GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,022 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5984 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
VK-II-86
CAS:VK-II-86 is a non-β-blocking carvedilol analog. It prevents ouabain-Induced cardiotoxicityFormula:C25H28N2O4Purity:98%Color and Shape:SolidMolecular weight:420.5Argiprestocin
CAS:Argiprestocin: antidiuretic, regulates osmolality, neurohypophysial hormone, vasoconstrictor.Formula:C43H67N15O12S2Purity:99.34%Color and Shape:SolidMolecular weight:1050.22VL-0395
CAS:VL-0395 is an antagonist of CCK1 receptor.Formula:C25H21N3O4Purity:98%Color and Shape:SolidMolecular weight:427.45Mabuterol, (S)-
CAS:Mabuterol, a β2 adrenoreceptor agonist, lowers rat blood pressure and boosts guinea pig heart rate/force, not affecting other receptors.Formula:C13H18ClF3N2OColor and Shape:SolidMolecular weight:310.74Colterol HCl
CAS:Colterol HCl, a β2-adrenoceptor agonist salt, is used for bronchospasm in asthma and COPD.Formula:C12H20ClNO3Color and Shape:SolidMolecular weight:261.75Dacemazine
CAS:Dacemazine is used to treat depression.Formula:C16H16N2OSColor and Shape:SolidMolecular weight:284.38Ambenoxan hydrochloride
CAS:Ambenoxan hydrochloride is a centrally acting skeletal muscle relaxant.Formula:C14H22ClNO4Color and Shape:SolidMolecular weight:303.78Ambucetamide
CAS:Ambucetamide is an antispasmodic, it may inhibit or diminish the spontaneous rhythmical activity of the human myometrium.Formula:C17H28N2O2Color and Shape:SolidMolecular weight:292.42BAY-386
CAS:BAY-386 is a PAR1 receptor inhibitor which suppresses activation of thrombin and platelet activity.Formula:C22H25F3N4O5SColor and Shape:SolidMolecular weight:514.52F-15599 tosylate
CAS:F-15599 tosylate is a selective 5-HT(1A) agonist.Formula:C26H29ClF2N4O4SColor and Shape:SolidMolecular weight:567.05VUF14738
CAS:VUF14738 is a robust and fatigue-resistant photoswitchable GPCR antagonist.Formula:C25H32N4O2Color and Shape:SolidMolecular weight:420.55Albuterol adipate
CAS:Albuterol adipate, a β2-AR agonist salt, treats asthma/COPD, with high selectivity for pulmonary over cardiac receptors.Formula:C32H52N2O10Color and Shape:SolidMolecular weight:624.77Levomepromazine Maleate
CAS:Levomepromazine Maleate: TCA and SNRI with antihistamine, antiadrenergic, and anticholinergic properties.Formula:C23H28N2O5SColor and Shape:SolidMolecular weight:444.546ZD7114 free base
CAS:ZD7114 (ICI-D7114) selectively activates brown fat, boosts thermogenesis, and aids in obesity and metabolic disorders.Formula:C22H30N2O6Color and Shape:SolidMolecular weight:418.48Aceprometazine
CAS:Aceprometazine (1664CB) is an antipsychotic which is orally active. Aceprometazine can be used in psychiatric disorders research, for example, depression [1].Formula:C19H22N2OSColor and Shape:SolidMolecular weight:326.46Ricinelaidic Acid
CAS:Ricinelaidic acid blocks LTB4 receptors; hampers human neutrophil responses; reduces rat bronchoconstriction by 46% at 1 mg/kg i.v.Formula:C18H34O3Color and Shape:SolidMolecular weight:298.46Darbufelone
CAS:Darbufelone (CI-1004) is a non-competitive dual inhibitor of PGF2α and LTB4.Formula:C18H24N2O2SPurity:99.72%Color and Shape:SolidMolecular weight:332.46Ref: TM-T10960
1mg42.00€5mg82.00€1mL*10mM (DMSO)104.00€10mg124.00€25mg264.00€50mg386.00€100mg532.00€500mg1,063.00€GBR-12935 maleate
CAS:GBR-12935: dopamine reuptake inhibitor, used in research for Parkinson's and brain's dopamine pathways.Formula:C32H38N2O5Color and Shape:SolidMolecular weight:530.665VRX 03011 Potassium salt
CAS:VRX 03011, a 5-HT4 partial agonist, is used potentially for the treatment of Alzheimer's disease.Formula:C19H27KN3O3SPurity:98%Color and Shape:SolidMolecular weight:416.6Quinpirole
CAS:Quinpirole is a dopamine D2/D3 receptor agonist.Formula:C13H21N3Color and Shape:SolidMolecular weight:219.33Thiothixene hydrochloride
CAS:Thiothixene hydrochloride is an antipsychotic agent that can be used in the study of schizophrenia and bipolar mania.Formula:C23H30ClN3O2S2Color and Shape:SolidMolecular weight:480.08Isoetharine hydrochloride
CAS:Isoetharine HCl, a selective, short-acting oral β-agonist, is used as a bronchodilator for inhalation therapy.Formula:C13H22ClNO3Color and Shape:SolidMolecular weight:275.77Trimethaphan camsylate
CAS:Trimethaphan camsylate is a nicotinic antagonist that has been used as a ganglionic blocker in hypertension.Formula:C32H40N2O5S2Color and Shape:SolidMolecular weight:596.801Ro 23-3423
CAS:Ro 23-3423 is a specific inhibitor of thromboxane synthetase.Formula:C23H22N4O2Color and Shape:SolidMolecular weight:386.45Proxodolol hydrochloride
