GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,023 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5986 products of "GPCR/G-Protein"
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(S)-Viloxazine Hydrochloride
CAS:(S)-Viloxazine Hydrochloride is an S-isomer and NRI used as an antidepressant.Formula:C13H20ClNO3Purity:99.95%Color and Shape:SolidMolecular weight:273.76Ref: TM-T22420
1mg34.00€5mg63.00€1mL*10mM (DMSO)65.00€10mg85.00€25mg117.00€50mg168.00€100mg239.00€500mg592.00€Octahydroisoindole
CAS:Octahydroisoindole is a natural product and a reference standard.Formula:C8H15NPurity:≥98%Color and Shape:SolidMolecular weight:125.21S(-)-8-Hydroxy-DPAT hydrobromide
CAS:S(-)-8-Hydroxy-DPAT hydrobromide is an agonist of 5-HT1A serotonin receptor.Formula:C16H26BrNOPurity:98%Color and Shape:SolidMolecular weight:328.29PD 118440
CAS:PD 118440 is a Dopamine antagonist. PD 118440 is an orally active dopamine (DA) agonists with pronounced central nervous system effects.Formula:C11H17N3SPurity:98%Color and Shape:SolidMolecular weight:223.34MK-0249
CAS:MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).
Formula:C23H24F3N3O2Purity:99.90%Color and Shape:SolidMolecular weight:431.45CCK-A receptor inhibitor 1
CAS:CCK-A receptor inhibitor 1 is a potent inhibitor of the cholecystokinin A (CCK-A) receptor (IC50: 340 nM).CCK-A receptor inhibitor 1 can be used for the studyFormula:C25H35NO6SPurity:99.47%Color and Shape:SolidMolecular weight:477.61Pamatolol
CAS:Pamatolol is a selective and potent beta-adrenoceptor antagonist that has not shown sympathomimetic activity in ex vivo experiments.Formula:C16H26N2O4Purity:>99.99%Color and Shape:SolidMolecular weight:310.39L-771688
CAS:L-771688 (SNAP 6383) is a novel potent and selective α1A-adrenoceptor antagonist with a Ki value of 0.43±0.02 nM.L-771688 KE is used for the treatment of benignFormula:C28H33F2N5O5Purity:94.15%Color and Shape:SolidMolecular weight:557.59PAF-AN-1
CAS:PAF-AN-1 is a novel potent platelet-activating factor receptor (PAF) antagonist involved in the study of anaphylactic death.Formula:C28H28N2O3Purity:98.06%Color and Shape:SolidMolecular weight:440.53TD-5471 hydrochloride
CAS:TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment of chronic obstructive pulmonary disease (Formula:C32H32ClN3O4Purity:99.57%Color and Shape:SolidMolecular weight:558.07RP73870
CAS:RP73870 is a gastrin/cholecystokinin-B receptor antagonist and H2 receptor antagonist with potent anti-ulcer activity.Formula:C27H30N4O7SPurity:98%Color and Shape:SolidMolecular weight:554.61PD 118717
CAS:PD 118717: a piperazinyl benzopyranone dopamine agonist with potential antipsychotic properties and no neurological side effects in tests.Formula:C20H22N4O3Purity:98%Color and Shape:SolidMolecular weight:366.41Argiprestocin
CAS:Argiprestocin: antidiuretic, regulates osmolality, neurohypophysial hormone, vasoconstrictor.Formula:C43H67N15O12S2Purity:99.34%Color and Shape:SolidMolecular weight:1050.22Mabuterol, (S)-
CAS:Mabuterol, a β2 adrenoreceptor agonist, lowers rat blood pressure and boosts guinea pig heart rate/force, not affecting other receptors.Formula:C13H18ClF3N2OColor and Shape:SolidMolecular weight:310.74Ambucetamide
CAS:Ambucetamide is an antispasmodic, it may inhibit or diminish the spontaneous rhythmical activity of the human myometrium.Formula:C17H28N2O2Color and Shape:SolidMolecular weight:292.42GBR-12935 maleate
CAS:GBR-12935: dopamine reuptake inhibitor, used in research for Parkinson's and brain's dopamine pathways.Formula:C32H38N2O5Color and Shape:SolidMolecular weight:530.665Dicentrine HCl
CAS:Dicentrine HCl is the salt form of Dicentrine, an alpha 1-adrenoceptor antagonist effective against human hyperplastic prostates.Formula:C20H22ClNO4Color and Shape:SolidMolecular weight:375.85Esreboxetine
CAS:Esreboxetine( PNU-165442, (S,S) -reboxetine) is a selective inhibitor of norepinephrine reuptake.Formula:C19H23NO3Color and Shape:SolidMolecular weight:313.39Bitolterol
CAS:Bitolterol is a new beta 2-adrenergic agonist and classified as a pro-drug.Formula:C28H31NO5Color and Shape:SolidMolecular weight:461.555-HT4 antagonist 1
CAS:5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).Formula:C23H36N4O5SPurity:99.75%Color and Shape:SolidMolecular weight:480.62Sch 44643
CAS:Sch 44643 is an antagonist of platelet activating factor with oral activity.Formula:C25H22ClN3O2Color and Shape:SolidMolecular weight:431.91Iferanserin HCl
CAS:Iferanserin HCl is a selective serotonin receptor antagonist.Formula:C23H29ClN2OColor and Shape:SolidMolecular weight:384.95GYKI-13380
