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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5960 products of "GPCR/G-Protein"

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  • Calcium-Sensing Receptor Antagonists I

    CAS:
    Calcium-Sensing Receptor Antagonists I functions as an antagonist to the parathyroid hormone receptors that sense calcium.
    Formula:C23H24N2O2
    Color and Shape:Solid
    Molecular weight:360.45

    Ref: TM-T10665

    2mg
    62.00€
    5mg
    104.00€
    1mL*10mM (DMSO)
    166.00€
  • Travoprost (Standard)

    CAS:
    Travoprost (Standard) is the standard substance of Travoprost, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Travoprost (Fluprostenol isopropyl ester) is used to treat glaucoma and ocular hypertension,is a potent and selective FP prostaglandin receptor agonist.
    Formula:C26H35F3O6
    Color and Shape:Colorless Oil
    Molecular weight:500.55

    Ref: TM-TMSM-2282

    10mg
    231.00€
  • WAY-100635

    CAS:
    WAY-100635 is a potent 5-HT 1A receptor antagonist pyramidal neuron firing frequency during conditioned reflexes; a dopamine D4 receptor agonist .
    Formula:C25H34N4O2
    Purity:98.972%
    Color and Shape:Solid
    Molecular weight:422.56

    Ref: TM-T21561

    2mg
    44.00€
    5mg
    64.00€
    10mg
    98.00€
    25mg
    178.00€
    50mg
    265.00€
    100mg
    383.00€
    1mL*10mM (DMSO)
    70.00€
  • TFLLR-NH2(TFA)

    CAS:
    TFLLR-NH2 (TFA) is a selective PAR1 agonist with an EC50 of 1.9 μM. EC50: 1.9 μM (PAR1)
    Formula:C33H54F3N9O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:761.83

    Ref: TM-TP1334

    1mg
    163.00€
    5mg
    640.00€
  • Apraclonidine hydrochloride

    CAS:
    Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.
    Formula:C9H11Cl3N4
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:281.57

    Ref: TM-T21371

    10mg
    49.00€
    25mg
    84.00€
    50mg
    110.00€
    100mg
    165.00€
    200mg
    224.00€
    1mL*10mM (DMSO)
    34.00€
  • L 888607

    CAS:
    L 888607 is an effective and selective CRTH2 agonist (Ki: 0.8 nM).
    Formula:C19H15ClFNO2S
    Color and Shape:Solid
    Molecular weight:375.84

    Ref: TM-T15828

    5mg
    284.00€
    1mL*10mM (DMSO)
    281.00€
  • Brombuterol hydrochloride

    CAS:
    Brombuterol is an agonist of the β2-adrenergic receptor (β2-AR).1It has been used as an illicit feed additive to increase the muscle-to-fat ratio of livestock.
    Formula:C12H19Br2ClN2O
    Color and Shape:Solid
    Molecular weight:402.56

    Ref: TM-T37848

    2mg
    350.00€
  • Vilazodone-d8

    CAS:
    Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial.
    Formula:C26H27N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:449.57

    Ref: TM-T13300

    1mg
    310.00€
    5mg
    To inquire
  • BMS-986020 sodium

    CAS:
    BMS-986020 sodium (AM152 sodium) is a high-affinity LPA1 antagonist for investigating idiopathic pulmonary fibrosis.
    Formula:C29H25N2NaO5
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:504.51

    Ref: TM-T63439

    1mg
    41.00€
    5mg
    To inquire
    10mg
    To inquire
    1mL*10mM (DMSO)
    151.00€
  • SB-408124 Hydrochloride

    CAS:
    SB-408124 Hydrochloride is a non-peptide OX1 receptor antagonist(Ki of 57 nM and 27 nM in both whole cell and membrane, respectively).
    Formula:C19H19ClF2N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.83

    Ref: TM-T12844

    2mg
    50.00€
    5mg
    73.00€
  • Ziprasidone D8

    CAS:
    Ziprasidone D8, deuterium-labeled, is a potent antipsychotic, antagonizing 5-HT and dopamine receptors.
    Formula:C21H21ClN4OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:420.99

    Ref: TM-T13400

    1mg
    767.00€
    5mg
    1,108.00€
    10mg
    1,513.00€
  • Timapiprant sodium

    CAS:
    Timapiprant sodium: potent DP2 antagonist; inhibits mast cell activation; displaces [3H]PGD2, Ki=3-13 nM.
    Formula:C21H17FN2NaO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:371.367

    Ref: TM-T17099

    2mg
    34.00€
    1mL*10mM (DMSO)
    67.00€
  • Thioridazine

    CAS:
    Thioridazine: an antipsychotic, anti-anxiety drug, blocks dopamine D2, PI3K-Akt-mTOR; halts angiogenesis, kills cancer cells, targets CSCs.
    Formula:C21H26N2S2
    Color and Shape:Solid
    Molecular weight:370.57

    Ref: TM-T61476

    1mg
    42.00€
    5mg
    67.00€
    10mg
    100.00€
    25mg
    159.00€
    50mg
    238.00€
    100mg
    360.00€
  • Quetiapine-d8 Fumarate

    CAS:
    Quetiapine-d8 Fumarate is a deuterated compound of Quetiapine Fumarate. Quetiapine Fumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.
    Formula:C25H21D8N3O6S
    Color and Shape:Solid
    Molecular weight:507.63

    Ref: TM-TMIJ-0315

    1mg
    To inquire
    5mg
    To inquire
  • PD176252

    CAS:
    PD176252 is a BB1 and BB2 antagonist, GRPR inhibitor, and FPR1/FPR2 agonist that inhibits the growth and proliferation of a wide range of cancer cells.
    Formula:C32H36N6O5
    Purity:99.00%
    Color and Shape:Solid
    Molecular weight:584.67

    Ref: TM-T16449

    1mg
    35.00€
    5mg
    67.00€
    10mg
    To inquire
    25mg
    To inquire
    1mL*10mM (DMSO)
    88.00€
  • Granisetron

    CAS:

    Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.

    Formula:C18H24N4O
    Color and Shape:Solid
    Molecular weight:312.41

    Ref: TM-T22340

    5mg
    922.00€
  • Olanzapine D3

    CAS:
    Olanzapine D3 is the deuterium labeled Olanzapine.
    Formula:C17H20N4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:315.45

    Ref: TM-T12291

    1mg
    268.00€
    5mg
    670.00€
    10mg
    888.00€
  • 5-HT3 antagonist 5

    CAS:
    5-HT3 antagonist 5, a quinoxalin-2-carboxamide, blocks 5-HT3 receptors and has antidepressant effects in mice.
    Formula:C16H13N3O2
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:279.29

    Ref: TM-T9846

    5mg
    49.00€
    10mg
    71.00€
    25mg
    129.00€
    50mg
    203.00€
    100mg
    290.00€
    200mg
    371.00€
    1mL*10mM (DMSO)
    50.00€
  • SKF-82958 hydrobromide

    CAS:
    SKF-82958 hydrobromide is a D1/D5 receptor full agonist.
    Formula:C19H21BrClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:410.73

    Ref: TM-T16892

    2mg
    73.00€
  • Aripiprazole (D8)

    CAS:
    Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).
    Formula:C23H27Cl2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:456.44

    Ref: TM-T10368

    1mg
    254.00€
    5mg
    632.00€