174 receptor with an EC50 value of 34 nM.Formula:C27H47N2O9PColor and Shape:SolidMolecular weight:574.64Kisspeptin-10, human
CAS:Kisspeptin-10, human is an effective vasoconstrictor and inhibitor of angiogenesis.Formula:C63H83N17O14Purity:98%Color and Shape:SolidMolecular weight:1302.462LEK 8804
CAS:LEK 8804 is a 5-HT(2) receptor antagonist and 5-HT(1A) receptor agonist.Formula:C19H19N3OColor and Shape:SolidMolecular weight:305.37Apelin-36(human)
CAS:Endogenous APJ agonist, EC50=20nM, regulates cardiovascular function, fluid balance, and feeding; blocks certain HIV strains.Formula:C184H297N69O43SPurity:98%Color and Shape:SolidMolecular weight:4195.87Parstatin(human)
CAS:Cell-permeable PAR1-derived peptide; inhibits endothelial migration, proliferation (IC50 ~3μM), induces apoptosis, and has cardioprotective effects.Formula:C191H330N64O53S3Purity:98%Color and Shape:SolidMolecular weight:4467.29Phenoxybenzamine
CAS:Phenoxybenzamine blocks α-1 receptors, potentially reducing neuroinflammation post brain trauma.Formula:C18H22ClNOPurity:98%Color and Shape:Crystals From Petroleum Ether SolidMolecular weight:303.83Ono 3708
CAS:Ono-3708 is a potent antagonist of the thromboxane A2/prostaglandin endoperoxide receptor in vitro and in vivo.Formula:C23H37NO4Purity:98%Color and Shape:SolidMolecular weight:391.54RVD-Hpα
CAS:N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.Formula:C65H105N19O17Purity:98%Color and Shape:SolidMolecular weight:1424.66Dexchlorpheniramine free base
CAS:Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.Formula:C16H19ClN2Purity:98%Color and Shape:Oily Liquid SolidMolecular weight:274.79Apraglutide
CAS:Apraglutide (FE 203799 is a synthetic 33-amino acid peptide and long-acting glp-2 analogue.Formula:C172H263N43O52Purity:98%Color and Shape:SolidMolecular weight:3765.25Dexbrompheniramine maleate
CAS:Dexbrompheniramine is an antihistamine used for hay fever and urticaria, blocking H1 receptors in the body.Formula:C20H23BrN2O4Color and Shape:SolidMolecular weight:435.318Benzoquinamide hydrochloride
CAS:Benzoquinamide hydrochloride (3-carbamoyl-N,N-diethyl-1,3,4,6,7,11b-hexahydro-9,11-dimethoxy-2H-benzo[a]quinolizin-2-yl acetate hydrochloride) is an antiemeticFormula:C22H33ClN2O5Purity:97.13% - 99.56%Color and Shape:SolidMolecular weight:440.96[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide
CAS:Potent, selective NPY Y5 receptor agonist; IC50: 0.24 nM (Y5), >500 nM (Y2), 530 nM (Y1), 51 nM (Y4); Ki: 0.1-0.15 nM (Y5); increases food intake in vivo.Formula:C183H281N57O54S2Purity:98%Color and Shape:SolidMolecular weight:4207.67[D-Phe12]-Bombesin
CAS:<p>Bombesin receptor antagonist</p>Formula:C74H112N22O18SPurity:98%Color and Shape:SolidMolecular weight:1629.88Azirkitug
Azirkitug is a humanized IgG1κ antibody targeting CCR8, with HumanIgG1kappa, Isotype Control serving as its corresponding isotype control.Color and Shape:Odour LiquidNeurokinin B
CAS:NKB, a tachykinin peptide, impacts human functions like gonadotropin-releasing hormone secretion.Formula:C55H79N13O14S2Purity:98%Color and Shape:SolidMolecular weight:1210.42Adenosine 2',5'-diphosphate sodium
CAS:Adenosine 2',5'-diphosphate sodium is a competitive P2Y1 antagonist with non-selective antagonism at recombinant and human platelet P2X1 receptors.Formula:C10H15N5NaO10P2Color and Shape:SolidMolecular weight:450.192SHU 9119
CAS:SHU 9119 is a potent antagonist for human MC3R/MC4R and partial agonist for MC5R with IC50 values of 0.23, 0.06, 0.09 nM.Formula:C54H71N15O9Purity:98%Color and Shape:SolidMolecular weight:1074.258L-779976
CAS:L-779,976 is an agonist of somatostatin receptor.Formula:C33H43N7O3Color and Shape:SolidMolecular weight:585.74Glucagon receptor antagonists-1
CAS:Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.Formula:C29H34FNO2Purity:98%Color and Shape:SolidMolecular weight:447.58Adrenomedullin (11-50), rat
CAS:Adrenomedullin 11-50 rat is a peptide, stimulates CGRP1 receptor for vasodilation, used in bone growth research.Formula:C194H304N58O59S4Purity:98%Color and Shape:SolidMolecular weight:4521.17Amylin (8-37), human
CAS:Human-derived Amylin (8-37) is a vasodilator in rat arteries and forms aggregates linked to type II diabetes.Formula:C138H216N42O45Color and Shape:SolidMolecular weight:3183.495Methapyrilene hydrochloride
CAS:Methapyrilene hydrochloride is a biochemical.Formula:C14H20ClN3SColor and Shape:Liquid Solution) 5 5 (Ntp 1992)Molecular weight:297.85IRL-1620
