GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(3,031 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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Decynium 22
CAS:Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitorFormula:C23H23IN2Purity:99.92%Color and Shape:Dark Red CrystalsMolecular weight:454.35Ritanserin
CAS:Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Formula:C27H25F2N3OSPurity:99.77% - 99.89%Color and Shape:SolidMolecular weight:477.57Aripiprazole monohydrate
CAS:Aripiprazole (OPC-14597) is a potent D2 partial agonist and inverse agonist of 5-HT2 receptors, used for schizophrenia and COVID-19 studies.Formula:C23H29Cl2N3O3Color and Shape:SolidMolecular weight:466.4Renzapride hydrochloride
CAS:Renzapride is a 5-HT3 antagonist and 5-HT4 agonist. Renzapride also functions as a 5-HT2B antagonist and has some affinity for the 5-HT2A and 5-HT2C receptors.Formula:C16H23Cl2N3O2Color and Shape:SolidMolecular weight:360.28Maropitant
CAS:Maropitant is a selective neurokinin (NK1) receptor antagonist.Formula:C32H40N2OPurity:97.35% - 99.75%Color and Shape:SolidMolecular weight:468.67Ref: TM-T7209
5mg50.00€10mg80.00€25mg116.00€50mg212.00€100mg316.00€200mg454.00€1mL*10mM (DMSO)To inquireCYM-5520
CAS:CYM-5520 is a noncompetitive allosteric agonist of S1P2Formula:C21H19N3O2Purity:99.47%Color and Shape:SolidMolecular weight:345.39Ref: TM-T22703
1mg46.00€2mg60.00€5mg88.00€10mg135.00€25mg236.00€50mg354.00€100mg528.00€1mL*10mM (DMSO)98.00€MK 571
CAS:MK 571 (L660711) is an orally active antagonist of CysLT1 receptor.Formula:C26H27ClN2O3S2Purity:98.69% - 99.65%Color and Shape:SolidMolecular weight:515.09Ref: TM-T7841
2mg34.00€5mg50.00€10mg81.00€25mg165.00€50mg285.00€100mg432.00€200mg617.00€1mL*10mM (DMSO)59.00€HAEGTFTSDVSSYLE
HAEGTFTSDVSSYLE is a peptide. GLP-I analog contains the sequence.
Formula:C71H103N17O28Purity:>99.99%Color and Shape:SolidMolecular weight:1642.71Mecamylamine
CAS:Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.Formula:C11H21NColor and Shape:SolidMolecular weight:167.29Trimethobenzamide hydrochloride
CAS:Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.Formula:C21H29ClN2O5Purity:99.52%Color and Shape:SolidMolecular weight:424.921-(1-Naphthyl) piperazine hydrochloride
CAS:1-(1-Naphthyl) piperazine hydrochloride (1-naphthalen-1-ylpiperazine hydrochloride) is a serotonergic ligand which could bind nonselectively with multiple
Formula:C14H17ClN2Purity:98.27%Color and Shape:SolidMolecular weight:248.75CRF (6-33) acetate(120066-38-8 free base)
CRFBP inhibitor peptide; reduces weight gain, boosts activity in obese rats.Formula:C143H235N41O45SPurity:97.12%Color and Shape:SolidMolecular weight:3280.76GSK2018682 HCl
CAS:GSK2018682 is a novel sphingosine-1-phosphate receptor 1 (s1p1) and 5 (s1p5) agonist.Formula:C22H22Cl2N4O4Color and Shape:SolidMolecular weight:477.34TNCA
CAS:TNCA (Lycoperodine-1) is a high-affinity CaSR ligand (CaSRL) with co-agonist activity.Formula:C12H12N2O2Purity:97.33% - 97.73%Color and Shape:SolidMolecular weight:216.24Clobenpropit 2HBr
CAS:Clobenpropit 2HBr is a histamine H3 receptor antagonist. It has neuroprotective effects via stimulation of GABA release in the brain.Formula:C14H17ClN4SColor and Shape:SolidMolecular weight:308.83L-DOPA methyl ester (hydrochloride)
CAS:L-DOPA methyl ester (LDME) is an agonist of dopamine D1 receptor.
