GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,998 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5959 products of "GPCR/G-Protein"
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Bradykinin (1-5)
CAS:Bradykinin (1-5), a stable metabolite of BK produced by ACE, serves as a marker for in vivo BK generation.Formula:C27H40N8O6Color and Shape:SolidMolecular weight:572.66SB-674042
CAS:SB-674042 is a nonpeptide dual antagonist of the appetite peptides OX1 and OX2 receptors.SB-674042 is used in the treatment of depression.Formula:C24H21FN4O2SPurity:99.87% - 99.9%Color and Shape:SolidMolecular weight:448.51Haloperidol (D4')
CAS:Haloperidol D4' is deuterium-labeled haloperidol. Haloperidol is a dopamine D2 receptor antagonist.Formula:C21H23ClFNO2Purity:98%Color and Shape:SolidMolecular weight:379.893-Hydroxy agomelatine
CAS:3-Hydroxy agomelatine (3-Hydroxyagomelatine) is a 5-HT2C receptor antagonist used in the study of neurological disorders.Formula:C15H17NO3Color and Shape:SolidMolecular weight:259.3Diacetolol D7
CAS:Diacetolol D7 is deuterium-labeled diacetone Roller. Diacetol is the main metabolite of Acetolol. Diacetololβ-adrenoceptor shielding and anti-arrhythmic agent.Formula:C16H24N2O4Purity:98%Color and Shape:SolidMolecular weight:315.42SANT 2
CAS:SANT 2 is a Hedgehog (Hh) signaling pathway antagonist with potential anti-inflammatory and anti-cancer activities.Formula:C26H26ClN3O4Purity:99.23%Color and Shape:SolidMolecular weight:479.96Taranabant racemate
CAS:Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.Formula:C27H25ClF3N3O2Purity:98%Color and Shape:SolidMolecular weight:515.95Furprofen
CAS:Furprofen, an NSAID, inhibits PGE synthesis, offers analgesic effects, and is orally taken for pain relief.Formula:C14H12O4Purity:98.62% - 99.25%Color and Shape:SolidMolecular weight:244.241-Methyl-4-imidazoleacetic Acid (hydrochloride)
CAS:MIMA, a stable histamine byproduct from N-methylhistamine oxidation, indicates systemic mastocytosis via urinary levels.Formula:C6H9ClN2O2Color and Shape:SolidMolecular weight:176.601Piribedil D8
CAS:Piribedil D8 is the deuterium labeled Piribedil, which is an agent of antiparkinsonian.Formula:C16H18N4O2Purity:98%Color and Shape:SolidMolecular weight:306.39Agomelatine (L(+)-Tartaric acid)
CAS:Agomelatine (L(+)-Tartaric acid) is an MT1/MT2 agonist and selective 5-HT2C antagonist, supporting melatonergic and serotonergic signaling studies in neuroscience.Formula:C19H23NO8Purity:99.79%Color and Shape:SolidMolecular weight:393.39Fluvoxamine
CAS:Fluvoxamine (DU-23000) is a selective, orally available 5-HT and serotonin reuptake inhibitor (SSRI) exhibiting antidepressant effects.Formula:C15H21F3N2O2Purity:99.91%Color and Shape:SolidMolecular weight:318.33Quetiapine-d8 Fumarate
CAS:Quetiapine-d8 Fumarate is a deuterated compound of Quetiapine Fumarate. Quetiapine Fumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.Formula:C25H21D8N3O6SColor and Shape:SolidMolecular weight:507.63Pramipexole dihydrochloride
CAS:Pramipexole dihydrochloride could be used to treat Parkinson disease.Formula:C10H18ClN3SPurity:98%Color and Shape:White Crystalline PowderMolecular weight:247.79Virodhamine
CAS:Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of CB2 receptor.Formula:C22H37NO2Purity:98%Color and Shape:SoildMolecular weight:347.53MK-761 TFA
MK-761 TFA is an effective, orally active β2-adrenergic receptor blocker. It exhibits antihypertensive properties and positive inotropic effects, along with vasodilatory activity.Formula:C15H20F3N3O4Color and Shape:SolidMolecular weight:363.332GPR34 receptor antagonist 3
Compound 5e, a GPR34 receptor antagonist, exhibits selective inhibition of lysophosphatidylserine-induced ERK1/2 phosphorylation in a dose-dependent manner,Color and Shape:Odour SolidBMS-986020 sodium
CAS:BMS-986020 sodium (AM152 sodium) is a high-affinity LPA1 antagonist for investigating idiopathic pulmonary fibrosis.Formula:C29H25N2NaO5Purity:99.83%Color and Shape:SolidMolecular weight:504.51Ziprasidone D8
CAS:Ziprasidone D8, deuterium-labeled, is a potent antipsychotic, antagonizing 5-HT and dopamine receptors.Formula:C21H21ClN4OSPurity:98%Color and Shape:SolidMolecular weight:420.99(R)-Praziquantel-d11
CAS:(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel.Formula:C19H24N2O2Purity:98%Color and Shape:SolidMolecular weight:323.47
