GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,994 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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Zuclopenthixol
CAS:Zuclopenthixol (cis-Clopenthixol) is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics.Formula:C22H25ClN2OSPurity:98.9% - 99.82%Color and Shape:SolidMolecular weight:400.96CS 2100
CAS:CS 2100 (1-[[4-Ethyl-5-[5-(4-phenoxyphenyl)-1,2,4-oxadiazol-3-yl]-2-thienyl]methyl]-3-azetidinecarboxylic acid) is an S1P1 agonist.
Formula:C25H23N3O4SPurity:99.19%Color and Shape:SolidMolecular weight:461.53PAR-2 Activating Peptide acetate
PAR-2 Activating Peptide acetate (SLIGRL-NH2 acetate) is an agonist of Protease-Activated Receptor-2 (PAR-2).Formula:C31H60N10O9Purity:98.5% - 99.92%Color and Shape:SolidMolecular weight:716.88Pimavanserin tartrate
CAS:Pimavanserin tartrate is a potent 5-HT 2A receptor inverse agonist used to treat Parkinson's disease-related psychosis.Cost-effective and quality-assured.Formula:C50H68F2N6O4·C4H6O6Purity:99.24% - 99.98%Color and Shape:SolidMolecular weight:1005.2Gadolinium chloride
CAS:Gadolinium chloride is a calcium-sensing receptor (CaSR) agonistFormula:Cl3GdPurity:98%Color and Shape:White Crystalline SolidMolecular weight:263.61Propionylpromazine hydrochloride
CAS:Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist.Formula:C20H25ClN2OSPurity:99.17%Color and Shape:SolidMolecular weight:376.94H2L 5765834
CAS:H2L 5765834 is a lysophosphatidic acid receptors antagonistFormula:C21H12N2O7Purity:98.25% - 99.47%Color and Shape:SolidMolecular weight:404.33Ref: TM-T22834
1mg58.00€5mg113.00€10mg177.00€25mg334.00€50mg497.00€100mg708.00€1mL*10mM (DMSO)124.00€Ebastine
CAS:Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine.Formula:C32H39NO2Purity:99.65% - 99.99%Color and Shape:White To Off-White PowderMolecular weight:469.66NAV-2729
CAS:NAV-2729 inhibits six ArfGEFs (human ARNO, EFA6, BIG1, and BRAG2 and Legionella and Rickettsia RalF), the strongest effects being against BRAG2, Arf1 and Arf6.Formula:C25H17ClN4O3Purity:98.83% - 98.91%Color and Shape:SolidMolecular weight:456.88Ref: TM-T5142
2mg43.00€5mg63.00€10mg90.00€25mg193.00€50mg286.00€100mg429.00€500mg888.00€1mL*10mM (DMSO)71.00€Pasireotide Acetate
CAS:The pKi of Pasireotide (SOM230) acetate for sst1, 2, 3, 4, and 5 were 8.2, 9.0, 9.1, less than 7.0, and 9.9, respectively.Cost-effective and quality-assured.Formula:C60H70N10O11Purity:98.64% - 99.92%Color and Shape:SolidMolecular weight:1107.26Ref: TM-TP2207
1mg90.00€2mg138.00€5mg236.00€10mg409.00€25mg745.00€50mg1,189.00€100mg1,684.00€200mg2,268.00€9-FLUORENOL
CAS:9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.Formula:C13H10OPurity:99.98%Color and Shape:Off-White Crystalline PowderMolecular weight:182.22Pitolisant hydrochloride
CAS:Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).Formula:C17H27Cl2NOPurity:99.72% - 99.91%Color and Shape:SolidMolecular weight:332.31Ref: TM-T7176
5mg50.00€10mg74.00€25mg124.00€50mg197.00€100mg311.00€200mg467.00€500mg747.00€1mL*10mM (DMSO)52.00€5'-N-Ethylcarboxamidoadenosine
CAS:NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.Formula:C12H16N6O4Purity:98.95% - ≥95%Color and Shape:PowderMolecular weight:308.29Desvenlafaxine succinate hydrate
CAS:Desvenlafaxine succinate hydrate (WY 45233 Succinate) is an antidepressant of the serotonin-norepinephrine reuptake inhibitor (SNRI).Formula:C20H33NO7Purity:99.26%Color and Shape:White Crystalline PowdeMolecular weight:399.48Namodenoson
CAS:Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.Formula:C18H18ClIN6O4Purity:98.97%Color and Shape:SolidMolecular weight:544.73C14TKL-1 acetate
C14TKL-1 acetate is a NK1 receptor agonist.Formula:C65H102N20O15S2Purity:98.56%Color and Shape:SolidMolecular weight:1467.75Dapiprazole Hydrochloride
CAS:Dapiprazole Hydrochloride (Glamidolo Hydrochloride) is an alpha-1-adrenergic antagonist that acts by blocking alpha-adrenergic receptors.Formula:C19H28ClN5Purity:99.75% - 99.93%Color and Shape:SolidMolecular weight:361.92Azaphen
CAS:Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.Formula:C16H21Cl2N5OPurity:97.62%Color and Shape:SolidMolecular weight:370.28Dasotraline hydrochloride
CAS:Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.Formula:C16H16Cl3NPurity:98.92% - 99.6%Color and Shape:SolidMolecular weight:328.66Harmine hydrochloride
CAS:Harmine hydrochloride (telepathine hydrochloride) is extracted from Peganum Harmala Genus.Formula:C13H13ClN2OPurity:99.61% - >99.99%Color and Shape:Yellow To Slightly Green Crystalline PowderMolecular weight:248.71
