GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,027 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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Colterol (free base)
CAS:Colterol: short-acting β2 agonist; Bitolterol prodrug treats asthma, COPD bronchospasm.Formula:C12H19NO3Color and Shape:SolidMolecular weight:225.28BN-81,674
CAS:BN-81,674 is a bioactive chemical.Formula:C30H38N4Color and Shape:SolidMolecular weight:454.65Seprilose
CAS:Seprilose, prostaglandin E2 inhibitor, inhibits prostaglandin E2 synthesis.Formula:C16H30O6Color and Shape:SolidMolecular weight:318.41Vasopressin V2 receptor antagonist 1
CAS:Vasopressin V2 receptor antagonist 1 (Compound 4g) is a vasopressin V2receptor (V2R) antagonist (Ki: 3.8 nM). dominant polycystic kidney disease (ADPKD).Formula:C33H37ClN4O4Color and Shape:SolidMolecular weight:589.12threo Ifenprodil hemitartrate
CAS:σ receptor agonist and NR2B subunit-selective NMDA receptor antagonistFormula:C21H27NO2C4H6O6Purity:98%Color and Shape:SolidMolecular weight:400.492-Methyl-5-HT maleate
CAS:2-Methyl-5-HT maleate, a selective 5-HT3 agonist, shows anti-depressive effects.Formula:C15H18N2O5Purity:98%Color and Shape:SolidMolecular weight:306.31L-817,818
CAS:somatostatin sst5 receptor agonistFormula:C33H36N4O3Purity:98%Color and Shape:SolidMolecular weight:536.66Y2 Antagonist 36
CAS:Y2 Antagonist 36 is a highly potent, soluble and selective antagonist of NPY Y2.Formula:C27H29ClN4O3Color and Shape:SolidMolecular weight:493CID1792197
CAS:CID1792197 is a selective agonist of GPR55.Formula:C24H23N3O4S2Purity:98%Color and Shape:SolidMolecular weight:481.59Reversan
CAS:Reversan(CBLC4H10) is a potent, nontoxic, and glioblastoma-associated inhibitor of multidrug resistance-associated protein 1 (MRP1) and P-glycoprotein (Pgp).Formula:C26H27N5O2Purity:99.05%Color and Shape:SolidMolecular weight:441.53Ref: TM-T12714
1mg44.00€1mL*10mM (DMSO)92.00€5mg93.00€10mg130.00€25mg250.00€50mg401.00€100mg640.00€200mg884.00€SMM-189
CAS:SMM-189 is a potent and selective CB2 inverse agonist.Formula:C19H12Cl2O3Color and Shape:SolidMolecular weight:359.2GR 196429
CAS:GR 196429: MT1-selective melatonin receptor agonist; induces sleep, alters circadian rhythm, stimulates melatonin in mice.Formula:C14H18N2O2Purity:98%Color and Shape:SolidMolecular weight:246.3GW848687X
CAS:GW848687X, a potent and selective prostaglandin EP1 receptor antagonist, is used for the treatment of inflammatory pain.Formula:C24H18ClF2NO3Purity:98%Color and Shape:SolidMolecular weight:441.85MRS2298
CAS:MRS2298, a potent antagonists of the P2Y 1 receptor, has antiaggregatory activity in human platelets.Formula:C10H16ClN5O8P2Purity:98%Color and Shape:SolidMolecular weight:431.66Ro 60-0175 fumarate
CAS:5-HT2 receptor agonistFormula:C15H16ClFN2O4Purity:98%Color and Shape:SolidMolecular weight:342.75Carcinine
CAS:Carcinine ditrifluoroacetate is a H3 receptor antagonist.Formula:C8H14N4OPurity:98%Color and Shape:SolidMolecular weight:182.22L-Alprenolol
CAS:L-Alprenolol is a non-selective beta-blocker and a 5-HT1A and 5-HT1B receptor antagonist.Formula:C15H23NO2Purity:98%Color and Shape:SolidMolecular weight:249.35(RS)-Butyryltimolol
