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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5968 products of "GPCR/G-Protein"

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  • Landiolol hydrochloride

    CAS:
    Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.
    Formula:C25H40ClN3O8
    Purity:99.91%
    Color and Shape:White Crystalline Powder
    Molecular weight:546.05

    Ref: TM-T5028

    5mg
    35.00€
    10mg
    48.00€
    25mg
    80.00€
    50mg
    104.00€
    100mg
    144.00€
    200mg
    207.00€
    1mL*10mM (DMSO)
    52.00€
  • ML-191

    CAS:
    ML-191 is an inhibitor of LPI-induced phosphorylation of ERK1/2.
    Formula:C24H25N3O3
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:403.47

    Ref: TM-T22996

    5mg
    50.00€
    10mg
    77.00€
    25mg
    135.00€
    50mg
    212.00€
    100mg
    313.00€
    200mg
    442.00€
  • BETP

    CAS:
    BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).
    Formula:C20H17F3N2O2S
    Purity:98.51%
    Color and Shape:Solid
    Molecular weight:406.42

    Ref: TM-TQ0124

    1mg
    48.00€
    5mg
    93.00€
    10mg
    139.00€
    25mg
    264.00€
    50mg
    424.00€
    100mg
    677.00€
    1mL*10mM (DMSO)
    97.00€
  • 5-Benzyloxygramine

    CAS:
    5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.
    Formula:C18H20N2O
    Purity:99.13%
    Color and Shape:Solid
    Molecular weight:280.36

    Ref: TM-T35841

    100mg
    54.00€
  • Vilanterol trifenatate

    CAS:
    Vilanterol trifenatate is a long-acting agonist of β2-adrenoceptor (β2-AR) with inherent 24-hour activity(β2-AR, β1-AR and β3-AR pEC50s of 10.37, 6.98 and 7.36, respectively)
    Formula:C44H49Cl2NO7
    Purity:99.51% - >99.99%
    Color and Shape:Solid
    Molecular weight:774.77

    Ref: TM-T5134

    1mg
    37.00€
    5mg
    93.00€
    10mg
    124.00€
    25mg
    219.00€
    50mg
    350.00€
    100mg
    505.00€
    1mL*10mM (DMSO)
    106.00€
  • Fluparoxan HCl

    CAS:
    Fluparoxan is a potent α2-adrenergic receptor antagonist (pKB = 7.9) with excellent α2/α1 selectivity (2630 fold).
    Formula:C10H11ClFNO2
    Color and Shape:Solid
    Molecular weight:231.65

    Ref: TM-T27340

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Opaganib

    CAS:
    Opaganib (ABC294640) is an orally active and specific sphingosine kinase-2 (SphK2) inhibitor (IC50: 60 μM).
    Formula:C23H25ClN2O
    Purity:98.86% - 99.85%
    Color and Shape:Solid
    Molecular weight:380.91

    Ref: TM-T6750

    1mg
    40.00€
    2mg
    52.00€
    5mg
    85.00€
    10mg
    124.00€
    25mg
    240.00€
    50mg
    415.00€
    100mg
    615.00€
    1mL*10mM (DMSO)
    87.00€
  • Namodenoson

    CAS:
    Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.
    Formula:C18H18ClIN6O4
    Purity:98.97%
    Color and Shape:Solid
    Molecular weight:544.73

    Ref: TM-T6884

    1mg
    37.00€
    5mg
    79.00€
    10mg
    119.00€
    25mg
    235.00€
    50mg
    378.00€
    100mg
    567.00€
    1mL*10mM (DMSO)
    95.00€
  • Loxiglumide

    CAS:
    <p>Loxiglumide (CR-1505) is an antagonist of cholecystokinin (CCK-1) receptor.</p>
    Formula:C21H30Cl2N2O5
    Purity:97.55% - 99.81%
    Color and Shape:Solid
    Molecular weight:461.38

    Ref: TM-T2312

    10mg
    40.00€
    25mg
    78.00€
    50mg
    123.00€
    100mg
    202.00€
    200mg
    346.00€
  • Sonepiprazole mesylate