CAS:GYKI-13380, also known as LS-79445, is a small molecule with potent bioactivity. Detail information has not been published yet.Formula:C16H22N2O3Color and Shape:SolidMolecular weight:290.36Reproterol hydrochloride
CAS:Reproterol hydrochloride, a β2 adrenoreceptor agonist, is used to treat asthma and chronic obstructive pulmonary disease (COPD).Formula:C18H24ClN5O5Purity:98%Color and Shape:SolidMolecular weight:425.87Toreforant
CAS:Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).Formula:C23H32N6Purity:98%Color and Shape:SolidMolecular weight:392.54TISCH
CAS:TISCH is a potent and selective iodinated ligand for CNS D1 dopamine receptor.Formula:C17H17ClINOColor and Shape:SolidMolecular weight:413.68Cannabicitran
CAS:Cannabicitran is a cannabinoid that can decrease rabbits intraocular pressure [1] [2].Formula:C21H30O2Color and Shape:SolidMolecular weight:314.46PF-06412154 HCl
CAS:PF-06412154 HCl is a glucagon receptor antagonist.Formula:C24H28ClN3O3Color and Shape:SolidMolecular weight:441.96Z-335 sodium
CAS:Z-335 Salt, a thromboxane A2 receptor antagonist, is used potentially for the treatment of arterial occlusive disease.Formula:C18H18ClNNaO4SColor and Shape:SolidMolecular weight:402.84Trimazosin hydrochloride
CAS:Trimazosin hydrochloride is used in the treatment of hypertensive patients failing to respond to thiazides.Formula:C20H32ClN5O7Color and Shape:SolidMolecular weight:489.95mCPBG
CAS:mCPBG is a potent high affinity agonist of 5-HT3 receptor.Formula:C8H10ClN5Color and Shape:SolidMolecular weight:211.65ChemR23-IN-2
CAS:ChemR23-IN-2 is a potent, orally active inhibitor of ChemR23 (IC50: 3.2 nM).Formula:C29H26N4O5Color and Shape:SolidMolecular weight:510.54(R)-Azelastine
CAS:(R)-Azelastine, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Formula:C22H24ClN3OColor and Shape:SolidMolecular weight:381.9Amibegron
CAS:Amibegron: oral β3 adrenergic agonist, CNS-penetrating, with antidepressant and anxiolytic properties.Formula:C22H26ClNO4Color and Shape:SolidMolecular weight:403.95-OxoETE methyl ester
CAS:5-OxoETE methyl ester is a 5-oxoETE ester, an OXER1 agonist with stronger β-arrestin response, EC50 = 1.54 μM.Formula:C21H32O3Color and Shape:SolidMolecular weight:332.48Ethiazide
CAS:Ethiazide is a benzothiadiazine sulfonamide derivative belonging to the class of the thiazide diuretics.Formula:C9H12ClN3O4S2Color and Shape:SolidMolecular weight:325.79Tiamenidine hydrochloride
CAS:Tiamenidine hydrochloride is a centrally-acting alpha1 adrenergic receptor antagonist.Formula:C8H11Cl2N3SColor and Shape:SolidMolecular weight:252.16Clopenthixol
CAS:Clopenthixol is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors.Formula:C22H25ClN2OSColor and Shape:SolidMolecular weight:400.96CM304
CAS:CM304 is a highly selective sigma-1 receptor antagonist.Formula:C18H26ClFN2OSColor and Shape:SolidMolecular weight:372.93Elzasonan
CAS:Elzasonan is a selective 5-hydroxytryptamine 1B receptor antagonist used to treat patients with major depressive disorder and obsessive compulsive disorder.Formula:C22H23Cl2N3OSColor and Shape:SolidMolecular weight:448.41Naxifylline
CAS:Naxifylline is an A1 adenosine receptor blocker that increases urine and protects kidneys during edema treatment in heart failure.Formula:C18H24N4O3Color and Shape:SolidMolecular weight:344.41SUN 1334H
CAS:SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).Formula:C23H28Cl2F2N2O3Purity:98%Color and Shape:SolidMolecular weight:489.38GAT229
CAS:GAT229 is a CB1 positive modulator, enhancing CB agonist activity without direct activation; influences binding, signaling, and lowers ocular pressure in mice.Formula:C22H18N2O2Color and Shape:SolidMolecular weight:342.39BN-81,674
CAS:BN-81,674 is a bioactive chemical.Formula:C30H38N4Color and Shape:SolidMolecular weight:454.65Seprilose
CAS:Seprilose, prostaglandin E2 inhibitor, inhibits prostaglandin E2 synthesis.Formula:C16H30O6Color and Shape:SolidMolecular weight:318.41M-25
CAS:M-25 is a Smoothened antagonist and inhibitor of the Hedgehog pathway.Formula:C23H29N3O2Color and Shape:SolidMolecular weight:379.5TR4161
CAS:TR4161 is a prostaglandin bronchodilator of low tracheobronchial irritancy.Formula:C20H36O4Color and Shape:SolidMolecular weight:340.5FK-1052 HCl
CAS:FK-1052 HCl is a serotonin 3 & 4 dual receptor antagonist.Formula:C18H20ClN3OColor and Shape:SolidMolecular weight:329.83NR2F1 agonist 1
CAS:NR2F1 agonist 1 activates cancer cell dormancy, suppresses growth in HNSCC, and inhibits tumor growth in mice.Formula:C28H30N4OSColor and Shape:SolidMolecular weight:470.63Dothiepin HCl
CAS:Dothiepin HCl: TCA, SNRI, with antihistamine, antiadrenergic, anticholinergic, and sodium block properties.Formula:C19H22ClNSColor and Shape:SolidMolecular weight:331.9
