
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(13 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5968 products of "GPCR/G-Protein"
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Landiolol hydrochloride
CAS:Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.Formula:C25H40ClN3O8Purity:99.91%Color and Shape:White Crystalline PowderMolecular weight:546.05ML-191
CAS:ML-191 is an inhibitor of LPI-induced phosphorylation of ERK1/2.Formula:C24H25N3O3Purity:99.58%Color and Shape:SolidMolecular weight:403.47BETP
CAS:BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).Formula:C20H17F3N2O2SPurity:98.51%Color and Shape:SolidMolecular weight:406.425-Benzyloxygramine
CAS:5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.Formula:C18H20N2OPurity:99.13%Color and Shape:SolidMolecular weight:280.36Vilanterol trifenatate
CAS:Vilanterol trifenatate is a long-acting agonist of β2-adrenoceptor (β2-AR) with inherent 24-hour activity(β2-AR, β1-AR and β3-AR pEC50s of 10.37, 6.98 and 7.36, respectively)Formula:C44H49Cl2NO7Purity:99.51% - >99.99%Color and Shape:SolidMolecular weight:774.77Fluparoxan HCl
CAS:Fluparoxan is a potent α2-adrenergic receptor antagonist (pKB = 7.9) with excellent α2/α1 selectivity (2630 fold).Formula:C10H11ClFNO2Color and Shape:SolidMolecular weight:231.65Opaganib
CAS:Opaganib (ABC294640) is an orally active and specific sphingosine kinase-2 (SphK2) inhibitor (IC50: 60 μM).Formula:C23H25ClN2OPurity:98.86% - 99.85%Color and Shape:SolidMolecular weight:380.91Ref: TM-T6750
1mg40.00€2mg52.00€5mg85.00€10mg124.00€25mg240.00€50mg415.00€100mg615.00€1mL*10mM (DMSO)87.00€Namodenoson
CAS:Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.Formula:C18H18ClIN6O4Purity:98.97%Color and Shape:SolidMolecular weight:544.73Loxiglumide
CAS:<p>Loxiglumide (CR-1505) is an antagonist of cholecystokinin (CCK-1) receptor.</p>Formula:C21H30Cl2N2O5Purity:97.55% - 99.81%Color and Shape:SolidMolecular weight:461.38Sonepiprazole mesylate
CAS:Sonepiprazole mesylate is a selective D4 antagonistFormula:C22H31N3O6S2Color and Shape:SolidMolecular weight:497.63BMS-813160
CAS:BMS-813160 is the first dual CCR2/CCR5 antagonist to enter Clinical development for cardiovascular.Formula:C25H40N8O2Purity:99.66% - 99.79%Color and Shape:SolidMolecular weight:484.64Ref: TM-T4584
1mg63.00€5mg137.00€10mg187.00€25mg341.00€50mg567.00€100mg810.00€500mg1,644.00€1mL*10mM (DMSO)145.00€BMY 7378 dihydrochloride
CAS:BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.Formula:C22H33Cl2N3O3Purity:97.32% - 99.08%Color and Shape:SolidMolecular weight:458.42Ursodeoxycholic acid sodium
CAS:<p>Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities.</p>Formula:C24H40NaO4Purity:99.66% - 99.96%Color and Shape:SolidMolecular weight:415.56FK962
CAS:FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.Formula:C14H17FN2O2Purity:99.89%Color and Shape:SolidMolecular weight:264.3Ref: TM-T7829
2mg37.00€5mg56.00€10mg87.00€25mg153.00€50mg212.00€100mg293.00€200mg411.00€1mL*10mM (DMSO)60.00€Pipamperone HCl
CAS:Pipamperone blocks 5-HT2A/B/C, D2/D3/D4, α1/α2 receptors; favors 5-HT2A/D4 over D2; negligible affinity for H1, mACh. Highly selective at low doses.Formula:C21H31ClFN3O2Color and Shape:SolidMolecular weight:411.95(E)-3,4,5-Trimethoxycinnamic acid
CAS:(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.Formula:C12H14O5Purity:99.83%Color and Shape:SolidMolecular weight:238.24Arformoterol Tartrate
CAS:Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.Formula:C23H30N2O10Purity:99.98%Color and Shape:SolidMolecular weight:494.49Ref: TM-T22245
5mg60.00€10mg87.00€25mg150.00€50mg221.00€100mg329.00€200mg487.00€1mL*10mM (DMSO)85.00€Metoclopramide dihydrochloride
CAS:Metoclopramide dihydrochloride is a dopamine D2 antagonist that is used as an antiemetic.Formula:C14H24Cl3N3O2Color and Shape:SolidMolecular weight:372.72Eptapirone
CAS:Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.Formula:C16H23N7O2Purity:99.39% - 99.65%Color and Shape:SolidMolecular weight:345.4N-Acetylhistamine acetate
N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.Formula:C9H15N3O3Purity:98%Color and Shape:SolidMolecular weight:213.23
