GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5972 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Dobutamine tartrate
CAS:Dobutamine tartrate is a cardiotonic.Formula:C22H29NO9Color and Shape:SolidMolecular weight:451.472Tetradecyl Phosphonate
CAS:Tetradecyl Phosphonate 是溶血磷脂酸 1 (LPA1)、LPA2 和 LPA3 受体的泛拮抗剂。Formula:C14H31O3PPurity:99.95%Color and Shape:White To Off-White PowderMolecular weight:278.37Ambrisentan sodium
CAS:Ambrosentan (BSF 208075) sodium is a selective and oral effective antagonist of ET type A receptor ( ETAR ).Formula:C22H21N2NaO4Color and Shape:SolidMolecular weight:400.41BAR 501 impurity
CAS:BAR 501 impurity 在 BAR501 制剂中发现的一种杂质，可作为 G 蛋白偶联胆汁酸激活受体 (GP-BAR1) 的激动剂。 BAR501 杂质 (10 µM) 在 GP-BAR1 报告基因检测中诱导荧光素酶活性增加 150%。Formula:C26H46O3Purity:98.78%Color and Shape:SolidMolecular weight:406.64Carmoxirole (free base)
CAS:Carmoxirole: a dopamine D2 agonist, reduces pre-load/afterload, aids heart failure, lowers blood pressure by inhibiting noradrenaline release.Formula:C24H26N2O2Color and Shape:SolidMolecular weight:374.48Pizuglanstat
CAS:Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.Formula:C27H36N6O4Purity:99.62%Color and Shape:SolidMolecular weight:508.61Midodrine
CAS:Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.Formula:C12H18N2O4Purity:99.89%Color and Shape:SolidMolecular weight:254.28RTICBM-189
CAS:RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.Formula:C15H14Cl2N2OPurity:99.96%Color and Shape:SolidMolecular weight:309.19Ref: TM-T9466
2mg37.00€5mg50.00€10mg88.00€25mg170.00€50mg264.00€100mg389.00€200mg550.00€1mL*10mM (DMSO)71.00€MRT-10
CAS:<p>MRT-10 is a Smoothened (Smo) receptor antagonist.</p>Formula:C24H23N3O5SPurity:99.73%Color and Shape:SolidMolecular weight:465.52Sigma-LIGAND-1 hydrochloride
CAS:Sigma-LIGAND-1 HCl: selective sigma receptor ligand; DTG IC50: 16 nM, PPP IC50: 19 nM; weak D2 receptor affinity, Ki: 4000 nM.Formula:C27H34ClNO4Color and Shape:SolidMolecular weight:472.02Methyldopa hydrate
CAS:Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.Formula:C10H13NO4H2OPurity:99.67%Color and Shape:White SolidMolecular weight:238.24GRA Ex-25
CAS:<p>GRA Ex-25 (GRA-Ex-25) is an inhibitor of glucagon receptor.</p>Formula:C29H36F3N3O5Purity:98.2% - 98.88%Color and Shape:SolidMolecular weight:563.61Afamelanotide acetate
CAS:<p>Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist.</p>Formula:C80H115N21O21Purity:98% - 99.494%Color and Shape:SolidMolecular weight:1706.9Naftopidil hydrochloride
CAS:Naftopidil HCl (BM-15275) is a selective alpha1 blocker with Ki: α1a-3.7 nM, α1b-20 nM, α1d-1.2 nM; it also inhibits cell growth.Formula:C24H29ClN2O3Purity:99.5%Color and Shape:SolidMolecular weight:428.95Ref: TM-T9220
1mg44.00€5mg87.00€10mg117.00€25mg202.00€50mg304.00€100mg437.00€200mg612.00€1mL*10mM (DMSO)97.00€RS102895
CAS:<p>RS102895 is a potent CCR2 antagonist (IC50: 360 nM) and shows no effect on CCR1.</p>Formula:C21H21F3N2O2Purity:97.64% - 99.80%Color and Shape:SolidMolecular weight:390.4Hemopressin (human, mouse) acetate
Hemopressin: Nonapeptide, α1-hemoglobin derivative, CB1 inverse agonist, isolated from rats, oral, reduces inflammatory pain.Formula:C52H83N13O14Purity:99.86%Color and Shape:SolidMolecular weight:1114.29Calcitonin(salmon) Acetate(47931-85-1(free base))
Calcitonin(salmon)Acetate(47931-85-1(free base))(Salmon calcitonin) , a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5Formula:C145H240N44O48S2Purity:99.29%Color and Shape:SolidMolecular weight:3431.85Rizatriptan sulfate
CAS:Rizatriptan sulfate is a selective serotonin 5-HTID receptor agonist derived from tryptamine.Formula:C15H21N5O4SColor and Shape:SolidMolecular weight:367.42SAX-187
CAS:SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.Formula:C15H13ClN4O2S2Purity:97.82% - 98%Color and Shape:SolidMolecular weight:380.87Ref: TM-T3183
1mg84.00€5mg160.00€10mg259.00€25mg419.00€50mg562.00€100mg775.00€200mg1,026.00€1mL*10mM (DMSO)170.00€Volinanserin
CAS:Volinanserin (MDL100907) is a potent 5-HT2 receptor antagonist with a Ki of 0.36 nM, 300x selective over 5-HT1c, alpha-1, and sigma receptors.Formula:C22H28FNO3Purity:98.94% - 99.95%Color and Shape:SolidMolecular weight:373.46Ref: TM-T5389
1mg42.00€5mg88.00€10mg124.00€25mg233.00€50mg301.00€100mg393.00€200mg560.00€1mL*10mM (DMSO)96.00€
