GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,028 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(61 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6012 products of "GPCR/G-Protein"
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Blonanserin HCl
CAS:Blonanserin is an antagonist of dopamine-D2 and serotonin-S2.Formula:C23H32Cl2FN3Purity:98%Color and Shape:SolidMolecular weight:440.42S-1-Propenyl-L-cysteine
CAS:S-1-Propenyl-L-cysteine, a stereoisomer of S-allyl-l-cysteine, exhibits immunomodulatory effects and has been shown to decrease blood pressure in hypertensiveFormula:C6H11NO2SPurity:98%Color and Shape:SolidMolecular weight:161.22RXFP3 agonist 1
CAS:RXFP3 agonist 1 is a nonpeptide RXFP3 agonist ( EC 50 =6937 nM) [1].Formula:C18H18ClN5Color and Shape:SolidMolecular weight:339.82SKF-82958
CAS:SKF 82958 is a D1/D5 receptor full agonist.Formula:C19H20ClNO2Purity:98%Color and Shape:SolidMolecular weight:329.82Dopamine D2 receptor antagonist-1
CAS:Dopamine D2 Receptor Antagonist-1 functions as a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R), demonstrating sub-millimolar affinity.Formula:C14H17N3SPurity:99.86%Color and Shape:SolidMolecular weight:259.37Ref: TM-T11077
1mg57.00€5mg120.00€1mL*10mM (DMSO)133.00€10mg178.00€25mg334.00€50mg492.00€100mg692.00€UR-PI376
CAS:UR-PI376 is a selective histamine H4 receptor agonist with low H1/H2 activity and moderate H3 affinity.Formula:C17H22N6SColor and Shape:SolidMolecular weight:342.46VSN-16
CAS:VSN-16, a cannabinoid receptor agonist, is used potentially for the treatment of spasticity in multiple sclerosis.Formula:C18H26N2O3Color and Shape:SolidMolecular weight:318.41BKM-570
CAS:BKM-570, a bradykinin antagonist, causes impressive growth inhibition of lung and prostate tumors.Formula:C34H34Cl2F5N3O3Purity:98%Color and Shape:SolidMolecular weight:698.55BMS-457
CAS:BMS-457 is a potent, CCR1-selective antagonist.Formula:C24H35ClN2O4Purity:98%Color and Shape:SolidMolecular weight:451GSK-215083
CAS:GSK-215083: a PET quinoline-based 5-HT6 antagonist radioligand, binds 5HT6 in striatum and 5HT2A in frontal cortex.Formula:C20H20FN3O2SColor and Shape:SolidMolecular weight:385.46Zimelidine dihydrochloride
CAS:5-HT re-uptake inhibitorFormula:C16H18BrClN2Purity:98%Color and Shape:SolidMolecular weight:353.69(R)-Carvedilol
CAS:(R)-Carvedilol is a non-selective blocker of β/α-1. (R)-Carvedilol exerts protection against the vascular or cardiac toxicity of Doxorubicin (DOX).Formula:C24H26N2O4Purity:98%Color and Shape:SolidMolecular weight:406.47Tropodifene
CAS:Tropodifene is an inhibitor of the α-Adrenergic receptor.Formula:C25H29NO4Purity:98%Color and Shape:SolidMolecular weight:407.52-Methylthio-AMP diTEA
CAS:2-MeSAMP diTEA blocks P2Y12 receptor, inhibits ADP platelet clumping.Formula:C23H46N7O7PSColor and Shape:SolidMolecular weight:595.69Falintolol, (Z)-
CAS:Falintolol, (Z)-, is a novel β-adrenergic antagonist compound distinguished by the inclusion of an oxime moiety.Formula:C12H24N2O2Purity:98%Color and Shape:SolidMolecular weight:228.33Mezilamine
CAS:Mezilamine is an antagonist of dopamine. It also blocks presynaptic but stimulating postsynaptic alpha-adrenoceptors.Formula:C11H18ClN5SPurity:98%Color and Shape:SolidMolecular weight:287.81TC-G1003
CAS:TC-G1003 is an effective agonist of the somatostatin sst2 receptor.Formula:C26H25ClN2O2Purity:98%Color and Shape:SolidMolecular weight:432.94Cinalukast
CAS:CysLT1 leukotriene receptor antagonistFormula:C23H28N2O3SPurity:98%Color and Shape:SolidMolecular weight:412.55Way 100289
CAS:Way 100289 is a selective 5-HT3 receptor antagonist.Formula:C20H27N3O3Color and Shape:SolidMolecular weight:357.45CM764
CAS:CM764 is a potent and selective antagonist of sigma-2 receptors, a novel derivative of SN79.Formula:C23H27FN4O3Color and Shape:SolidMolecular weight:426.48BGC 20-761
CAS:BGC20-761: selective 5-HT6/Dopamine antagonist; enhances memory, potential antipsychotic. K i - 5-HT6: 20 nM, 5-HT2A: 69 nM, D2: 140 nM.Formula:C19H22N2OColor and Shape:SolidMolecular weight:294.39WB 4101 hydrochloride
CAS:α1A-adrenergic antagonistFormula:C19H24ClNO5Purity:98%Color and Shape:SolidMolecular weight:381.85Amitriptylinoxide
CAS:Amitriptylinoxide is an antidepressant.Formula:C20H23NOPurity:98%Color and Shape:SolidMolecular weight:293.4PF-3246799
CAS:PF-3246799 is an effective and selective agonist of the 5-HT2C receptor.Formula:C15H17N3Purity:98%Color and Shape:SolidMolecular weight:239.32Impromidine