Formula:C10H14ClNO4Purity:98.69% - 99.81%Color and Shape:White SolidMolecular weight:247.675SB 242084 dihydrochloride
CAS:SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9.0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively.Formula:C21H21Cl3N4O2Color and Shape:SolidMolecular weight:467.78ML 10302
CAS:ML 10302 is a potent 5-HT4 agonist with Ki of 1.07 nM, boosts bowel movement, and may aid in neurology research.Formula:C15H21ClN2O3Color and Shape:SolidMolecular weight:312.79CRT0273750
CAS:CRT0273750 regulates plasma LPA levels and is suitable for in vivo studies. CRT0273750 is an autotaxin (ATX) inhibitor with IC50 of 0.014 μM.Formula:C25H22ClF3N4O2Purity:99.91%Color and Shape:SolidMolecular weight:502.92Pipamperone HCl
CAS:Pipamperone blocks 5-HT2A/B/C, D2/D3/D4, α1/α2 receptors; favors 5-HT2A/D4 over D2; negligible affinity for H1, mACh. Highly selective at low doses.Formula:C21H31ClFN3O2Color and Shape:SolidMolecular weight:411.95Phentolamine
CAS:Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonistFormula:C17H19N3OPurity:99.86% - 99.94%Color and Shape:Crystals SolidMolecular weight:281.35Metoclopramide dihydrochloride
CAS:Metoclopramide dihydrochloride is a dopamine D2 antagonist that is used as an antiemetic.Formula:C14H24Cl3N3O2Color and Shape:SolidMolecular weight:372.72Fluparoxan HCl
CAS:Fluparoxan is a potent α2-adrenergic receptor antagonist (pKB = 7.9) with excellent α2/α1 selectivity (2630 fold).Formula:C10H11ClFNO2Color and Shape:SolidMolecular weight:231.65Vilanterol trifenatate
CAS:Vilanterol trifenatate is a long-acting agonist of β2-adrenoceptor (β2-AR) with inherent 24-hour activity(β2-AR, β1-AR and β3-AR pEC50s of 10.37, 6.98 and 7.36, respectively)Formula:C44H49Cl2NO7Purity:99.51% - >99.99%Color and Shape:SolidMolecular weight:774.77BGC-20-1531 hydrochloride(1186532-61-5 free base)
CAS:BGC-20-1531 hydrochloride(1186532-61-5 free base) (GTPL3380 hydrochloride) is a EP4 antagonist for the treatment of acute migraine.
Formula:C26H25ClN2O6SPurity:98.94% - 99.85%Color and Shape:SolidMolecular weight:529Cutamesine dihydrochloride
CAS:Cutamesine dihydrochloride is a σ1 receptor agonist, selective over σ2, combating cardiomyocyte hypertrophy and improving stroke recovery.Formula:C23H32N2O2·2HClPurity:99.96%Color and Shape:SolidMolecular weight:441.43Ref: TM-T3597
2mg34.00€5mg50.00€10mg86.00€25mg167.00€50mg260.00€100mg401.00€200mg580.00€1mL*10mM (DMSO)55.00€FK962
CAS:FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.Formula:C14H17FN2O2Purity:99.89%Color and Shape:SolidMolecular weight:264.3Ref: TM-T7829
2mg34.00€5mg52.00€10mg82.00€25mg144.00€50mg200.00€100mg278.00€200mg389.00€1mL*10mM (DMSO)57.00€Arformoterol Tartrate
CAS:Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.Formula:C23H30N2O10Purity:99.98%Color and Shape:SolidMolecular weight:494.49Ref: TM-T22245
5mg60.00€10mg87.00€25mg150.00€50mg221.00€100mg329.00€200mg487.00€1mL*10mM (DMSO)85.00€Bromodiphenhydramine hydrochloride
CAS:Bromodiphenhydramine hydrochloride is a new antihistaminic in the control of cutaneous.Formula:C17H21BrClNOPurity:97.29%Color and Shape:SolidMolecular weight:370.71Protease-Activated Receptor-2, amide
CAS:Protease-Activated Receptor-2, amide (SLIGKV-NH2) is an agonist of PAR2 (IC50 : 10.4 M)Formula:C28H54N8O7Purity:>99.99%Color and Shape:SolidMolecular weight:614.78Cinaciguat
CAS:Cinaciguat (BAY 58-2667) is a pioneering sGC activator for acute heart failure treatment.