    CAS:
    Sonepiprazole mesylate is a selective D4 antagonist
    Formula:C22H31N3O6S2
    Color and Shape:Solid
    Molecular weight:497.63

    Ref: TM-T28828

    25mg
    1,586.00€
    50mg
    2,072.00€
    100mg
    2,660.00€
  • BMS-813160

    CAS:
    BMS-813160 is the first dual CCR2/CCR5 antagonist to enter Clinical development for cardiovascular.
    Formula:C25H40N8O2
    Purity:99.66% - 99.79%
    Color and Shape:Solid
    Molecular weight:484.64

    Ref: TM-T4584

    1mg
    63.00€
    5mg
    137.00€
    10mg
    187.00€
    25mg
    341.00€
    50mg
    567.00€
    100mg
    810.00€
    500mg
    1,644.00€
    1mL*10mM (DMSO)
    145.00€
  • BMY 7378 dihydrochloride

    CAS:
    BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.
    Formula:C22H33Cl2N3O3
    Purity:97.32% - 99.08%
    Color and Shape:Solid
    Molecular weight:458.42

    Ref: TM-T3046

    10mg
    48.00€
    25mg
    85.00€
    50mg
    101.00€
    1mL*10mM (DMSO)
    35.00€
  • Ursodeoxycholic acid sodium

    CAS:
    <p>Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities.</p>
    Formula:C24H40NaO4
    Purity:99.66% - 99.96%
    Color and Shape:Solid
    Molecular weight:415.56

    Ref: TM-T29078

    100mg
    34.00€
  • FK962

    CAS:
    FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.
    Formula:C14H17FN2O2
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:264.3

    Ref: TM-T7829

    2mg
    37.00€
    5mg
    56.00€
    10mg
    87.00€
    25mg
    153.00€
    50mg
    212.00€
    100mg
    293.00€
    200mg
    411.00€
    1mL*10mM (DMSO)
    60.00€
  • Pipamperone HCl

    CAS:
    Pipamperone blocks 5-HT2A/B/C, D2/D3/D4, α1/α2 receptors; favors 5-HT2A/D4 over D2; negligible affinity for H1, mACh. Highly selective at low doses.
    Formula:C21H31ClFN3O2
    Color and Shape:Solid
    Molecular weight:411.95

    Ref: TM-T28417

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • (E)-3,4,5-Trimethoxycinnamic acid

    CAS:
    (E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.
    Formula:C12H14O5
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:238.24

    Ref: TM-TN2865

    1g
    133.00€
    100mg
    48.00€
    500mg
    90.00€
    1mL*10mM (DMSO)
    35.00€
  • Arformoterol Tartrate

    CAS:
    Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.
    Formula:C23H30N2O10
    Purity:99.98%
    Color and Shape:Solid
    Molecular weight:494.49

    Ref: TM-T22245

    5mg
    60.00€
    10mg
    87.00€
    25mg
    150.00€
    50mg
    221.00€
    100mg
    329.00€
    200mg
    487.00€
    1mL*10mM (DMSO)
    85.00€
  • Metoclopramide dihydrochloride

    CAS:
    Metoclopramide dihydrochloride is a dopamine D2 antagonist that is used as an antiemetic.
    Formula:C14H24Cl3N3O2
    Color and Shape:Solid
    Molecular weight:372.72

    Ref: TM-T69575

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Eptapirone

    CAS:
    Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.
    Formula:C16H23N7O2
    Purity:99.39% - 99.65%
    Color and Shape:Solid
    Molecular weight:345.4

    Ref: TM-T3179

    10mg
    52.00€
    25mg
    90.00€
    50mg
    145.00€
    100mg
    210.00€
    200mg
    304.00€
    1mL*10mM (DMSO)
    35.00€
  • N-Acetylhistamine acetate


    N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.
    Formula:C9H15N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:213.23

    Ref: TM-T19443L

    5mg
    55.00€