CAS:(RS)-Butyryltimolol, a racemic prodrug of Timolol, enhances its corneal absorption and acts as a β-adrenergic blocker.Formula:C17H30N4O4SPurity:98%Color and Shape:SolidMolecular weight:386.51Benzatropine
CAS:Benzatropine: Central muscarinic blocker, inhibits dopamine uptake, treats Parkinson's symptoms.Formula:C21H25NOPurity:98%Color and Shape:SolidMolecular weight:307.43A 49816
CAS:A 49816 is a high-ceiling diuretic.Formula:C18H17Cl2NO5Color and Shape:SolidMolecular weight:398.24γ-Linolenic acid ethyl ester
CAS:γ-Linolenic acid ethyl ester (Ethyl γ-linolenate) is a leukotriene B 4 receptor 4 (LTB 4 ) antagonist which has a potential anti-inflammatory effect[1].Formula:C20H34O2Color and Shape:SolidMolecular weight:306.48Stresson
CAS:Stresson is a beta-blocking agent bunitrolol.Formula:C14H21ClN2O2Color and Shape:SolidMolecular weight:284.78Levemopamil HCl
CAS:Levemopamil HCl is used as a calcium channel blocker.Formula:C23H31ClN2Purity:98%Color and Shape:SolidMolecular weight:370.96TR4161
CAS:TR4161 is a prostaglandin bronchodilator of low tracheobronchial irritancy.Formula:C20H36O4Color and Shape:SolidMolecular weight:340.5hGPR91 antagonist 3
CAS:hGPR91 antagonist 3 is an hGPR91 antagonist. hGPR91 antagonist 3 can be used to study diseases in hypertension and retinal angiogenesis.Formula:C23H18F4N4O2Purity:98.82% - 99.347%Color and Shape:SolidMolecular weight:458.41Ref: TM-T62858
1mg123.00€5mg295.00€1mL*10mM (DMSO)299.00€10mg490.00€25mg792.00€50mg1,071.00€100mg1,468.00€200mg1,972.00€SB 206553 hydrochloride
CAS:SB 206553 hydrochloride is a 5-HT2C inverse agonist and a 5-HT2C/5-HT2B receptor antagonist with anxiolytic activity, useful for studying neurological disordersFormula:C17H17ClN4OPurity:99.56%Color and Shape:SolidMolecular weight:328.8Photoregulin1
CAS:Photoregulin1 modulates Nr2e3, slows photoreceptor degeneration in RhoP23H, Pde6brd1 mouse RP models.Formula:C21H23N3O2SColor and Shape:SolidMolecular weight:381.49Savoxepin mesylate
CAS:Savoxepin mesylate, a tetracyclic cyano-dibenzoxepino-azepine derivative, has potent antidopaminergic activity.Formula:C26H30N2O4SPurity:98%Color and Shape:SolidMolecular weight:466.59LEQ-506
CAS:LEQ506, an oral Smoothened antagonist, may inhibit cancer growth by blocking the Hedgehog signaling pathway.Formula:C27H29N5OColor and Shape:SolidMolecular weight:439.55PF-4522654
CAS:PF-4522654 is a potent and selective 5-HT2C receptor agonist.Formula:C16H18F2N4Color and Shape:SolidMolecular weight:304.34NVS-CRF38
CAS:NVS-CRF38 is an antagonist of corticotropin-releasing factor receptor 1 (CRF1).Formula:C19H21N5O2Purity:98%Color and Shape:SolidMolecular weight:351.4PNU-142633
CAS:PNU-142633: anti-migraine, selective 5-HT1D agonist, Ki=6 nM; >18,000 nM for 5-HT1B.Formula:C24H30N4O3Purity:98%Color and Shape:SolidMolecular weight:422.52Medroxalol hydrochloride
CAS:Medroxalol hydrochloride is an antihypertensive agent that possesses both alpha and beta-adrenergic antagonistic properties.Formula:C20H25ClN2O5Color and Shape:SolidMolecular weight:408.88Carboprost
