GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5972 products of "GPCR/G-Protein"
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Eprazinone
CAS:Erazinone is a mucus dissolver and bronchospasm reliever.Formula:C24H32N2O2Color and Shape:SolidMolecular weight:380.52Orexin 2 Receptor Agonist
CAS:Orexin 2 Receptor Agonist (OX2R) is an effective (EC50: 23 nM) and OX2R-selective (OX1R/OX2R EC50 ratio: 70) agonist.Formula:C32H34N4O5SPurity:98.26% - 99.43%Color and Shape:SolidMolecular weight:586.7Ref: TM-T3177
2mg42.00€5mg64.00€10mg80.00€25mg137.00€50mg233.00€100mg340.00€200mg472.00€1mL*10mM (DMSO)81.00€Sotagliflozin
CAS:Sotagliflozin (LP-802034) is an orally bioavailable inhibitor of the sodium-glucose co-transporter subtype 1 (SGLT1) and 2 (SGLT2), with potentialFormula:C21H25ClO5SPurity:99% - 99.86%Color and Shape:SolidMolecular weight:424.94Ref: TM-T3547
1mg46.00€2mg57.00€5mg87.00€10mg131.00€25mg248.00€50mg378.00€100mg560.00€500mg1,198.00€1mL*10mM (DMSO)88.00€Haloperidol hydrochloride
CAS:Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist which is a potent antipsychotic agent.Formula:C21H24Cl2FNO2Color and Shape:SolidMolecular weight:412.33Lys-Bradykinin acetate(342-10-9 free base)
CAS:Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.Formula:C58H89N17O14Purity:99.86%Color and Shape:SolidMolecular weight:1248.43Flibanserin hydrochloride
CAS:Flibanserin HCl: oral 5-HT1A agonist & 5-HT2A antagonist, Ki values 1 nM & 49 nM, for HSDD, has antidepressant/anxiolytic properties.Formula:C20H22ClF3N4OColor and Shape:SolidMolecular weight:426.87Nuciferine
CAS:Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.Formula:C19H21NO2Purity:98.76% - 99.79%Color and Shape:SolidMolecular weight:295.38Atipamezole hydrochloride
CAS:<p>Atipamezole is a synthetic α2 adrenergic receptor antagonist.</p>Formula:C14H16N2·HClPurity:99.74%Color and Shape:SolidMolecular weight:248.75BMY-25368
CAS:BMY-25368 is a long-acting antagonist of the H2-receptor.Formula:C19H25N3O3Color and Shape:SolidMolecular weight:343.42Vortioxetine
CAS:Vortioxetine (Lu AA 21004) is a serotonergic antidepressant used for major depression disorders.Formula:C18H22N2SPurity:99.34% - 99.34%Color and Shape:SolidMolecular weight:298.45Ref: TM-T2395
1g505.00€10mg50.00€25mg69.00€50mg95.00€100mg124.00€200mg215.00€500mg350.00€1mL*10mM (DMSO)48.00€Dolasetron Mesylate hydrate
CAS:Dolasetron Mesylate hydrate blocks 5HT3 to prevent chemo and radiotherapy nausea.Formula:C20H26N2O7SPurity:99.86% - 99.99%Color and Shape:SolidMolecular weight:438.49MK-3697
CAS:<p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>Formula:C23H21N5O3SPurity:97.69% - 98.15%Color and Shape:SolidMolecular weight:447.51[Des-Arg9]-Bradykinin TFA
CAS:[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.Formula:C46H62F3N11O12Purity:>99.99%Color and Shape:SolidMolecular weight:1018.05Etelcalcetide hydrochloride
CAS:Etelcalcetide HCl, a synthetic peptide modulator of CaSR, lowers PTH in dialysis patients with secondary hyperparathyroidism.Formula:C38H73N21O10S2HClPurity:>99.99%Color and Shape:SolidMolecular weight:1353.33Praliciguat
CAS:Praliciguat (IW-1973) is an orally active sGC stimulator with a 197 nM EC50 in HEK-293 cells, enhances NO signaling, and is a vasodilator.Formula:C21H14F8N6O2Purity:98.82%Color and Shape:SolidMolecular weight:534.36Ref: TM-T16569
1mg150.00€2mg217.00€5mg368.00€10mg567.00€25mg905.00€50mg1,225.00€100mg1,644.00€1mL*10mM (DMSO)432.00€ML-193
CAS:ML-193: GPR55 antagonist, IC50 221nM, 27x selective over GPR35/CB1/CB2, may aid Parkinson's symptoms.Formula:C28H25N5O4SPurity:97.74%Color and Shape:SolidMolecular weight:527.59Betahistine
CAS:<p>Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.</p>Formula:C8H12N2Purity:99.87% - 99.87%Color and Shape:Yellowish Liquid Liquid LiquidMolecular weight:136.19SB756050
CAS:SB756050 is a specific TGR5 agonist.Formula:C21H28N2O8S2Purity:98.78% - >99.99%Color and Shape:SolidMolecular weight:500.59Cyclopiazonic acid
CAS:Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.Formula:C20H20N2O3Purity:99.27% - 99.80%Color and Shape:SolidMolecular weight:336.38SR 57227 hydrochloride
CAS:SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.Formula:C10H14ClN3·HClPurity:99.89%Color and Shape:SolidMolecular weight:248.15
![[Des-Arg9]-Bradykinin TFA](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT8809.webp&w=3840&q=75)
