GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(3,031 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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Elagolix sodium
CAS:Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).Formula:C32H29F5N3NaO5Purity:99.71%Color and Shape:SolidMolecular weight:653.57Ref: TM-T5031
2mg35.00€5mg52.00€10mg80.00€25mg144.00€50mg227.00€100mg359.00€200mg532.00€1mL*10mM (DMSO)74.00€Bimatoprost
CAS:Bimatoprost (AGN 192024) is a cloprostenol-derived amide that is used as an antihypertensive agent in the treatment of open-angle glaucoma and ocularFormula:C25H37NO4Purity:98% - >99.99%Color and Shape:Crystalline SolidMolecular weight:415.57Ref: TM-T2538
2mg34.00€5mg48.00€10mg75.00€25mg127.00€50mg219.00€100mg371.00€200mg547.00€1mL*10mM (DMSO)50.00€Neuromedin N acetate(92169-45-4 free base)
Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinctFormula:C40H67N7O10Purity:99.95%Color and Shape:SolidMolecular weight:805.9Chlorphenoxamine
CAS:Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.Formula:C18H22ClNOPurity:99.44% - 99.85%Color and Shape:SolidMolecular weight:303.83Ref: TM-T7564
2mg35.00€5mg51.00€10mg81.00€25mg106.00€50mg147.00€100mg207.00€200mg306.00€1mL*10mM (DMSO)63.00€UFP 803 acetate
UFP 803 acetate is a potent ligand of urotensin-II (UT) receptor. UFP-803 displays the activity of a lower residual agonist.Formula:C52H68N10O14S2Purity:99.78%Color and Shape:SolidMolecular weight:1121.29Vorapaxar
CAS:Vorapaxar (MK-5348) (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).Formula:C29H33FN2O4Purity:98.77% - 99.93%Color and Shape:SolidMolecular weight:492.58Ref: TM-T7013
1mg74.00€5mg145.00€10mg202.00€25mg344.00€50mg472.00€100mg677.00€200mg937.00€1mL*10mM (DMSO)160.00€Octreotide Acetate
CAS:Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.Formula:C51H70N10O12S2Purity:99.03% - 99.87%Color and Shape:Less To Off-White Lyophilised Solid Colourless To Off-White Lyophilised SolidMolecular weight:1079.3Betahistine
CAS:Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.Formula:C8H12N2Purity:99.87% - 99.87%Color and Shape:Yellowish Liquid Liquid LiquidMolecular weight:136.19Sotagliflozin
CAS:Sotagliflozin (LP-802034) is an orally bioavailable inhibitor of the sodium-glucose co-transporter subtype 1 (SGLT1) and 2 (SGLT2), with potentialFormula:C21H25ClO5SPurity:99% - 99.86%Color and Shape:SolidMolecular weight:424.94Ref: TM-T3547
1mg46.00€2mg57.00€5mg87.00€10mg131.00€25mg248.00€50mg378.00€100mg560.00€500mg1,198.00€1mL*10mM (DMSO)88.00€M617 acetate
M617 acetate is a selective agonist of galanin receptor 1 (GAL1).Formula:C112H161N29O28Purity:96.02%Color and Shape:SolidMolecular weight:2361.65HS024
CAS:HS024 is a highly potent melanocortin MC4 receptor antagonist, increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats.Formula:C58H79N19O10S2Purity:>99.99%Color and Shape:SolidMolecular weight:1266.5SB-222200
CAS:SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).Formula:C26H24N2OPurity:97.13%Color and Shape:SolidMolecular weight:380.48Guanabenz Acetate
CAS:Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor.Formula:C8H8Cl2N4·C2H4O2Purity:99% - 99.66%Color and Shape:White Solid From Acetonitrile White SolidMolecular weight:291.13SKF38393 hydrobromide
CAS:SKF38393 hydrobromide is the salt form of SKF38393.a dopamine D1 receptor agonist that increases the expression of Shati/Nat8L mRNA in the NAc of mice;Formula:C16H18BrNO2Purity:98.99%Color and Shape:SolidMolecular weight:336.22m-Chlorophenylbiguanide hydrochloride
CAS:m-Chlorophenylbiguanide hydrochloride is a 5-HT3 receptor agonist.Formula:C8H11Cl2N5Purity:99.43% - 99.87%Color and Shape:SolidMolecular weight:248.11BQU57
CAS:BQU57 shows selective inhibition for Ral relative to Ras or Rho and inhibit xenograft tumor growth.Formula:C16H13F3N4OPurity:97.45% - 98.72%Color and Shape:SolidMolecular weight:334.3[D-Phe12]-Bombesin acetate
[D-Phe12]-Bombesin acetate inhibits bombesin-stimulated secretion.Formula:C76H116N22O20SPurity:99.81%Color and Shape:SolidMolecular weight:1689.94Tecadenoson
CAS:Tecadenoson (CVT-510) is a selective agonist of A1 adenosine receptor.
Formula:C14H19N5O5Purity:98.83%Color and Shape:SolidMolecular weight:337.33AZD1283
CAS:AZD1283 is an effective P2Y12 receptor antagonist (EC50: 3.0 ug/kg/min, binding IC50: 11 nM).Formula:C23H26N4O5SPurity:98.37% - 99.63%Color and Shape:SolidMolecular weight:470.542-Methoxyidazoxan monohydrochloride
CAS:L-Albizziin (2-Methoxyidazoxan monohydrochloride) is a highly potent selective antagonist of the alpha 2r adrenergic receptor.Formula:C12H14N2O3·HClPurity:98.99%Color and Shape:SolidMolecular weight:270.72
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