GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,028 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(61 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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Fosnetupitant
CAS:Fosnetupitant is a methylene phosphate prodrug of Netupitant. It has a pKi of 9.5 for the human NK1 receptor.Formula:C31H35F6N4O5PPurity:98%Color and Shape:SolidMolecular weight:688.6Albuterol adipate
CAS:Albuterol adipate, a β2-AR agonist salt, treats asthma/COPD, with high selectivity for pulmonary over cardiac receptors.Formula:C32H52N2O10Color and Shape:SolidMolecular weight:624.77Levomepromazine Maleate
CAS:Levomepromazine Maleate: TCA and SNRI with antihistamine, antiadrenergic, and anticholinergic properties.Formula:C23H28N2O5SColor and Shape:SolidMolecular weight:444.546ZD7114 free base
CAS:ZD7114 (ICI-D7114) selectively activates brown fat, boosts thermogenesis, and aids in obesity and metabolic disorders.Formula:C22H30N2O6Color and Shape:SolidMolecular weight:418.48p-MPPF dihydrochloride
CAS:p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.Formula:C25H29Cl2FN4O2Purity:99.55%Color and Shape:SolidMolecular weight:507.43Ricinelaidic Acid
CAS:Ricinelaidic acid blocks LTB4 receptors; hampers human neutrophil responses; reduces rat bronchoconstriction by 46% at 1 mg/kg i.v.Formula:C18H34O3Color and Shape:SolidMolecular weight:298.46Darbufelone
CAS:Darbufelone (CI-1004) is a non-competitive dual inhibitor of PGF2α and LTB4.Formula:C18H24N2O2SPurity:99.72%Color and Shape:SolidMolecular weight:332.46Ref: TM-T10960
1mg42.00€5mg82.00€1mL*10mM (DMSO)104.00€10mg124.00€25mg264.00€50mg386.00€100mg532.00€500mg1,063.00€VRX 03011 Potassium salt
CAS:VRX 03011, a 5-HT4 partial agonist, is used potentially for the treatment of Alzheimer's disease.Formula:C19H27KN3O3SPurity:98%Color and Shape:SolidMolecular weight:416.6Quinpirole
CAS:Quinpirole is a dopamine D2/D3 receptor agonist.Formula:C13H21N3Color and Shape:SolidMolecular weight:219.33Thiothixene hydrochloride
CAS:Thiothixene hydrochloride is an antipsychotic agent that can be used in the study of schizophrenia and bipolar mania.Formula:C23H30ClN3O2S2Color and Shape:SolidMolecular weight:480.08Isoetharine hydrochloride
CAS:Isoetharine HCl, a selective, short-acting oral β-agonist, is used as a bronchodilator for inhalation therapy.Formula:C13H22ClNO3Color and Shape:SolidMolecular weight:275.77Trimethaphan camsylate
CAS:Trimethaphan camsylate is a nicotinic antagonist that has been used as a ganglionic blocker in hypertension.Formula:C32H40N2O5S2Color and Shape:SolidMolecular weight:596.801Ro 23-3423
CAS:Ro 23-3423 is a specific inhibitor of thromboxane synthetase.Formula:C23H22N4O2Color and Shape:SolidMolecular weight:386.45MAT2A-IN-2
CAS:MAT2A-IN-2 is a potent inhibitor of MAT2A. MAT2A-IN-2 has potential for cancer disease research.Formula:C23H17F3N6O2Color and Shape:SolidMolecular weight:466.42Proxodolol hydrochloride
CAS:Proxodolol, a β-adrenergic receptor antagonist, is used potentially for the treatment of glaucoma, hypertension and angina.Formula:C17H26ClN3O4Color and Shape:SolidMolecular weight:371.86Opaganib HCl
CAS:ABC294640 (Opaganib) is an SK2 inhibitor with potential anti-cancer effects; it blocks S1P production to induce apoptosis.Formula:C23H26Cl2N2OColor and Shape:SolidMolecular weight:417.37Esreboxetine
CAS:Esreboxetine( PNU-165442, (S,S) -reboxetine) is a selective inhibitor of norepinephrine reuptake.Formula:C19H23NO3Color and Shape:SolidMolecular weight:313.39PGN-9856
CAS:PGN-9856 is an EP2 receptor ligand and EP2 receptor agonist with anti-inflammatory and intraocular pressure-lowering properties, useful for glaucoma research.Formula:C21H15F2NO4Purity:99.27%Color and Shape:SolidMolecular weight:383.35Melatonin receptor agonist 1
CAS:Melatonin receptor agonist 1 (compound 20c) is a potent agonist of melatonin receptor (MT) with Ki values of 108 nM for MT2 and 1140 nM for MT 1 [1].Formula:C15H19N3O2Color and Shape:SolidMolecular weight:273.33Bitolterol
CAS:Bitolterol is a new beta 2-adrenergic agonist and classified as a pro-drug.Formula:C28H31NO5Color and Shape:SolidMolecular weight:461.55Tacitin
CAS:Tacitin (Benzoctamine Hydrochloride) shows sedative and anti-anxiety properties. Tacitin blocks the central postsynaptic serotonin receptors.Formula:C18H20ClNPurity:98%Color and Shape:SolidMolecular weight:285.81Sch 44643
CAS:Sch 44643 is an antagonist of platelet activating factor with oral activity.Formula:C25H22ClN3O2Color and Shape:SolidMolecular weight:431.91LUF6000
CAS:LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR).Formula:C22H20Cl2N4Color and Shape:SolidMolecular weight:411.33WIN 62,577
