GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,994 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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SDZ WAG 994
CAS:SDZ WAG 994 is an A1 adenosine receptor agonist.Formula:C17H25N5O4Purity:99.82%Color and Shape:SolidMolecular weight:363.41Ref: TM-T23347
1mg63.00€5mg114.00€10mg172.00€25mg299.00€50mg432.00€100mg587.00€200mg792.00€1mL*10mM (DMSO)120.00€LY255283
CAS:LY255283 is a specific antagonit of leukotriene B4 (LTB4) receptor. It inhibits the production of LTB(4) in human PMNL and in monocytes.Formula:C19H28N4O3Purity:99.18%Color and Shape:SolidMolecular weight:360.45Ref: TM-T22946
2mg47.00€5mg88.00€10mg127.00€25mg250.00€50mg401.00€100mg645.00€200mg898.00€1mL*10mM (DMSO)87.00€Dynamin inhibitory peptide Acetate
Dynamin inhibitory peptide Acetate is a peptide with the sequence Gln-Val-Pro-Ser-Arg-Pro-Asn-Arg-Ala-Pro that inhibit the GTPase dynamin.Formula:C49H84N18O16Purity:97.28%Color and Shape:SolidMolecular weight:1181.3Ref: TM-T21798L
1mg73.00€5mg198.00€10mg294.00€25mg467.00€50mg642.00€100mg853.00€1mL*10mM (DMSO)474.00€Fexofenadine hydrochloride
CAS:Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the treatment of allergic rhinitis,Formula:C32H39NO4·HClPurity:99.39% - ≥95%Color and Shape:SolidMolecular weight:538.13Physalaemin acetate
Physalaemin acetate is a non-mammalian tachykinin with high affinity when binding selectively to neurokinin-1 (NK1) receptor.Formula:C60H88N14O18SPurity:99.13%Color and Shape:SolidMolecular weight:1325.49Tofogliflozin (hydrate)
CAS:Tofogliflozin hydrate (CSG-452 hydrate) is a potent and highly specific inhibitor of SGLT2(Ki of 2.9 nM, 14.9 nM, and 6.4 nM for human, rat, and mouse SGLT2).Formula:C22H28O7Purity:97.03% - 98.78%Color and Shape:SolidMolecular weight:404.45Ref: TM-T5016
1mg38.00€2mg52.00€5mg79.00€10mg115.00€25mg213.00€50mg341.00€100mg533.00€200mg757.00€1mL*10mM (DMSO)87.00€Triptorelin acetate(57773-63-4 free base)
CAS:Triptorelin acetate is a GnRH agonist for hormone-responsive cancers, precocious puberty, and assisted reproduction.Formula:C66H86N18O15Purity:99.59% - 99.90%Color and Shape:White PowderMolecular weight:1371.53Ref: TM-T21410
5mg52.00€10mg78.00€25mg119.00€50mg172.00€100mg259.00€200mg388.00€1mL*10mM (DMSO)116.00€Myristicin
CAS:Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.
Formula:C11H12O3Purity:99.828%Color and Shape:LiquidMolecular weight:192.21GR 94800 acetate
GR 94800 acetate is a potent and selective neurokinin 2(NK-2) antagonist.
Formula:C51H65N9O10Purity:97.86%Color and Shape:SolidMolecular weight:964.12Hypidone hydrochloride
CAS:Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitorFormula:C18H23ClN2O2Purity:99.82% - 99.93%Color and Shape:SolidMolecular weight:334.84Acrivastine
CAS:Acrivastine (Acrivastin) is a short-acting histamine 1 receptor antagonist.Formula:C22H24N2O2Purity:99.73% - >99.99%Color and Shape:SolidMolecular weight:348.44Protease-Activated Receptor-4 diTFA
Protease-Activated Receptor-4 diTFA,2454 is the proteinase-activated receptor-4 (PAR4)agonistFormula:C37H48F6N8O11Purity:98.54%Color and Shape:SolidMolecular weight:894.81Ref: TM-T7740
1mg48.00€2mg60.00€5mg86.00€10mg138.00€25mg274.00€50mg411.00€100mg607.00€1mL*10mM (DMSO)170.00€BML-190
CAS:BML-190 (Indomethacin morpholinylamide) 是一种 CB2 受体的配体，其对 CB2 受体 (Ki:435 nM) 和 CB1受体 (Ki> 2 μM)。Formula:C23H23ClN2O4Purity:97.70%Color and Shape:SolidMolecular weight:426.89(±)-Ibipinabant
CAS:(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.Formula:C23H20Cl2N4O2SPurity:99.28% - 99.83%Color and Shape:SolidMolecular weight:487.4Glucagon-like peptide 1 (1-37), human acetate
Glucagon-like peptide 1 (1-37), human acetate is a highly potent the GLP-1 receptor agonist.Purity:98%Color and Shape:LiquidMolecular weight:N/AOxyntomodulin acetate
Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].Purity:99.24%Color and Shape:LiquidMolecular weight:N/ABRL 54443
CAS:BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).Formula:C14H18N2OPurity:98.07%Color and Shape:SolidMolecular weight:230.31BIBO3304
CAS:BIBO3304: Selective NPY Y1 blocker, IC50 of 0.38nM (human), 0.72nM (rat); curbs hunger from NPY/fasting when injected centrally.Formula:C29H35N7O3Color and Shape:SolidMolecular weight:529.63Ufenamate
CAS:Ufenamate (Flufenamic acid butyl ester) is an anthranilic acid-based anti-inflammatory drug developed for skin diseasesFormula:C18H18F3NO2Purity:99.89%Color and Shape:SolidMolecular weight:337.34Pergolide mesylate
CAS:Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.Formula:C20H30N2O3S2Purity:99.70%Color and Shape:White To Off-White SolidMolecular weight:410.59
