
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,999 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5960 products of "GPCR/G-Protein"
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Calcium-Sensing Receptor Antagonists I
CAS:Calcium-Sensing Receptor Antagonists I functions as an antagonist to the parathyroid hormone receptors that sense calcium.Formula:C23H24N2O2Color and Shape:SolidMolecular weight:360.45Travoprost (Standard)
CAS:Travoprost (Standard) is the standard substance of Travoprost, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Travoprost (Fluprostenol isopropyl ester) is used to treat glaucoma and ocular hypertension,is a potent and selective FP prostaglandin receptor agonist.Formula:C26H35F3O6Color and Shape:Colorless OilMolecular weight:500.55WAY-100635
CAS:WAY-100635 is a potent 5-HT 1A receptor antagonist pyramidal neuron firing frequency during conditioned reflexes; a dopamine D4 receptor agonist .Formula:C25H34N4O2Purity:98.972%Color and Shape:SolidMolecular weight:422.56TFLLR-NH2(TFA)
CAS:TFLLR-NH2 (TFA) is a selective PAR1 agonist with an EC50 of 1.9 μM. EC50: 1.9 μM (PAR1)Formula:C33H54F3N9O8Purity:98%Color and Shape:SolidMolecular weight:761.83Apraclonidine hydrochloride
CAS:Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.Formula:C9H11Cl3N4Purity:99.74%Color and Shape:SolidMolecular weight:281.57L 888607
CAS:L 888607 is an effective and selective CRTH2 agonist (Ki: 0.8 nM).Formula:C19H15ClFNO2SColor and Shape:SolidMolecular weight:375.84Brombuterol hydrochloride
CAS:Brombuterol is an agonist of the β2-adrenergic receptor (β2-AR).1It has been used as an illicit feed additive to increase the muscle-to-fat ratio of livestock.Formula:C12H19Br2ClN2OColor and Shape:SolidMolecular weight:402.56Vilazodone-d8
CAS:Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial.Formula:C26H27N5O2Purity:98%Color and Shape:SolidMolecular weight:449.57BMS-986020 sodium
CAS:BMS-986020 sodium (AM152 sodium) is a high-affinity LPA1 antagonist for investigating idiopathic pulmonary fibrosis.Formula:C29H25N2NaO5Purity:99.83%Color and Shape:SolidMolecular weight:504.51SB-408124 Hydrochloride
CAS:SB-408124 Hydrochloride is a non-peptide OX1 receptor antagonist(Ki of 57 nM and 27 nM in both whole cell and membrane, respectively).Formula:C19H19ClF2N4OPurity:98%Color and Shape:SolidMolecular weight:392.83Ziprasidone D8
CAS:Ziprasidone D8, deuterium-labeled, is a potent antipsychotic, antagonizing 5-HT and dopamine receptors.Formula:C21H21ClN4OSPurity:98%Color and Shape:SolidMolecular weight:420.99Timapiprant sodium
CAS:Timapiprant sodium: potent DP2 antagonist; inhibits mast cell activation; displaces [3H]PGD2, Ki=3-13 nM.Formula:C21H17FN2NaO2Purity:98%Color and Shape:SolidMolecular weight:371.367Thioridazine
CAS:Thioridazine: an antipsychotic, anti-anxiety drug, blocks dopamine D2, PI3K-Akt-mTOR; halts angiogenesis, kills cancer cells, targets CSCs.Formula:C21H26N2S2Color and Shape:SolidMolecular weight:370.57Quetiapine-d8 Fumarate
CAS:Quetiapine-d8 Fumarate is a deuterated compound of Quetiapine Fumarate. Quetiapine Fumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.Formula:C25H21D8N3O6SColor and Shape:SolidMolecular weight:507.63PD176252
CAS:PD176252 is a BB1 and BB2 antagonist, GRPR inhibitor, and FPR1/FPR2 agonist that inhibits the growth and proliferation of a wide range of cancer cells.Formula:C32H36N6O5Purity:99.00%Color and Shape:SolidMolecular weight:584.67Granisetron
CAS:Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.
Formula:C18H24N4OColor and Shape:SolidMolecular weight:312.41Olanzapine D3
CAS:Olanzapine D3 is the deuterium labeled Olanzapine.Formula:C17H20N4SPurity:98%Color and Shape:SolidMolecular weight:315.455-HT3 antagonist 5
CAS:5-HT3 antagonist 5, a quinoxalin-2-carboxamide, blocks 5-HT3 receptors and has antidepressant effects in mice.Formula:C16H13N3O2Purity:99.84%Color and Shape:SolidMolecular weight:279.29SKF-82958 hydrobromide
CAS:SKF-82958 hydrobromide is a D1/D5 receptor full agonist.Formula:C19H21BrClNO2Purity:98%Color and Shape:SolidMolecular weight:410.73Aripiprazole (D8)
CAS:Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).Formula:C23H27Cl2N3O2Purity:98%Color and Shape:SolidMolecular weight:456.44