CAS:Proxodolol, a β-adrenergic receptor antagonist, is used potentially for the treatment of glaucoma, hypertension and angina.Formula:C17H26ClN3O4Color and Shape:SolidMolecular weight:371.86Opaganib HCl
CAS:ABC294640 (Opaganib) is an SK2 inhibitor with potential anti-cancer effects; it blocks S1P production to induce apoptosis.Formula:C23H26Cl2N2OColor and Shape:SolidMolecular weight:417.37Dicentrine HCl
CAS:Dicentrine HCl is the salt form of Dicentrine, an alpha 1-adrenoceptor antagonist effective against human hyperplastic prostates.Formula:C20H22ClNO4Color and Shape:SolidMolecular weight:375.85DH-97
CAS:DH-97 is a potent MT2 melatonin receptor antagonist (pKi value = 8.03).Formula:C22H26N2OColor and Shape:SolidMolecular weight:334.45Esreboxetine
CAS:Esreboxetine( PNU-165442, (S,S) -reboxetine) is a selective inhibitor of norepinephrine reuptake.Formula:C19H23NO3Color and Shape:SolidMolecular weight:313.39Bitolterol
CAS:Bitolterol is a new beta 2-adrenergic agonist and classified as a pro-drug.Formula:C28H31NO5Color and Shape:SolidMolecular weight:461.555-HT4 antagonist 1
CAS:5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).Formula:C23H36N4O5SPurity:99.75%Color and Shape:SolidMolecular weight:480.62Glucagon Receptor Antagonist I
CAS:Glucagon antagonist I blocks the GCGR (IC50=181 nM), stops glucagon-induced glycogenolysis, and lowers glucose in glucagon-treated humanized mice.Formula:C20H30N2OSColor and Shape:SolidMolecular weight:346.53Sch 44643
CAS:Sch 44643 is an antagonist of platelet activating factor with oral activity.Formula:C25H22ClN3O2Color and Shape:SolidMolecular weight:431.91Iferanserin HCl
CAS:Iferanserin HCl is a selective serotonin receptor antagonist.Formula:C23H29ClN2OColor and Shape:SolidMolecular weight:384.95GYKI-13380
CAS:GYKI-13380, also known as LS-79445, is a small molecule with potent bioactivity. Detail information has not been published yet.Formula:C16H22N2O3Color and Shape:SolidMolecular weight:290.36VER-3323
CAS:VER-3323 is a selective agonist for the 5-HT2B and 5-HT2C serotonin receptor with potent anorectic effects in animal studies.Formula:C11H15BrN2Purity:98%Color and Shape:SolidMolecular weight:255.15Reproterol hydrochloride
CAS:Reproterol hydrochloride, a β2 adrenoreceptor agonist, is used to treat asthma and chronic obstructive pulmonary disease (COPD).Formula:C18H24ClN5O5Purity:98%Color and Shape:SolidMolecular weight:425.87U 101958
CAS:U 101958 is a putative antipsychotic agent It is also a highly selective dopamine D4 receptor antagonist.Formula:C20H27N3OColor and Shape:SolidMolecular weight:325.45Fonazine hydrochloride
CAS:Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.Formula:C19H26ClN3O2S2Color and Shape:SolidMolecular weight:428.01Sch 40120
CAS:Sch 40120 is an inhibitor of 5-lipoxygenase.Formula:C18H15ClN2OPurity:98%Color and Shape:SolidMolecular weight:310.78MRS2690
CAS:MRS2690 is a potent P2Y14 receptor agonist (EC50 = 49 nM) that displays 7-fold higher potency than UDP-glucose.Formula:C15H24N2O16P2SColor and Shape:SolidMolecular weight:582.37Toreforant
CAS:Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).Formula:C23H32N6Purity:98%Color and Shape:SolidMolecular weight:392.54TISCH
CAS:TISCH is a potent and selective iodinated ligand for CNS D1 dopamine receptor.Formula:C17H17ClINOColor and Shape:SolidMolecular weight:413.68Fonazine mesylate
CAS:Fonazine mesylate is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.Formula:C20H29N3O5S3Color and Shape:SolidMolecular weight:487.65Flerobuterol HCl
CAS:"Flerobuterol, a β adrenergic agonist, may treat depression by boosting serotonin synthesis and Trp in the brain."Formula:C12H19ClFNOPurity:98%Color and Shape:SolidMolecular weight:247.74Zimelidine
CAS:Zimelidine, a withdrawn antidepressant, posed Guillain-Barre risk.Formula:C16H17BrN2Purity:98%Color and Shape:SolidMolecular weight:317.22RP-72540
CAS:RP-72540: CCKB receptor blocker, 200x more selective for CCKA, binds to stomach gastrin, limits [3H]pCCK-8 in mouse brain, <0.01% reaches forebrain.Formula:C28H30N4O6Purity:98%Color and Shape:SolidMolecular weight:518.56A-971432
CAS:A-971432: selective S1P5 agonist, IC50 = 0.006 µM. Enhances blood-brain barrier, reduces Huntington’s symptoms in mice at 0.1 mg/kg.Formula:C18H17Cl2NO3Color and Shape:SolidMolecular weight:366.24Brl 22321
CAS:Brl 22321 is a mast cell stabilizer.Formula:C12H9N3O2Color and Shape:SolidMolecular weight:227.22(R)-Bambuterol
CAS:Bambuterol is a β2-agonist prodrug for asthma and COPD, taken daily, with a good safety profile and reduces plasma LDL-C and cholesterol.Formula:C18H29N3O5Color and Shape:SolidMolecular weight:367.44