CAS:WIN 62,577 is a allosteric antagonist of mAChR.Formula:C29H31N3OPurity:98%Color and Shape:SolidMolecular weight:437.58Iferanserin HCl
CAS:Iferanserin HCl is a selective serotonin receptor antagonist.Formula:C23H29ClN2OColor and Shape:SolidMolecular weight:384.95GYKI-13380
CAS:GYKI-13380, also known as LS-79445, is a small molecule with potent bioactivity. Detail information has not been published yet.Formula:C16H22N2O3Color and Shape:SolidMolecular weight:290.36VER-3323
CAS:VER-3323 is a selective agonist for the 5-HT2B and 5-HT2C serotonin receptor with potent anorectic effects in animal studies.Formula:C11H15BrN2Purity:98%Color and Shape:SolidMolecular weight:255.15YQA14
CAS:YQA14 is a selective, high-affinity dopamine D3 receptor antagonist that inhibits cocaine self-administration in rats and mice, opioid addiction research.Formula:C23H27ClN4O3Purity:99.52%Color and Shape:SolidMolecular weight:442.94U 101958
CAS:U 101958 is a putative antipsychotic agent It is also a highly selective dopamine D4 receptor antagonist.Formula:C20H27N3OColor and Shape:SolidMolecular weight:325.45Fonazine hydrochloride
CAS:Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.Formula:C19H26ClN3O2S2Color and Shape:SolidMolecular weight:428.01AChE-IN-14
CAS:AChE-IN-14 inhibits eeAChE, hAChE, eqBuChE (IC50: 0.46-0.48 μM) and binds to H3R (Ki: 159.8 nM), useful for Alzheimer's research.Formula:C28H35NO3Color and Shape:SolidMolecular weight:433.58Sch 40120
CAS:Sch 40120 is an inhibitor of 5-lipoxygenase.Formula:C18H15ClN2OPurity:98%Color and Shape:SolidMolecular weight:310.78SB357134
CAS:SB357134 is a potent, selective and orally active antagonist of 5-HT6 receptor and shows nootropic effects in animal studies.Formula:C17H18Br2FN3O3SPurity:98%Color and Shape:SolidMolecular weight:523.21Toreforant
CAS:Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).Formula:C23H32N6Purity:98%Color and Shape:SolidMolecular weight:392.54TISCH
CAS:TISCH is a potent and selective iodinated ligand for CNS D1 dopamine receptor.Formula:C17H17ClINOColor and Shape:SolidMolecular weight:413.68Fonazine mesylate
CAS:Fonazine mesylate is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.Formula:C20H29N3O5S3Color and Shape:SolidMolecular weight:487.65Flerobuterol HCl
CAS:"Flerobuterol, a β adrenergic agonist, may treat depression by boosting serotonin synthesis and Trp in the brain."Formula:C12H19ClFNOPurity:98%Color and Shape:SolidMolecular weight:247.74MRS 1334
CAS:antagonist for the human adenosine A3 receptorFormula:C31H26N2O6Purity:98%Color and Shape:SolidMolecular weight:522.55A-971432
CAS:A-971432: selective S1P5 agonist, IC50 = 0.006 µM. Enhances blood-brain barrier, reduces Huntington’s symptoms in mice at 0.1 mg/kg.Formula:C18H17Cl2NO3Color and Shape:SolidMolecular weight:366.24Brl 22321
CAS:Brl 22321 is a mast cell stabilizer.Formula:C12H9N3O2Color and Shape:SolidMolecular weight:227.22PF-06256142
CAS:PF-06256142 is a potent and selective orthosteric D1 receptor agonist(D1 EC50=30 nM ).Formula:C21H16N4O2Purity:98%Color and Shape:SolidMolecular weight:356.38AZD-2207
CAS:AZD-2207 is a cannabinoid receptor CB1 antagonist and highly lipophilic compound for the treatment of type 2 diabetes mellitus and obesity.Formula:C25H25Cl2F3N4O4SColor and Shape:SolidMolecular weight:605.46Cannabicitran
CAS:Cannabicitran is a cannabinoid that can decrease rabbits intraocular pressure [1] [2].Formula:C21H30O2Color and Shape:SolidMolecular weight:314.46AZD5213
CAS:AZD5213: selective human H3 receptor antagonist, pKi 9.3, for sleep/cognition research.Formula:C19H25N3O2Color and Shape:SolidMolecular weight:327.42(R,R)-Reboxetine mesylate
CAS:(R,R)-Reboxetine mesylate: Antidepressant, high bioavailability, (R,R) enantiomer, selective for noradrenaline, low toxicity.Formula:C20H27NO6SColor and Shape:SolidMolecular weight:409.5TCS-OX2-29 HCl
CAS:TCS-OX2-29 is a selective orexin-2 receptor antagonist (IC50 = 40 nM), which plays an important role in pain modulation.Formula:C23H32ClN3O3Purity:98%Color and Shape:SolidMolecular weight:433.97A331440
CAS:A331440 is an modulator of L-histidine and histamine H3 receptor.Formula:C22H27N3OColor and Shape:SolidMolecular weight:349.47BL 6341A
CAS:BL 6341A is related to Tumor data and H2-antagonists or anti-histaminsFormula:C9H14N8OS3Color and Shape:SolidMolecular weight:346.46Cyclazosin HCl
CAS:Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.Formula:C23H28ClN5O4Purity:99.10%Color and Shape:SolidMolecular weight:473.95Carbuterol hydrochloride
CAS:Carbuterol hydrochloride is a short-acting β2 adrenoreceptor agonist.Formula:C13H22ClN3O3Color and Shape:SolidMolecular weight:303.79
