GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(53 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5981 products of "GPCR/G-Protein"
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ICI 118,551 hydrochloride
CAS:ICI 118,551 hydrochloride (ICI 118551 hydrochloride) is a highly selective β2 adrenergic receptor antagonist (Kis: 0.7, 49.5, and 611 nM for β2, β1, and β3Formula:C17H28ClNO2Purity:99.296% - 99.76%Color and Shape:SolidMolecular weight:313.86A-836339
CAS:A-836339: Potent cannabinoid, CB2-focused (Ki=0.64nM), lesser CB1 affinity (Ki=270nM); analgesic, anti-inflammatory in mice.Formula:C16H26N2O2SPurity:99.94%Color and Shape:SolidMolecular weight:310.45Ref: TM-T7375
2mg35.00€5mg71.00€10mg115.00€25mg187.00€50mg274.00€100mg390.00€200mg527.00€1mL*10mM (DMSO)66.00€Bilastine
CAS:Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration ofFormula:C28H37N3O3Purity:99.86% - >99.99%Color and Shape:SolidMolecular weight:463.61ML 154
CAS:ML 154 is a potent neuropeptide S receptor (NPSR) antagonist.Formula:C29H26BrN2PSPurity:99.53%Color and Shape:SolidMolecular weight:545.47Pranlukast hemihydrate
CAS:Pranlukast hemihydrate (ONO-1078 hemihydrate) is an LT antagonist with anti-asthmatic activity.Formula:C27H23N5O40·5H2OPurity:99.28%Color and Shape:SolidMolecular weight:490.52MK 212 hydrochloride
CAS:MK 212 hydrochloride is a 5-HT2C receptor agonistFormula:C8H11ClN4·HClPurity:99.88%Color and Shape:SolidMolecular weight:235.12carfenazine
CAS:<p>carfenazine targets the Dopamine receptor and is used for schizophrenia research.</p>Formula:C24H31N3O2SPurity:98.06%Color and Shape:SolidMolecular weight:425.59Tianeptine
CAS:Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。Formula:C21H25ClN2O4SPurity:99.04%Color and Shape:SolidMolecular weight:436.95Alprenolol benzoate
CAS:Alprenolol benzoate is the benzoate salt of Alprenolol -- a beta blocker.Formula:C22H29NO4Color and Shape:SolidMolecular weight:371.48Adrenocorticotropic Hormone (ACTH) (4-10) TFA
Adrenocorticotropic Hormone (ACTH) (4-10) TFA (Acth (4-10)) is an agonist of potent melanocortin(MC4R) receptor .Formula:C46H60F3N13O12SPurity:98.49%Color and Shape:SolidMolecular weight:1076.12Ref: TM-T7627L
1mg57.00€2mg74.00€5mg97.00€10mg160.00€25mg341.00€50mg512.00€100mg653.00€200mg947.00€1mL*10mM (DMSO)213.00€Pramlintide acetate(151126-32-8 free base)
CAS:Pramlintide acetate is a polypeptide analogue of human amylin. It serves as an antidiabetic agent and exhibits antineoplastic activity in colorectal cancer.Formula:C173H271N51O55S2Purity:>99.99%Color and Shape:SolidMolecular weight:4009Tasimelteon
CAS:Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.Formula:C15H19NO2Purity:98.93% - 99.93%Color and Shape:SolidMolecular weight:245.32Melitracen
CAS:Melitracen is a tricyclic antidepressant.Formula:C21H25NColor and Shape:SolidMolecular weight:291.43[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate
Broad-spectrum neuropeptide inverse agonist/antagonist; potent at ghrelin receptor (EC50 = 5.2 nM); inhibits cancer growth, induces apoptosis.Formula:C81H113N19O14Purity:97.68%Color and Shape:SolidMolecular weight:1576.91Cloprostenol sodium salt
CAS:Cloprostenol sodium salt (ICI 80996 sodium salt) is a synthetic prostaglandin analogue, an agonist at the PGF2α receptor, with luteolytic properties.Formula:C22H28ClNaO6Purity:97.17% - 98.47%Color and Shape:White To Almost White Hygroscopic PowderMolecular weight:446.9Terazosin hydrochloride dihydrate
CAS:<p>Terazosin hydrochloride dihydrate (Heitrin dihydrate) is a selective α1-adrenoceptor antagonist, used for treatment of symptoms of an enlarged prostate (BPH).</p>Formula:C19H25N5O4·HCl·2H2OPurity:99.81%Color and Shape:White Or Off-White Crystalline PowderMolecular weight:459.92Ipsapirone hydrochloride
CAS:Ipsapirone, a pyrimidinylpiperazine ligand, is potent and specific for 5-HT1A receptors and has potential therapeutic use in affective disorders.Formula:C19H24ClN5O3SColor and Shape:SolidMolecular weight:437.94Zatebradine
CAS:Zatebradine is a potent hyperpolarization-activated cyclic nucleotide-gated (HCN) channels inhibitor(IC50 of 1.96 μM).Formula:C26H36N2O5Purity:98%Color and Shape:SolidMolecular weight:456.57Donitriptan Mesylate
CAS:Donitriptan Mesylate, a 5-HT1B/1D agonist, is used potentially for the treatment of migraines.Formula:C24H29N5O5SColor and Shape:SolidMolecular weight:499.58SSR240612
CAS:SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,Formula:C42H53ClN4O7SPurity:98.59% - 99.16%Color and Shape:SolidMolecular weight:793.41Ref: TM-T5048
1mg235.00€5mg540.00€10mg740.00€25mg1,035.00€50mg1,406.00€100mg1,882.00€1mL*10mM (DMSO)645.00€
![[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P acetate](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1931L1.webp&w=3840&q=75)