CAS:Impromidine is a highly potent and specific agonist of the histamine H2 receptor.Formula:C14H23N7SPurity:98%Color and Shape:SolidMolecular weight:321.44L 665871
CAS:L 665871 is used as a beta-agonist. It works as a potential swine growth promoter.Formula:C11H19N3OPurity:98%Color and Shape:SolidMolecular weight:209.29Azatadine
CAS:Azatadine is histamine and cholinergic inhibitor (IC50: 6.5 nM and 10 nM, respectively).Formula:C20H22N2Purity:98%Color and Shape:SolidMolecular weight:290.4SN 003
CAS:SN 003 is a CRF1 antagonist.Formula:C19H25N5O2Purity:98%Color and Shape:SolidMolecular weight:355.43EPAC 5376753
CAS:EPAC 5376753 is an allosteric inhibitor of EPAC1 with an IC50 of 4 µM in Swiss 3T3 cells.Formula:C15H8Cl2N2O3SPurity:97.48%Color and Shape:SolidMolecular weight:367.21Amibegron hydrochloride
CAS:Amibegron hydrochloride is a selective β3-adrenoceptor agonist (EC50: 3.5 nM for β-adrenoceptor in rat colon). It has anxiolytic and antidepressant activity.Formula:C22H27Cl2NO4Color and Shape:SolidMolecular weight:440.36Sograzepide
CAS:Sograzepide (Netazepide) is a gastrin/CCK-B antagonist, inhibits gastrin/CCK-A activity, and can induce regression of type 1 gastric neuroendocrine tumorsFormula:C28H30N6O3Purity:98%Color and Shape:SolidMolecular weight:498.58Dopamine D4 receptor antagonist-1
CAS:Dopamine D4 receptor antagonist-1 can be used in schizophrenia study.Formula:C18H19ClN4Color and Shape:SolidMolecular weight:326.82Org37684
CAS:5-HT2 receptors agonistFormula:C14H20ClNO2Purity:98%Color and Shape:SolidMolecular weight:269.77OX2R-IN-1
CAS:OX2R-IN-1: OX2R antagonist, low cytotoxicity, blood-brain barrier permeable, short half-life.Formula:C20H28ClN3O5SColor and Shape:SolidMolecular weight:457.97Prasugrel (Maleic acid)
CAS:Prasugrel Maleic acid: oral P2Y12 antagonist, thienopyridine prodrug, inhibits ADP-induced platelet aggregation.Formula:C24H24FNO7SPurity:98%Color and Shape:SolidMolecular weight:489.51GSK 894281
CAS:GSK 894281 is a ghrelin receptor agonist. It may produces myocardial degeneration/necrosis in rats.Formula:C24H28FN3O4SPurity:98%Color and Shape:SolidMolecular weight:473.56CB1R Allosteric modulator 4
CAS:Modulates CB1R positively; inhibits cAMP production; strong β-arrestin-2 recruitment.Formula:C20H17N3O2SColor and Shape:SolidMolecular weight:363.43CGS-12066 maleate salt
CAS:CGS-12066 maleate salt is an agonist of 5-HT1B serotonin receptor.Formula:C21H21F3N4O4Color and Shape:SolidMolecular weight:450.41(4-Acetamidocyclohexyl) nitrate
CAS:(4-Acetamidocyclohexyl) nitrate (BM121307) is an activator of guanylate cyclase.Formula:C8H14N2O4Purity:98%Color and Shape:SolidMolecular weight:202.21A412997
CAS:A412997 is a selective agonist of dopamine D4 receptor.Formula:C19H23N3OPurity:98%Color and Shape:SolidMolecular weight:309.41GP531
CAS:GP531, a second-gen adenosine regulator, is inactive at rest but boosts adenosine in ischemia.Formula:C16H21N5O4Color and Shape:SolidMolecular weight:347.37LG 82-4-01
CAS:LG 82-4-01 is an inhibitor of thromboxane (TX) synthetase.Formula:C10H10Cl2N2O3SPurity:98%Color and Shape:SolidMolecular weight:309.17EMD 386088 hydrochloride
CAS:EMD 386088 hydrochloride is a 5-HT6 receptor agonist.Formula:C14H16Cl2N2Purity:98%Color and Shape:SolidMolecular weight:283.2Guanadrel
CAS:Guanadrel is an antihypertensive agent.Formula:C10H19N3O2Purity:98%Color and Shape:SolidMolecular weight:213.288-M-PDOT
CAS:8-M-PDOT (AH-002) is an MT2 receptor agonist that inhibits MT1.8-M-PDOT has anxiolytic activity and may be used in the study of neuropathic pain.Formula:C14H19NO2Purity:99.54% - 99.54%Color and Shape:SolidMolecular weight:233.31SKI 5C
CAS:SKI 5C is a selective inhibitor of Sphingosine Kinase 1.Formula:C26H45NO4Purity:98%Color and Shape:SolidMolecular weight:435.64LY 290324
CAS:LY 290324 is an orally active, potent and selective antagonist of cysteinyl leukotriene (LTD4) receptor.Formula:C29H24Cl2N6Purity:98%Color and Shape:SolidMolecular weight:527.45PD-159020
CAS:PD-159020 is a non-selective antagonist of ETA/ETB(hETA and hETB with IC50s of 30 and 50 nM , respectively).Formula:C32H25NO8Purity:98%Color and Shape:SolidMolecular weight:551.54N-0861 racemate
CAS:N-0861 racemate is the racemate of N-0861.Formula:C13H17N5Purity:98%Color and Shape:SolidMolecular weight:243.31PD 120697
CAS:PD 120697 is a dopamine antagonist with central dopamine agonist properties.Formula:C11H15N3SPurity:98%Color and Shape:SolidMolecular weight:221.32