CAS:IRL-1620 is an effective and selective agonist of endothelin receptor type B (ETB) (Ki: 16 pM).Formula:C86H117N17O27Purity:98%Color and Shape:SolidMolecular weight:1820.974Prazobind
CAS:Prazobind is a prazosinoid substance that blocks insulin stimulation of IP1 (inositol phosphate) accumulation and is an effective α1 adrenoceptor blocker.Formula:C23H27N5O3Color and Shape:SolidMolecular weight:421.501α-CGRP, rat
CAS:Endogenous neuropeptide, potent vasodilatorFormula:C162H262N50O52S2Purity:98%Color and Shape:SolidMolecular weight:3806.2515(S)-15-methyl Prostaglandin F2α methyl ester
CAS:15(S)-15-methyl Prostaglandin F2α methyl ester can be used in related research in the field of life sciences.Formula:C22H38O5Color and Shape:SolidMolecular weight:382.53IRL-1038
CAS:<p>ETB endothelin receptor antagonist</p>Formula:C68H92N14O15S2Purity:98%Color and Shape:SolidMolecular weight:1409.67Pneumadin, rat
CAS:Rat Pneumadin (PNM), a decapeptide, stimulates AVP release, exerting strong antidiuretic effects in animals with an active AVP system.Formula:C47H74N12O15Purity:98%Color and Shape:SolidMolecular weight:1047.17816,16-dimethyl Prostaglandin F2α
CAS:<p>16,16-dimethyl Prostaglandin F2α can be used in related research in the field of life sciences. Its product number is T37993 and CAS number is 39746-23-1.</p>Formula:C22H38O5Color and Shape:SolidMolecular weight:382.541Cortistatin-29 (rat) (trifluoroacetate salt)
CAS:Cortistatin-29, similar to somatostatin-28, derives from preprocortistatin and binds to SST receptors 1-5 with varying IC50 values.Formula:C161H240N46O41S2Color and Shape:SolidMolecular weight:3540.09β-CGRP, human
CAS:β-CGRP, human ,a 37-amino acid peptide,is the beta form of Calcitonin-gene-related peptide (β-CGRP), involved extensively in regulation of the cardiovascularFormula:C162H267N51O48S3Purity:98%Color and Shape:SolidMolecular weight:3793.41PACAP-38 (16-38), human, mouse, rat
CAS:PACAP-38 (16-38), human, mouse, rat demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal NPY and catecholamine productionFormula:C123H215N39O28SPurity:98%Color and Shape:SolidMolecular weight:2720.33ELA-21 (human)
CAS:Apelin receptor agonist with high affinity for normal/PAH hearts (pKi 9.31/9.46). Blocks cAMP, promotes β-arrestin in vitro. Part of ELA-32.Formula:C112H184N40O25S3Purity:98%Color and Shape:SolidMolecular weight:2587.12RFRP-3(human)
CAS:NPFF1 receptor agonist, IC50 0.7 nM, blocks cAMP by forskolin. A GnIH homolog, it inhibits GnRH neuron activity.Formula:C45H72N14O10Purity:98%Color and Shape:SolidMolecular weight:969.15Neuropeptide S(Rat)
CAS:Potent endogenous neuropeptide S receptor (NSPR) agonist (EC50 = 3.2 nM).Formula:C95H160N34O27Purity:98%Color and Shape:SolidMolecular weight:2210.52(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
CAS:V1A receptor antagonist; blocks vasopressin & oxytocin, lowers Ca²⁺ levels (IC50: 5/30 nM); long-acting antivasopressor; anxiolytic in dorsal hippocampus.Formula:C52H74N14O12S2Purity:98%Color and Shape:White Lyophilized PowderMolecular weight:1151.38ARL 15849XX
CAS:ARL 15849XX, a CCK-8 analog, is a novel anti-obesity agent.Formula:C47H60N8O13SPurity:98%Color and Shape:SolidMolecular weight:977.09Antibiotic Sch 60057
CAS:Antibiotic Sch 60057 is a useful organic compound for research related to life sciences. The catalog number is T125403 and the CAS number is 203061-35-2.Formula:C45H84O6Color and Shape:SolidMolecular weight:721.161(D-Trp6)-LHRH free acid
CAS:(D-Trp6)-LHRH free acid is a luteinizing hormone-releasing hormone ( LHRH ) agonist [1] .Formula:C64H81N17O14Molecular weight:1312.43DOTA-EB-TATE
DOTA-EB-TATE is formed by combining the SST peptide derivative DOTA-octreotate with an Evans blue analog (EB). This peptide drug conjugate (PDC) enhances the pharmacokinetics of SSTR2 analogs and reduces PRRT toxicity. Additionally, DOTA-EB-TATE serves in the synthesis/research of radiopharmaceutical conjugates (RDC).Formula:C105H133N21O30S5Molecular weight:2329.6316-phenoxy tetranor Prostaglandin F2α
CAS:16-phenoxy PGF2α is a metabolically stable analog of PGF2α. It binds to the FP receptor on ovine luteal cells with much greater affinity (440%) than PGF2α.Formula:C22H30O6Color and Shape:SolidMolecular weight:390.47
![[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1963.webp&w=3840&q=75)
![[D-Phe12]-Bombesin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP2239.webp&w=3840&q=75)