Formula:C36H39NO5Purity:98% - 99.18%Color and Shape:SolidMolecular weight:565.7Picotamide
CAS:Picotamide has anticoagulant and fibrinolytic properties.Formula:C21H20N4O3Purity:98.90%Color and Shape:SolidMolecular weight:376.41Ref: TM-T9153
1mg38.00€5mg92.00€10mg147.00€25mg241.00€50mg349.00€100mg479.00€200mg657.00€1mL*10mM (DMSO)94.00€Benzotript
CAS:Benzotript is an gastrin-receptor antagonist, with anti-gastrinic.Formula:C18H15ClN2O3Purity:97.82%Color and Shape:SolidMolecular weight:342.776Ref: TM-T8578
1mg124.00€2mg178.00€5mg269.00€10mg408.00€25mg672.00€50mg945.00€100mg1,279.00€1mL*10mM (DMSO)286.00€5-Benzyloxygramine
CAS:5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.Formula:C18H20N2OPurity:99.13%Color and Shape:SolidMolecular weight:280.36Buserelin Acetate (57982-77-1 free base)
CAS:Buserelin Acetate (57982-77-1 free base) (Buserelin Acetate) is an agonist of gonadotropin-releasing hormone receptor(GnRHR).Formula:C62H90N16O15Purity:99.31% - 99.78%Color and Shape:SolidMolecular weight:1299.48Eformoterol Hemifumarate
CAS:Formoterol fumarate (Eformoterol Hemifumarate), an effective, specific and long-acting β2-adrenoceptor agonist, is utilized in the treatment of COPD and asthmaFormula:C19H24N2O4C4H4O4Purity:99.86% - >99.99%Color and Shape:White PowderMolecular weight:402.4Mecamylamine hydrochloride
CAS:Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.Formula:C11H22ClNPurity:99.76% - >99.99%Color and Shape:White SolidMolecular weight:203.75Bevantolol
CAS:Bevantolol, a selective β-1 adrenoceptor antagonist, is utilized for the investigation of angina pectoris and hypertension [1].Formula:C20H27NO4Color and Shape:SolidMolecular weight:345.43Syk Inhibitor II dihydrochloride
CAS:Syk inhibitor II selectively blocks Syk (IC50 = 41 nM), impacting platelet function and inflammation, with lower potency against other kinases.Formula:C14H17Cl2F3N6OPurity:98.53%Color and Shape:SolidMolecular weight:413.22Ref: TM-T4391
1mg130.00€2mg212.00€5mg455.00€10mg647.00€25mg947.00€50mg1,264.00€100mg1,700.00€1mL*10mM (DMSO)455.00€Nonapeptide-1
CAS:Nonapeptide-1 (Melanostatine™ 5) can inhibit the synthesis of melanin, which makes it of interest for treating certain skin conditions.Formula:C61H87N15O9SPurity:100%Color and Shape:SolidMolecular weight:1206.5Xanthine amine congener hydrochloride
CAS:Xanthine amine congener (XAC) hydrochloride is a non-selective adenosine receptor antagonist that induces convulsions in mice.Formula:C21H29ClN6O4Color and Shape:SolidMolecular weight:464.95[D-Phe12]-Bombesin acetate
[D-Phe12]-Bombesin acetate inhibits bombesin-stimulated secretion.Formula:C76H116N22O20SPurity:99.81%Color and Shape:SolidMolecular weight:1689.94Tripelennamine
CAS:Tripelennamine: ethylenediamine derivative, H1-receptor blocker, reduces allergic reactions, treats rhinitis and conjunctivitis.Formula:C16H21N3Color and Shape:SolidMolecular weight:255.36ACTH 1-14 acetate(25696-21-3 free base)
ACTH 1-14 acetate regulates cortisol and androgen, is part of the hypothalamic-pituitary-adrenal stress response.Formula:C79H113N21O22SPurity:>99.99%Color and Shape:SolidMolecular weight:1740.96Lodoxamide
CAS:Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.Formula:C11H6ClN3O6Purity:99.13% - 99.96%Color and Shape:SolidMolecular weight:311.63Ambrisentan sodium
CAS:Ambrosentan (BSF 208075) sodium is a selective and oral effective antagonist of ET type A receptor ( ETAR ).Formula:C22H21N2NaO4Color and Shape:SolidMolecular weight:400.41WAY-100635 Monomaleate
CAS:WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.Formula:C25H34N4O2·C4H4O4Purity:98.44% - 99.46%Color and Shape:SolidMolecular weight:538.64Ref: TM-T2631
2mg46.00€5mg66.00€10mg95.00€25mg180.00€50mg334.00€100mg495.00€200mg717.00€500mg1,111.00€1mL*10mM (DMSO)79.00€LM11A-31 dihydrochloride
CAS:LM11A-31 dihydrochloride is a water-soluble, BBB-penetrating p75NTR ligand and proNGF antagonist.Formula:C12H27Cl2N3O2Purity:99.47% - 99.9%Color and Shape:SolidMolecular weight:316.27Fuscoside
CAS:Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value of 0.4 μM.Cost-effective and quality-assured.Formula:C26H31N3O4Purity:98.13% - 99.66%Color and Shape:SolidMolecular weight:449.54SCH-37370
CAS:SCH-37370 is an effective and orally active dual antagonist of platelet-activating factor and histamine.Formula:C21H21ClN2OPurity:99.07%Color and Shape:SolidMolecular weight:352.86Ref: TM-T19686
1mg48.00€5mg89.00€10mg115.00€25mg195.00€50mg290.00€100mg393.00€200mg520.00€1mL*10mM (DMSO)90.00€
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