CAS:Carboprost (15(S)-15-Methyl Prostaglandin F2α) is a synthetic prostaglandin analogue of PGF2α which has the effect of oxytocic.Formula:C21H36O5Purity:98.18%Color and Shape:White Or Almost White PowderMolecular weight:368.51Ref: TM-T22285
1mg43.00€5mg110.00€1mL*10mM (DMSO)122.00€10mg166.00€25mg290.00€50mg425.00€100mg577.00€200mg778.00€Zelandopam free base
CAS:Zelandopam: dopamine D1 agonist, boosts pancreatic secretion, renal vasodilator, counters renal dysfunction.Formula:C15H15NO4Color and Shape:SolidMolecular weight:273.28Isamoltane
CAS:Isamoltane is a serotonin 5-HT1 Receptor AntagonistFormula:C16H23ClN2O2Color and Shape:SolidMolecular weight:310.82Thioperamide
CAS:histamine H3 and H4 antagonist/inverse agonistFormula:C15H24N4SPurity:98%Color and Shape:White SolidMolecular weight:292.44Ro 22-9194
CAS:Ro 22-9194, a class I antiarrhythmic, reduces upstroke velocity and shortens action potential in guinea-pig hearts at ≥10 μM.Formula:C19H27Cl2N3OPurity:98%Color and Shape:SolidMolecular weight:384.35S 32212 hydrochloride
CAS:S 32212 hydrochloride is a high-affinity inverse agonist at the 5-HT2C receptor and an antagonist at the α2-adrenergic receptor, which is antidepressant .Formula:C25H29ClN4O2Purity:97.11% - 99.57%Color and Shape:SolidMolecular weight:452.98Ro 63-0563
CAS:Ro 63-0563 is a potent, 5-HT6 receptors selective antagonist.Formula:C13H17N5O2SPurity:98%Color and Shape:SolidMolecular weight:307.37A2A receptor antagonist 3
CAS:A2A receptor antagonist 3 (Example 92) is an adenosine A2a receptor antagonist (Ki: 0.4 nM). receptor (Ki: 1467 nM).Formula:C26H26N6O2Color and Shape:SolidMolecular weight:454.52Lexipafant
CAS:Lexipafant is a platelet-activating factor (PAF) receptor antagonist.Formula:C23H30N4O4SColor and Shape:SolidMolecular weight:458.57Todralazine
CAS:Todralazine is an anti-hypertensive agent and acts as a β2AR blocker. It also has an antioxidant and free radical scavenging activity.Formula:C11H12N4O2Purity:98%Color and Shape:SolidMolecular weight:232.24Lu AA41063
CAS:Lu AA41063 is a potent and selective antagonist of the hA2A receptor.Formula:C16H17F2N3O2SColor and Shape:SolidMolecular weight:353.39SKF-83566 hydrobromide
CAS:D1-like dopamine receptor antagonistFormula:C17H19BrClNOPurity:98%Color and Shape:SolidMolecular weight:368.7A1AR antagonist 6
CAS:A1AR antagonist 6 (compound 15) is a potent and selective antagonist of A1 adenosine receptor(A1AR) with a pKi of 7.13 and a pIC 50 of 6.38[1].Formula:C17H15N3O2Color and Shape:SolidMolecular weight:293.32SB 235375
CAS:SB 235375 is a potent and selective antagonist of neurokinin-3 receptor with a low central nervous system-penetrant.Formula:C27H24N2O4Purity:98%Color and Shape:SolidMolecular weight:440.49N-Salicyloyltryptamine
CAS:N-Salicyloyltryptamine (STP): a tryptamine with anticonvulsant, anti-inflammatory, analgesic effects; inhibits Na+, Ca2+, K+ channels (IC50 34.6 μM).Formula:C17H16N2O2Color and Shape:SolidMolecular weight:280.32MS 245 oxalate
CAS:MS 245 oxalate is a 5-HT6 antagonist.Formula:C21H24N2O7SPurity:98%Color and Shape:SolidMolecular weight:448.49
