GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(55 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5985 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
RU 24969 free base
CAS:RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.
Formula:C14H16N2OPurity:97.38%Color and Shape:SolidMolecular weight:228.29Neuropeptide FF acetate(99566-27-5 free base)
Neuropeptide FF acetate(99566-27-5 free base) (NPFF acetate) is an octapeptide belonging to the RF amide family.Formula:C56H80N14O12Purity:98.03%Color and Shape:SolidMolecular weight:1141.32Conivaptan hydrochloride
CAS:Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia andFormula:C32H26N4O2·HClPurity:98.33% - 99.86%Color and Shape:SolidMolecular weight:535.04Ro 46-2005
CAS:Ro 46-2005: Synthetic non-peptide, blocks 125I-ET-1 at ETA receptors on human vascular cells (IC50: 220 nM).Formula:C23H27N3O6SPurity:98.02% - 98.8%Color and Shape:SolidMolecular weight:473.54SORT-PGRN interaction inhibitor 1
CAS:SORT-PGRN interaction inhibitor 1 is a potent sortilin-progranulin interaction inhibitor(IC50 of 2 μM).Formula:C15H18N2O2Purity:98.72%Color and Shape:SolidMolecular weight:258.32MDL 100009
CAS:MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is a selective antagonist of 5-HT2A.Formula:C22H28FNO3Purity:98.96%Color and Shape:SolidMolecular weight:373.46Ref: TM-T22359
1mg99.00€5mg187.00€10mg280.00€25mg434.00€50mg585.00€100mg775.00€200mg1,054.00€1mL*10mM (DMSO)222.00€Cotadutide acetate
Cotadutide acetate is a potent GLP-1 and glucagon receptor dual agonist with EC50s of 6.9 pM and 10.2 pM.Formula:C169H256N42O57Purity:98.28%Color and Shape:SolidMolecular weight:3788.14Bosentan
CAS:Bosentan is a competitive endothelin receptor antagonist, used for treating pulmonary arterial hypertension.Formula:C27H29N5O6SPurity:99.74% - 99.84%Color and Shape:Pale Yellow To Off-White SolidMolecular weight:551.614Ref: TM-T6264
10mg38.00€25mg56.00€50mg81.00€100mg127.00€200mg207.00€500mg310.00€1mL*10mM (DMSO)88.00€Neuropeptide SF(mouse,rat) acetate
Neuropeptide SF (mouse,rat) acetate is a NPFF receptor agonist with Ki of 48.4 nM (NPFF1) & 12.1 nM (NPFF2), enhancing ASIC3 current.Formula:C42H69N13O12Purity:98.37%Color and Shape:SolidMolecular weight:948.08CJC-1295 acetate(863288-34-0 free base)
CJC-1295 acetate is a synthetic GHRH analogue and GHS.Formula:C154H256N44O44Purity:97.29%Color and Shape:SolidMolecular weight:3428.01CP 376395
CAS:CP 376395 (CP-316311) is an effective and specific Corticotropin-releasing factor 1 (CRF1) receptor antagonist.Formula:C21H30N2OPurity:99.86% - 99.94%Color and Shape:SolidMolecular weight:326.48Substance P 1-9 aceate
Substance P 1-9 aceate is nonapeptide, which decreases the inactivation of substance P by the guinea-pig ileum and urinary bladder.Formula:C54H81N15O14Purity:99.01%Color and Shape:SolidMolecular weight:1164.31Protease-Activated Receptor-1, PAR-1 Agonist acetate
PAR-1 Agonist acetate is a selective PAR-1 agonist that mimics thrombin action.Formula:C37H62N10O11Purity:98.1800%Color and Shape:SolidMolecular weight:822.95Etilevodopa hydrochloride
CAS:Etilevodopa hydrochloride (L-DOPA ethyl ester) is a prodrug of levodopa. It also has greater gastric solubility and significant brain penetration.Formula:C11H16ClNO4Purity:95.00%Color and Shape:SolidMolecular weight:261.7Exendin-4
CAS:Exenatide: GLP-1 receptor agonist, 39-amino acid, longer half-life (2.4 hrs), IC50 of 3.22 nM.Formula:C184H282N50O60SPurity:97.71% - 99.78%Color and Shape:SolidMolecular weight:4186.57Bay 59-3074
CAS:Bay 59-3074 is a CB1/CB2 receptor partial agonist (Ki: 48.3/45.5 nM).
Formula:C18H13F6NO4SPurity:97.68% - 99.69%Color and Shape:SolidMolecular weight:453.36Galanin (1-16), mouse, porcine, rat
CAS:Galanin (1-16), mouse, porcine, rat is a hippocampal galanin receptor agonist(Kd = 3 nM) with high biological activity on locus coeruleus neurons.Formula:C78H116N20O21Purity:98.65%Color and Shape:White PowderMolecular weight:1669.88(+)-PD 128907 hydrochloride
CAS:(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .
Formula:C14H20ClNO3Purity:97.76%Color and Shape:SolidMolecular weight:285.77Montelukast sodium
CAS:Montelukast sodium (MK0476), an oral leukotriene antagonist for asthma, can cause rare liver injury.Formula:C35H35ClNNaO3SPurity:99.14% - 99.89%Color and Shape:White To Off-White Crystalline PowderMolecular weight:608.17RFRP3(human) acetate(311309-27-0 free base)
RFRP-3(human) acetate inhibits gonadotropin, blocks Ca2+ mobilization, acts on NPFF1 receptors, and has an IC50 of 0.7 nM against cAMP production.Formula:C47H76N14O12Purity:97.09%Color and Shape:SolidMolecular weight:1029.19
